Results
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A novel series of histone deacetylase inhibitors incorporating hetero aromatic ring systems as connection units. [electronic resource] by
- Dai, Yujia
- Guo, Yan
- Curtin, Michael L
- Li, Junling
- Pease, Lori J
- Guo, Jun
- Marcotte, Patrick A
- Glaser, Keith B
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20040616
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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4.
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Succinimide hydroxamic acids as potent inhibitors of histone deacetylase (HDAC). [electronic resource] by
- Curtin, Michael L
- Garland, Robert B
- Heyman, H Robin
- Frey, Robin R
- Michaelides, Michael R
- Li, Junling
- Pease, Lori J
- Glaser, Keith B
- Marcotte, Patrick A
- Davidsen, Steven K
Producer: 20030311
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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5.
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Indole amide hydroxamic acids as potent inhibitors of histone deacetylases. [electronic resource] by
- Dai, Yujia
- Guo, Yan
- Guo, Jun
- Pease, Lori J
- Li, Junling
- Marcotte, Patrick A
- Glaser, Keith B
- Tapang, Paul
- Albert, Daniel H
- Richardson, Paul L
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20040217
In:
Bioorganic & medicinal chemistry letters vol. 13
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6.
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Discovery and development of potent and selective inhibitors of histone methyltransferase g9a. [electronic resource] by
- Sweis, Ramzi F
- Pliushchev, Marina
- Brown, Peter J
- Guo, Jun
- Li, Fengling
- Maag, David
- Petros, Andrew M
- Soni, Nirupama B
- Tse, Chris
- Vedadi, Masoud
- Michaelides, Michael R
- Chiang, Gary G
- Pappano, William N
Producer: 20140606
In:
ACS medicinal chemistry letters vol. 5
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Trifluoromethyl ketones as inhibitors of histone deacetylase. [electronic resource] by
- Frey, Robin R
- Wada, Carol K
- Garland, Robert B
- Curtin, Michael L
- Michaelides, Michael R
- Li, Junling
- Pease, Lori J
- Glaser, Keith B
- Marcotte, Patrick A
- Bouska, Jennifer J
- Murphy, Shannon S
- Davidsen, Steven K
Producer: 20030520
In:
Bioorganic & medicinal chemistry letters vol. 12
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Discovery of potent and selective thienopyrimidine inhibitors of Aurora kinases. [electronic resource] by
- McClellan, William J
- Dai, Yujia
- Abad-Zapatero, Cele
- Albert, Daniel H
- Bouska, Jennifer J
- Glaser, Keith B
- Magoc, Terry J
- Marcotte, Patrick A
- Osterling, Donald J
- Stewart, Kent D
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20111219
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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Exploration of diverse hinge-binding scaffolds for selective Aurora kinase inhibitors. [electronic resource] by
- Ji, Zhiqin
- Dai, Yujia
- Abad-Zapatero, Cele
- Albert, Daniel H
- Bouska, Jennifer J
- Glaser, Keith B
- Marcotte, Patrick A
- Soni, Nirupama B
- Magoc, Terry J
- Stewart, Kent D
- Wei, Ru-Qi
- Davidsen, Steve K
- Michaelides, Michael R
Producer: 20130104
In:
Bioorganic & medicinal chemistry letters vol. 22
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10.
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7-Aminopyrazolo[1,5-a]pyrimidines as potent multitargeted receptor tyrosine kinase inhibitors. [electronic resource] by
- Frey, Robin R
- Curtin, Michael L
- Albert, Daniel H
- Glaser, Keith B
- Pease, Lori J
- Soni, Niru B
- Bouska, Jennifer J
- Reuter, David
- Stewart, Kent D
- Marcotte, Patrick
- Bukofzer, Gail
- Li, Junling
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20080812
In:
Journal of medicinal chemistry vol. 51
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11.
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The Histone Methyltransferase Inhibitor A-366 Uncovers a Role for G9a/GLP in the Epigenetics of Leukemia. [electronic resource] by
- Pappano, William N
- Guo, Jun
- He, Yupeng
- Ferguson, Debra
- Jagadeeswaran, Sujatha
- Osterling, Donald J
- Gao, Wenqing
- Spence, Julie K
- Pliushchev, Marina
- Sweis, Ramzi F
- Buchanan, Fritz G
- Michaelides, Michael R
- Shoemaker, Alexander R
- Tse, Chris
- Chiang, Gary G
Producer: 20160419
In:
PloS one vol. 10
Availability: No items available.
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12.
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Heterocyclic ketones as inhibitors of histone deacetylase. [electronic resource] by
- Vasudevan, Anil
- Ji, Zhiqin
- Frey, Robin R
- Wada, Carol K
- Steinman, Douglas
- Heyman, H Robin
- Guo, Yan
- Curtin, Michael L
- Guo, Jun
- Li, Junling
- Pease, Lori
- Glaser, Keith B
- Marcotte, Patrick A
- Bouska, Jennifer J
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20040706
In:
Bioorganic & medicinal chemistry letters vol. 13
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13.
