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CYP-dependent metabolism of antitumor pyrazolo[3,4-d]pyrimidine derivatives is characterized by an oxidative dechlorination reaction. [electronic resource] by
- Zamperini, Claudio
- Dreassi, Elena
- Vignaroli, Giulia
- Radi, Marco
- Dragoni, Stefania
- Schenone, Silvia
- Musumeci, Francesca
- Valoti, Massimo
- Antiochia, Riccarda
- Botta, Maurizio
Producer: 20151026
In:
Drug metabolism and pharmacokinetics vol. 29
Availability: No items available.
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The small molecule SI113 hinders epithelial-to-mesenchymal transition and subverts cytoskeletal organization in human cancer cells. [electronic resource] by
- Abbruzzese, Claudia
- Matteoni, Silvia
- Persico, Michele
- Ascione, Barbara
- Schenone, Silvia
- Musumeci, Francesca
- Amato, Rosario
- Perrotti, Nicola
- Matarrese, Paola
- Paggi, Marco G
Producer: 20200622
In:
Journal of cellular physiology vol. 234
Availability: No items available.
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16.
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A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: from in silico screening to cyclodextrin formulation. [electronic resource] by
- Radi, Marco
- Evensen, Lasse
- Dreassi, Elena
- Zamperini, Claudio
- Caporicci, Marialessandra
- Falchi, Federico
- Musumeci, Francesca
- Schenone, Silvia
- Lorens, James B
- Botta, Maurizio
Producer: 20130107
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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17.
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Matrine in association with FD‑2 stimulates F508del‑cystic fibrosis transmembrane conductance regulator activity in the presence of corrector VX809. [electronic resource] by
- Marengo, Barbara
- Speciale, Andrea
- Senatore, Lisa
- Garibaldi, Silvano
- Musumeci, Francesca
- Nieddu, Erika
- Pollarolo, Benedetta
- Pronzato, Maria Adelaide
- Schenone, Silvia
- Mazzei, Mauro
- Domenicotti, Cinzia
Producer: 20180626
In:
Molecular medicine reports vol. 16
Availability: No items available.
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18.
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Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma. [electronic resource] by
- Musumeci, Francesca
- Fallacara, Anna Lucia
- Brullo, Chiara
- Grossi, Giancarlo
- Botta, Lorenzo
- Calandro, Pierpaolo
- Chiariello, Mario
- Kissova, Miroslava
- Crespan, Emmanuele
- Maga, Giovanni
- Schenone, Silvia
Producer: 20170228
In:
European journal of medicinal chemistry vol. 127
Availability: No items available.
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Substituted pyrazolo[3,4-b]pyridines as human A1 adenosine antagonists: developments in understanding the receptor stereoselectivity. [electronic resource] by
- Tuccinardi, Tiziano
- Zizzari, Alessandra Tania
- Brullo, Chiara
- Daniele, Simona
- Musumeci, Francesca
- Schenone, Silvia
- Trincavelli, Maria Letizia
- Martini, Claudia
- Martinelli, Adriano
- Giorgi, Gianluca
- Botta, Maurizio
Producer: 20120316
In:
Organic & biomolecular chemistry vol. 9
Availability: No items available.
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20.
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Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors. [electronic resource] by
- Vignaroli, Giulia
- Zamperini, Claudio
- Dreassi, Elena
- Radi, Marco
- Angelucci, Adriano
- Sanità, Patrizia
- Crespan, Emmanuele
- Kissova, Miroslava
- Maga, Giovanni
- Schenone, Silvia
- Musumeci, Francesca
- Botta, Maurizio
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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