Synthesis, transport and mechanism of a type I prodrug: L-carnitine ester of prednisolone. [electronic resource]
Producer: 20120224Description: 1629-40 p. digitalISSN:- 1543-8392
- Animals
- Anti-Inflammatory Agents -- blood
- Biological Transport
- Biotransformation
- Bronchi -- drug effects
- Carnitine -- analogs & derivatives
- Cell Line
- Drug Stability
- Gene Expression Regulation
- Glucocorticoids -- blood
- HEK293 Cells
- Humans
- Interleukin-6 -- metabolism
- Mice
- Organic Cation Transport Proteins -- antagonists & inhibitors
- Prednisolone -- analogs & derivatives
- Prodrugs -- analysis
- RNA, Messenger -- metabolism
- Respiratory Mucosa -- drug effects
- Solute Carrier Family 22 Member 5
- Substrate Specificity
- Succinates -- blood
- Symporters
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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