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Structure-based design and synthesis of pyrrole derivatives as MEK inhibitors. [electronic resource] by
- Wallace, Michael B
- Adams, Mark E
- Kanouni, Toufike
- Mol, Clifford D
- Dougan, Douglas R
- Feher, Victoria A
- O'Connell, Shawn M
- Shi, Lihong
- Halkowycz, Petro
- Dong, Qing
Producer: 20101207
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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Structure of a c-kit product complex reveals the basis for kinase transactivation. [electronic resource] by
- Mol, Clifford D
- Lim, Kheng B
- Sridhar, Vandana
- Zou, Hua
- Chien, Ellen Y T
- Sang, Bi-Ching
- Nowakowski, Jacek
- Kassel, Daniel B
- Cronin, Ciarán N
- McRee, Duncan E
Producer: 20031029
In:
The Journal of biological chemistry vol. 278
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Structural basis for the autoinhibition and STI-571 inhibition of c-Kit tyrosine kinase. [electronic resource] by
- Mol, Clifford D
- Dougan, Douglas R
- Schneider, Thomas R
- Skene, Robert J
- Kraus, Michelle L
- Scheibe, Daniel N
- Snell, Gyorgy P
- Zou, Hua
- Sang, Bi-Ching
- Wilson, Keith P
Producer: 20040921
In:
The Journal of biological chemistry vol. 279
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8.
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Design, synthesis and structure-activity relationships of 1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3beta. [electronic resource] by
- Saitoh, Morihisa
- Kunitomo, Jun
- Kimura, Eiji
- Hayase, Yoji
- Kobayashi, Hiromi
- Uchiyama, Noriko
- Kawamoto, Tomohiro
- Tanaka, Toshimasa
- Mol, Clifford D
- Dougan, Douglas R
- Textor, Garret S
- Snell, Gyorgy P
- Itoh, Fumio
Producer: 20090529
In:
Bioorganic & medicinal chemistry vol. 17
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Design, stereoselective synthesis, and biological evaluation of novel tri-cyclic compounds as inhibitor of apoptosis proteins (IAP) antagonists. [electronic resource] by
- Asano, Moriteru
- Hashimoto, Kentaro
- Saito, Bunnai
- Shiokawa, Zenyu
- Sumi, Hiroyuki
- Yabuki, Masato
- Yoshimatsu, Mie
- Aoyama, Kazunobu
- Hamada, Teruki
- Morishita, Nao
- Dougan, Douglas R
- Mol, Clifford D
- Yoshida, Sei
- Ishikawa, Tomoyasu
Producer: 20140326
In:
Bioorganic & medicinal chemistry vol. 21
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2-{3-[4-(Alkylsulfinyl)phenyl]-1-benzofuran-5-yl}-5-methyl-1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3beta with good brain permeability. [electronic resource] by
- Saitoh, Morihisa
- Kunitomo, Jun
- Kimura, Eiji
- Iwashita, Hiroki
- Uno, Yumiko
- Onishi, Tomohiro
- Uchiyama, Noriko
- Kawamoto, Tomohiro
- Tanaka, Toshimasa
- Mol, Clifford D
- Dougan, Douglas R
- Textor, Garret P
- Snell, Gyorgy P
- Takizawa, Masayuki
- Itoh, Fumio
- Kori, Masakuni
Producer: 20091124
In:
Journal of medicinal chemistry vol. 52
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Design, synthesis, and structure-activity relationships of spirolactones bearing 2-ureidobenzothiophene as acetyl-CoA carboxylases inhibitors. [electronic resource] by
- Yamashita, Tohru
- Kamata, Makoto
- Endo, Satoshi
- Yamamoto, Mitsuo
- Kakegawa, Keiko
- Watanabe, Hiroyuki
- Miwa, Katsuhiko
- Yamano, Toru
- Funata, Masaaki
- Sakamoto, Jyun-Ichi
- Tani, Akiyoshi
- Mol, Clifford D
- Zou, Hua
- Dougan, Douglas R
- Sang, Biching
- Snell, Gyorgy
- Fukatsu, Kohji
Producer: 20120131
In:
Bioorganic & medicinal chemistry letters vol. 21
