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The discovery and SAR of cyclopenta[b]furans as inhibitors of CCR2. [electronic resource] by
- Winters, Michael P
- Teleha, Christopher A
- Kang, Fu-An
- McComsey, David
- O'Neill, John C
- Hou, Cuifen
- Kirchner, Thomas
- Wang, Ping
- Johnson, Dana
- Sui, Zhihua
Producer: 20141201
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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10.
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Inhibitors of Ketohexokinase: Discovery of Pyrimidinopyrimidines with Specific Substitution that Complements the ATP-Binding Site. [electronic resource] by
- Maryanoff, Bruce E
- O'Neill, John C
- McComsey, David F
- Yabut, Stephen C
- Luci, Diane K
- Jordan, Alfonzo D
- Masucci, John A
- Jones, William J
- Abad, Marta C
- Gibbs, Alan C
- Petrounia, Ioanna
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 2
Availability: No items available.
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11.
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Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3. [electronic resource] by
- Zhang, Han-Cheng
- White, Kimberly B
- Ye, Hong
- McComsey, David F
- Derian, Claudia K
- Addo, Michael F
- Andrade-Gordon, Patricia
- Eckardt, Annette J
- Conway, Bruce R
- Westover, Lori
- Xu, Jun Z
- Look, Richard
- Demarest, Keith T
- Emanuel, Stuart
- Maryanoff, Bruce E
Producer: 20040521
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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12.
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7-fluoroindazoles as potent and selective inhibitors of factor Xa. [electronic resource] by
- Lee, Yu-Kai
- Parks, Daniel J
- Lu, Tianbao
- Thieu, Tho V
- Markotan, Thomas
- Pan, Wenxi
- McComsey, David F
- Milkiewicz, Karen L
- Crysler, Carl S
- Ninan, Nisha
- Abad, Marta C
- Giardino, Edward C
- Maryanoff, Bruce E
- Damiano, Bruce P
- Player, Mark R
Producer: 20080417
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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13.
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Suzuki-Miyaura approach to JNJ-26076713, an orally active tetrahydroquinoline-containing alphaVbeta3/alphaVbeta5 integrin antagonist. enantioselective synthesis and stereochemical studies. [electronic resource] by
- Kinney, William A
- Teleha, Christopher A
- Thompson, Andrew S
- Newport, Maria
- Hansen, Ryan
- Ballentine, Scott
- Ghosh, Shyamali
- Mahan, Andrew
- Grasa, Gabriela
- Zanotti-Gerosa, Antonio
- Dingenen, Jules
- Schubert, Carsten
- Zhou, Yong
- Leo, Gregory C
- McComsey, David F
- Santulli, Rosemary J
- Maryanoff, Bruce E
Producer: 20080506
In:
The Journal of organic chemistry vol. 73
Availability: No items available.
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14.
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Next-generation spirobenzazepines: identification of RWJ-676070 as a balanced vasopressin V1a/V2 receptor antagonist for human clinical studies. [electronic resource] by
- Xiang, Min Amy
- Rybczynski, Philip J
- Patel, Mona
- Chen, Robert H
- McComsey, David F
- Zhang, Han-Cheng
- Gunnet, Joseph W
- Look, Richard
- Wang, Yuanping
- Minor, Lisa K
- Zhong, H Marlon
- Villani, Frank J
- Demarest, Keith T
- Damiano, Bruce P
- Maryanoff, Bruce E
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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15.
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Novel, broad-spectrum anticonvulsants containing a sulfamide group: pharmacological properties of (S)-N-[(6-chloro-2,3-dihydrobenzo[1,4]dioxin-2-yl)methyl]sulfamide (JNJ-26489112). [electronic resource] by
- McComsey, David F
- Smith-Swintosky, Virginia L
- Parker, Michael H
- Brenneman, Douglas E
- Malatynska, Ewa
- White, H Steve
- Klein, Brian D
- Wilcox, Karen S
- Milewski, Michael E
- Herb, Mark
- Finley, Michael F A
- Liu, Yi
- Lubin, Mary Lou
- Qin, Ning
- Reitz, Allen B
- Maryanoff, Bruce E
Producer: 20140130
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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16.
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Novel, broad-spectrum anticonvulsants containing a sulfamide group: advancement of N-((benzo[b]thien-3-yl)methyl)sulfamide (JNJ-26990990) into human clinical studies. [electronic resource] by
- Parker, Michael H
- Smith-Swintosky, Virginia L
- McComsey, David F
- Huang, Yifang
- Brenneman, Douglas
- Klein, Brian
- Malatynska, Ewa
- White, H Steve
- Milewski, Michael E
- Herb, Mark
- Finley, Michael F A
- Liu, Yi
- Lubin, Mary Lou
- Qin, Ning
- Iannucci, Robert
- Leclercq, Laurent
- Cuyckens, Filip
- Reitz, Allen B
- Maryanoff, Bruce E
Producer: 20091231
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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17.
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Novel indolylindazolylmaleimides as inhibitors of protein kinase C-beta: synthesis, biological activity, and cardiovascular safety. [electronic resource] by
- Zhang, Han-Cheng
- Derian, Claudia K
- McComsey, David F
- White, Kimberly B
- Ye, Hong
- Hecker, Leonard R
- Li, Jian
- Addo, Michael F
- Croll, Diane
- Eckardt, Annette J
- Smith, Charles E
- Li, Quan
- Cheung, Wai-Man
- Conway, Bruce R
- Emanuel, Stuart
- Demarest, Keith T
- Andrade-Gordon, Patricia
- Damiano, Bruce P
- Maryanoff, Bruce E
Producer: 20050503
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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