Results
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5-Amidinoindoles as dual inhibitors of coagulation factors IXa and Xa. [electronic resource] by
- Batt, Douglas G
- Qiao, Jennifer X
- Modi, Dilip P
- Houghton, Gregory C
- Pierson, Deborah A
- Rossi, Karen A
- Luettgen, Joseph M
- Knabb, Robert M
- Jadhav, P K
- Wexler, Ruth R
Producer: 20050505
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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3.
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Design and synthesis of benzoazepinone-derived cyclic malonamides and aminoamides as potent gamma-secretase inhibitors. [electronic resource] by
- Yang, Michael G
- Shi, Jian-Liang
- Modi, Dilip P
- Wells, Jennifer
- Cochran, Brian M
- Wolf, Mark A
- Thompson, Lorin A
- Ramanjulu, Mercy M
- Roach, Arthur H
- Zaczek, Robert
- Robertson, David W
- Wexler, Ruth R
- Olson, Richard E
Producer: 20070924
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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4.
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Potent benzimidazole sulfonamide protein tyrosine phosphatase 1B inhibitors containing the heterocyclic (S)-isothiazolidinone phosphotyrosine mimetic. [electronic resource] by
- Combs, Andrew P
- Zhu, Wenyu
- Crawley, Matthew L
- Glass, Brian
- Polam, Padmaja
- Sparks, Richard B
- Modi, Dilip
- Takvorian, Amy
- McLaughlin, Erin
- Yue, Eddy W
- Wasserman, Zelda
- Bower, Michael
- Wei, Min
- Rupar, Mark
- Ala, Paul J
- Reid, Brian M
- Ellis, Dawn
- Gonneville, Lucie
- Emm, Thomas
- Taylor, Nancy
- Yeleswaram, Swamy
- Li, Yanlong
- Wynn, Richard
- Burn, Timothy C
- Hollis, Gregory
- Liu, Phillip C C
- Metcalf, Brian
Producer: 20060816
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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5.
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INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology. [electronic resource] by
- Yue, Eddy W
- Sparks, Richard
- Polam, Padmaja
- Modi, Dilip
- Douty, Brent
- Wayland, Brian
- Glass, Brian
- Takvorian, Amy
- Glenn, Joseph
- Zhu, Wenyu
- Bower, Michael
- Liu, Xiangdong
- Leffet, Lynn
- Wang, Qian
- Bowman, Kevin J
- Hansbury, Michael J
- Wei, Min
- Li, Yanlong
- Wynn, Richard
- Burn, Timothy C
- Koblish, Holly K
- Fridman, Jordan S
- Emm, Tom
- Scherle, Peggy A
- Metcalf, Brian
- Combs, Andrew P
Publication details: ACS medicinal chemistry letters May 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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6.
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Discovery of INCB3284, a Potent, Selective, and Orally Bioavailable hCCR2 Antagonist. [electronic resource] by
- Xue, Chu-Biao
- Feng, Hao
- Cao, Ganfeng
- Huang, Taisheng
- Glenn, Joseph
- Anand, Rajan
- Meloni, David
- Zhang, Ke
- Kong, Lingquan
- Wang, Anlai
- Zhang, Yingxin
- Zheng, Changsheng
- Xia, Michael
- Chen, Lihua
- Tanaka, Hiroyuki
- Han, Qi
- Robinson, D J
- Modi, Dilip
- Storace, Lou
- Shao, Lixin
- Sharief, Vaqar
- Li, Mei
- Galya, Laurine G
- Covington, Maryanne
- Scherle, Peggy
- Diamond, Sharon
- Emm, Tom
- Yeleswaram, Swamy
- Contel, Nancy
- Vaddi, Kris
- Newton, Robert
- Hollis, Greg
- Friedman, Steven
- Metcalf, Brian
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 2
Availability: No items available.
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7.
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Structure-based design and discovery of protein tyrosine phosphatase inhibitors incorporating novel isothiazolidinone heterocyclic phosphotyrosine mimetics. [electronic resource] by
- Combs, Andrew P
- Yue, Eddy W
- Bower, Michael
- Ala, Paul J
- Wayland, Brian
- Douty, Brent
- Takvorian, Amy
- Polam, Padmaja
- Wasserman, Zelda
- Zhu, Wenyu
- Crawley, Matthew L
- Pruitt, James
- Sparks, Richard
- Glass, Brian
- Modi, Dilip
- McLaughlin, Erin
- Bostrom, Lori
- Li, Mei
- Galya, Laurine
- Blom, Karl
- Hillman, Milton
- Gonneville, Lucie
- Reid, Brian G
- Wei, Min
- Becker-Pasha, Mary
- Klabe, Ronald
- Huber, Reid
- Li, Yanlong
- Hollis, Gregory
- Burn, Timothy C
- Wynn, Richard
- Liu, Phillip
- Metcalf, Brian
Producer: 20051209
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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