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Identification of aminopyrazolopyridine ureas as potent VEGFR/PDGFR multitargeted kinase inhibitors. [electronic resource] by
- Dai, Yujia
- Hartandi, Kresna
- Soni, Niru B
- Pease, Lori J
- Reuter, David R
- Olson, Amanda M
- Osterling, Donald J
- Doktor, Stella Z
- Albert, Daniel H
- Bouska, Jennifer J
- Glaser, Keith B
- Marcotte, Patrick A
- Stewart, Kent D
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20080212
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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14.
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Scaffold oriented synthesis. Part 2: Design, synthesis and biological evaluation of pyrimido-diazepines as receptor tyrosine kinase inhibitors. [electronic resource] by
- Gracias, Vijaya
- Ji, Zhiqin
- Akritopoulou-Zanze, Irini
- Abad-Zapatero, Cele
- Huth, Jeffrey R
- Song, Danying
- Hajduk, Philip J
- Johnson, Eric F
- Glaser, Keith B
- Marcotte, Patrick A
- Pease, Lori
- Soni, Nirupama B
- Stewart, Kent D
- Davidsen, Steven K
- Michaelides, Michael R
- Djuric, Stevan W
Producer: 20080516
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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15.
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Isothiazolopyrimidines and isoxazolopyrimidines as novel multi-targeted inhibitors of receptor tyrosine kinases. [electronic resource] by
- Ji, Zhiqin
- Ahmed, Asma A
- Albert, Daniel H
- Bouska, Jennifer J
- Bousquet, Peter F
- Cunha, George A
- Glaser, Keith B
- Guo, Jun
- Li, Junling
- Marcotte, Patrick A
- Moskey, Maria D
- Pease, Lori J
- Stewart, Kent D
- Yates, Melinda
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20061006
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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16.
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Hit-to-lead optimization of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of KDR kinase inhibitors. [electronic resource] by
- Dinges, Jürgen
- Akritopoulou-Zanze, Irini
- Arnold, Lee D
- Barlozzari, Teresa
- Bousquet, Peter F
- Cunha, George A
- Ericsson, Anna M
- Iwasaki, Nobuhiko
- Michaelides, Michael R
- Ogawa, Nobuo
- Phelan, Kathleen M
- Rafferty, Paul
- Sowin, Thomas J
- Stewart, Kent D
- Tokuyama, Ryukou
- Xia, Zhiren
- Zhang, Henry Q
Producer: 20061006
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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17.
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Isoindolinone ureas: a novel class of KDR kinase inhibitors. [electronic resource] by
- Curtin, Michael L
- Frey, Robin R
- Heyman, H Robin
- Sarris, Kathy A
- Steinman, Douglas H
- Holmes, James H
- Bousquet, Peter F
- Cunha, George A
- Moskey, Maria D
- Ahmed, Asma A
- Pease, Lori J
- Glaser, Keith B
- Stewart, Kent D
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20050209
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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18.
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1,4-Dihydroindeno[1,2-c]pyrazoles as novel multitargeted receptor tyrosine kinase inhibitors. [electronic resource] by
- Dinges, Jürgen
- Ashworth, Kimba L
- Akritopoulou-Zanze, Irini
- Akritopolou-Zanze, Irini
- Arnold, Lee D
- Baumeister, Steven A
- Bousquet, Peter F
- Cunha, George A
- Davidsen, Steven K
- Djuric, Stevan W
- Gracias, Vijaya J
- Michaelides, Michael R
- Rafferty, Paul
- Sowin, Thomas J
- Stewart, Kent D
- Xia, Zhiren
- Zhang, Henry Q
Producer: 20061006
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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19.
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3-amino-benzo[d]isoxazoles as novel multitargeted inhibitors of receptor tyrosine kinases. [electronic resource] by
- Ji, Zhiqin
- Ahmed, Asma A
- Albert, Daniel H
- Bouska, Jennifer J
- Bousquet, Peter F
- Cunha, George A
- Diaz, Gilbert
- Glaser, Keith B
- Guo, Jun
- Harris, Christopher M
- Li, Junling
- Marcotte, Patrick A
- Moskey, Maria D
- Oie, Tetsuro
- Pease, Lori
- Soni, Nirupama B
- Stewart, Kent D
- Davidsen, Steven K
- Michaelides, Michael R
Producer: 20080605
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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20.
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Pyrazole diaminopyrimidines as dual inhibitors of KDR and Aurora B kinases. [electronic resource] by
- Curtin, Michael L
- Heyman, H Robin
- Frey, Robin R
- Marcotte, Patrick A
- Glaser, Keith B
- Jankowski, James R
- Magoc, Terrance J
- Albert, Daniel H
- Olson, Amanda M
- Reuter, David R
- Bouska, Jennifer J
- Montgomery, Debra A
- Palma, Joann P
- Donawho, Cherrie K
- Stewart, Kent D
- Tse, Chris
- Michaelides, Michael R
Producer: 20130104
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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