Substitution scanning identifies a novel, catalytically active ibrutinib-resistant BTK cysteine 481 to threonine (C481T) variant. [electronic resource]
Producer: 20170830Description: 177-185 p. digitalISSN:- 1476-5551
- Adenine -- analogs & derivatives
- Agammaglobulinaemia Tyrosine Kinase
- Amino Acid Substitution
- Animals
- Biocatalysis
- Cell Line
- Cysteine
- Drug Resistance, Neoplasm -- genetics
- Humans
- Piperidines
- Protein Kinase Inhibitors -- pharmacology
- Protein-Tyrosine Kinases -- antagonists & inhibitors
- Pyrazoles -- pharmacology
- Pyrimidines -- pharmacology
- Threonine
- Transfection
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Publication Type: Journal Article
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