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Structures of the CXCR4 chemokine GPCR with small-molecule and cyclic peptide antagonists. [electronic resource] by
- Wu, Beili
- Chien, Ellen Y T
- Mol, Clifford D
- Fenalti, Gustavo
- Liu, Wei
- Katritch, Vsevolod
- Abagyan, Ruben
- Brooun, Alexei
- Wells, Peter
- Bi, F Christopher
- Hamel, Damon J
- Kuhn, Peter
- Handel, Tracy M
- Cherezov, Vadim
- Stevens, Raymond C
Producer: 20101214
In:
Science (New York, N.Y.) vol. 330
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Conserved structural chemistry for incision activity in structurally non-homologous apurinic/apyrimidinic endonuclease APE1 and endonuclease IV DNA repair enzymes. [electronic resource] by
- Tsutakawa, Susan E
- Shin, David S
- Mol, Clifford D
- Izumi, Tadahide
- Arvai, Andrew S
- Mantha, Anil K
- Szczesny, Bartosz
- Ivanov, Ivaylo N
- Hosfield, David J
- Maiti, Buddhadev
- Pique, Mike E
- Frankel, Kenneth A
- Hitomi, Kenichi
- Cunningham, Richard P
- Mitra, Sankar
- Tainer, John A
Producer: 20130515
In:
The Journal of biological chemistry vol. 288
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A new class of non-thiazolidinedione, non-carboxylic-acid-based highly selective peroxisome proliferator-activated receptor (PPAR) γ agonists: design and synthesis of benzylpyrazole acylsulfonamides. [electronic resource] by
- Rikimaru, Kentaro
- Wakabayashi, Takeshi
- Abe, Hidenori
- Imoto, Hiroshi
- Maekawa, Tsuyoshi
- Ujikawa, Osamu
- Murase, Katsuhito
- Matsuo, Takanori
- Matsumoto, Mitsuharu
- Nomura, Chisako
- Tsuge, Hiroko
- Arimura, Naoto
- Kawakami, Kazutoshi
- Sakamoto, Junichi
- Funami, Miyuki
- Mol, Clifford D
- Snell, Gyorgy P
- Bragstad, Kenneth A
- Sang, Bi-Ching
- Dougan, Douglas R
- Tanaka, Toshimasa
- Katayama, Nozomi
- Horiguchi, Yoshiaki
- Momose, Yu
Producer: 20120511
In:
Bioorganic & medicinal chemistry vol. 20
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15.
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Structure-activity relationships and key structural feature of pyridyloxybenzene-acylsulfonamides as new, potent, and selective peroxisome proliferator-activated receptor (PPAR) γ Agonists. [electronic resource] by
- Rikimaru, Kentaro
- Wakabayashi, Takeshi
- Abe, Hidenori
- Tawaraishi, Taisuke
- Imoto, Hiroshi
- Yonemori, Jinichi
- Hirose, Hideki
- Murase, Katsuhito
- Matsuo, Takanori
- Matsumoto, Mitsuharu
- Nomura, Chisako
- Tsuge, Hiroko
- Arimura, Naoto
- Kawakami, Kazutoshi
- Sakamoto, Junichi
- Funami, Miyuki
- Mol, Clifford D
- Snell, Gyorgy P
- Bragstad, Kenneth A
- Sang, Bi-Ching
- Dougan, Douglas R
- Tanaka, Toshimasa
- Katayama, Nozomi
- Horiguchi, Yoshiaki
- Momose, Yu
Producer: 20120810
In:
Bioorganic & medicinal chemistry vol. 20
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Structural snapshots of human HDAC8 provide insights into the class I histone deacetylases. [electronic resource] by
- Somoza, John R
- Skene, Robert J
- Katz, Bradley A
- Mol, Clifford
- Ho, Joseph D
- Jennings, Andy J
- Luong, Christine
- Arvai, Andrew
- Buggy, Joseph J
- Chi, Ellen
- Tang, Jie
- Sang, Bi-Ching
- Verner, Erik
- Wynands, Robert
- Leahy, Ellen M
- Dougan, Douglas R
- Snell, Gyorgy
- Navre, Marc
- Knuth, Mark W
- Swanson, Ronald V
- McRee, Duncan E
- Tari, Leslie W
Producer: 20050209
In:
Structure (London, England : 1993) vol. 12
Availability: No items available.
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