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Synthesis and pharmacological activity of angiotensin converting enzyme inhibitors: N-(mercaptoacyl)-4-substituted-(S)-prolines. [electronic resource] by
- Smith, E M
- Swiss, G F
- Neustadt, B R
- Gold, E H
- Sommer, J A
- Brown, A D
- Chiu, P J
- Moran, R
- Sybertz, E J
- Baum, T
Producer: 19880510
In:
Journal of medicinal chemistry vol. 31
Availability: No items available.
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Piperazine-based CCR5 antagonists as HIV-1 inhibitors. II. Discovery of 1-[(2,4-dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoromethyl)phenyl]ethyl]-1-piperazinyl]- piperidine N1-oxide (Sch-350634), an orally bioavailable, potent CCR5 antagonist. [electronic resource] by
- Tagat, J R
- Steensma, R W
- McCombie, S W
- Nazareno, D V
- Lin, S I
- Neustadt, B R
- Cox, K
- Xu, S
- Wojcik, L
- Murray, M G
- Vantuno, N
- Baroudy, B M
- Strizki, J M
Producer: 20011204
In:
Journal of medicinal chemistry vol. 44
Availability: No items available.
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