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Piperazine and piperidine carboxamides and carbamates as inhibitors of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL). [electronic resource] by
- Korhonen, Jani
- Kuusisto, Anne
- van Bruchem, John
- Patel, Jayendra Z
- Laitinen, Tuomo
- Navia-Paldanius, Dina
- Laitinen, Jarmo T
- Savinainen, Juha R
- Parkkari, Teija
- Nevalainen, Tapio J
Producer: 20151005
In:
Bioorganic & medicinal chemistry vol. 22
Availability: No items available.
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7.
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Evaluation of FASN inhibitors by a versatile toolkit reveals differences in pharmacology between human and rodent FASN preparations and in antiproliferative efficacy in vitro vs. in situ in human cancer cells. [electronic resource] by
- Singha, Prosanta K
- Mäklin, Kiira
- Vihavainen, Taina
- Laitinen, Tuomo
- Nevalainen, Tapio J
- Patil, Mahadeo R
- Tonduru, Arun K
- Poso, Antti
- Laitinen, Jarmo T
- Savinainen, Juha R
Publication details: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences Apr 2020
In:
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences vol. 149
Availability: No items available.
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8.
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Design, synthesis, and biological evaluation of 2,4-dihydropyrano[2,3-c]pyrazole derivatives as autotaxin inhibitors. [electronic resource] by
- Pantsar, Tatu
- Singha, Prosanta
- Nevalainen, Tapio J
- Koshevoy, Igor
- Leppänen, Jukka
- Poso, Antti
- Niskanen, Juha M A
- Pasonen-Seppänen, Sanna
- Savinainen, Juha R
- Laitinen, Tuomo
- Laitinen, Jarmo T
Producer: 20180515
In:
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences vol. 107
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Chemoproteomic, biochemical and pharmacological approaches in the discovery of inhibitors targeting human α/β-hydrolase domain containing 11 (ABHD11). [electronic resource] by
- Navia-Paldanius, Dina
- Patel, Jayendra Z
- López Navarro, Miriam
- Jakupović, Hermina
- Goffart, Steffi
- Pasonen-Seppänen, Sanna
- Nevalainen, Tapio J
- Jääskeläinen, Tiina
- Laitinen, Tuomo
- Laitinen, Jarmo T
- Savinainen, Juha R
Producer: 20170417
In:
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences vol. 93
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Synthesis, in vitro and in vivo evaluation of 1,3,5-triazines as cannabinoid CB2 receptor agonists. [electronic resource] by
- Yrjölä, Sari
- Sarparanta, Mirkka
- Airaksinen, Anu J
- Hytti, Maria
- Kauppinen, Anu
- Pasonen-Seppänen, Sanna
- Adinolfi, Barbara
- Nieri, Paola
- Manera, Clementina
- Keinänen, Outi
- Poso, Antti
- Nevalainen, Tapio J
- Parkkari, Teija
Producer: 20150831
In:
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences vol. 67
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11.
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Loratadine analogues as MAGL inhibitors. [electronic resource] by
- Patel, Jayendra Z
- Ahenkorah, Stephen
- Vaara, Miia
- Staszewski, Marek
- Adams, Yahaya
- Laitinen, Tuomo
- Navia-Paldanius, Dina
- Parkkari, Teija
- Savinainen, Juha R
- Walczyński, Krzysztof
- Laitinen, Jarmo T
- Nevalainen, Tapio J
Producer: 20151221
In:
Bioorganic & medicinal chemistry letters vol. 25
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Potent and selective N-(4-sulfamoylphenyl)thiourea-based GPR55 agonists. [electronic resource] by
- Yrjölä, Sari
- Parkkari, Teija
- Navia-Paldanius, Dina
- Laitinen, Tuomo
- Kaczor, Agnieszka A
- Kokkola, Tarja
- Adusei-Mensah, Frank
- Savinainen, Juha R
- Laitinen, Jarmo T
- Poso, Antti
- Alexander, Amy
- Penman, June
- Stott, Lisa
- Anskat, Marie
- Irving, Andrew J
- Nevalainen, Tapio J
Producer: 20160920
In:
European journal of medicinal chemistry vol. 107
Availability: No items available.
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13.
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Optimization of 1,2,5-thiadiazole carbamates as potent and selective ABHD6 inhibitors. [electronic resource] by
- Patel, Jayendra Z
- Nevalainen, Tapio J
- Savinainen, Juha R
- Adams, Yahaya
- Laitinen, Tuomo
- Runyon, Robert S
- Vaara, Miia
- Ahenkorah, Stephen
- Kaczor, Agnieszka A
- Navia-Paldanius, Dina
- Gynther, Mikko
- Aaltonen, Niina
- Joharapurkar, Amit A
- Jain, Mukul R
- Haka, Abigail S
- Maxfield, Frederick R
- Laitinen, Jarmo T
- Parkkari, Teija
Producer: 20150929
In:
ChemMedChem vol. 10
Availability: No items available.
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