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Biaryl-bridged macrocyclic peptides: conformational constraint via carbogenic fusion of natural amino acid side chains. [electronic resource] by
- Meyer, Falco-Magnus
- Collins, James C
- Borin, Brendan
- Bradow, James
- Liras, Spiros
- Limberakis, Chris
- Mathiowetz, Alan M
- Philippe, Laurence
- Price, David
- Song, Kun
- James, Keith
Producer: 20120823
In:
The Journal of organic chemistry vol. 77
Availability: No items available.
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9.
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Exploring aromatic chemical space with NEAT: novel and electronically equivalent aromatic template. [electronic resource] by
- Tu, Meihua
- Rai, Brajesh K
- Mathiowetz, Alan M
- Didiuk, Mary
- Pfefferkorn, Jeffrey A
- Guzman-Perez, Angel
- Benbow, John
- Guimarães, Cristiano R W
- Mente, Scot
- Hayward, Matthew M
- Liras, Spiros
Producer: 20120928
In:
Journal of chemical information and modeling vol. 52
Availability: No items available.
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10.
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Achieving selectivity between highly homologous tyrosine kinases: a novel selective erbB2 inhibitor. [electronic resource] by
- Bhattacharya, Samit K
- Cox, Eric D
- Kath, John C
- Mathiowetz, Alan M
- Morris, Joel
- Moyer, James D
- Pustilnik, Leslie R
- Rafidi, Kris
- Richter, Daniel T
- Su, Chunyan
- Wessel, Matthew D
Producer: 20030916
In:
Biochemical and biophysical research communications vol. 307
Availability: No items available.
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11.
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A potentiator of orthosteric ligand activity at GLP-1R acts via covalent modification. [electronic resource] by
- Nolte, Whitney M
- Fortin, Jean-Philippe
- Stevens, Benjamin D
- Aspnes, Gary E
- Griffith, David A
- Hoth, Lise R
- Ruggeri, Roger B
- Mathiowetz, Alan M
- Limberakis, Chris
- Hepworth, David
- Carpino, Philip A
Producer: 20141006
In:
Nature chemical biology vol. 10
Availability: No items available.
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12.
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Nonclassical Size Dependence of Permeation Defines Bounds for Passive Adsorption of Large Drug Molecules. [electronic resource] by
- Pye, Cameron R
- Hewitt, William M
- Schwochert, Joshua
- Haddad, Terra D
- Townsend, Chad E
- Etienne, Lyns
- Lao, Yongtong
- Limberakis, Chris
- Furukawa, Akihiro
- Mathiowetz, Alan M
- Price, David A
- Liras, Spiros
- Lokey, R Scott
Producer: 20170807
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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13.
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Revisiting N-to-O acyl shift for synthesis of natural product-like cyclic depsipeptides. [electronic resource] by
- Schwochert, Joshua
- Pye, Cameron
- Ahlbach, Christopher
- Abdollahian, Yashar
- Farley, Kathleen
- Khunte, Bhagyashree
- Limberakis, Chris
- Kalgutkar, Amit S
- Eng, Heather
- Shapiro, Michael J
- Mathiowetz, Alan M
- Price, David A
- Liras, Spiros
- Lokey, R Scott
Producer: 20150420
In:
Organic letters vol. 16
Availability: No items available.
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14.
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Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue. [electronic resource] by
- Price, David A
- Eng, Heather
- Farley, Kathleen A
- Goetz, Gilles H
- Huang, Yong
- Jiao, Zhaodong
- Kalgutkar, Amit S
- Kablaoui, Natasha M
- Khunte, Bhagyashree
- Liras, Spiros
- Limberakis, Chris
- Mathiowetz, Alan M
- Ruggeri, Roger B
- Quan, Jun-Min
- Yang, Zhen
Producer: 20180213
In:
Organic & biomolecular chemistry vol. 15
Availability: No items available.
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15.
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Probing the Physicochemical Boundaries of Cell Permeability and Oral Bioavailability in Lipophilic Macrocycles Inspired by Natural Products. [electronic resource] by
- Bockus, Andrew T
- Lexa, Katrina W
- Pye, Cameron R
- Kalgutkar, Amit S
- Gardner, Jarret W
- Hund, Kathryn C R
- Hewitt, William M
- Schwochert, Joshua A
- Glassey, Emerson
- Price, David A
- Mathiowetz, Alan M
- Liras, Spiros
- Jacobson, Matthew P
- Lokey, R Scott
Producer: 20150928
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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16.
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Optimizing PK properties of cyclic peptides: the effect of side chain substitutions on permeability and clearance(). [electronic resource] by
- Rand, Arthur C
- Leung, Siegfried S F
- Eng, Heather
- Rotter, Charles J
- Sharma, Raman
- Kalgutkar, Amit S
- Zhang, Yizhong
- Varma, Manthena V
- Farley, Kathleen A
- Khunte, Bhagyashree
- Limberakis, Chris
- Price, David A
- Liras, Spiros
- Mathiowetz, Alan M
- Jacobson, Matthew P
- Lokey, R Scott
Publication details: MedChemComm Oct 2012
In:
MedChemComm vol. 3
Availability: No items available.
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17.
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Peptide to Peptoid Substitutions Increase Cell Permeability in Cyclic Hexapeptides. [electronic resource] by
- Schwochert, Joshua
- Turner, Rushia
- Thang, Melissa
- Berkeley, Ray F
- Ponkey, Alexandra R
- Rodriguez, Kelsie M
- Leung, Siegfried S F
- Khunte, Bhagyashree
- Goetz, Gilles
- Limberakis, Chris
- Kalgutkar, Amit S
- Eng, Heather
- Shapiro, Michael J
- Mathiowetz, Alan M
- Price, David A
- Liras, Spiros
- Jacobson, Matthew P
- Lokey, R Scott
Producer: 20151012
In:
Organic letters vol. 17
Availability: No items available.
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18.
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On-resin N-methylation of cyclic peptides for discovery of orally bioavailable scaffolds. [electronic resource] by
- White, Tina R
- Renzelman, Chad M
- Rand, Arthur C
- Rezai, Taha
- McEwen, Cayla M
- Gelev, Vladimir M
- Turner, Rushia A
- Linington, Roger G
- Leung, Siegfried S F
- Kalgutkar, Amit S
- Bauman, Jonathan N
- Zhang, Yizhong
- Liras, Spiros
- Price, David A
- Mathiowetz, Alan M
- Jacobson, Matthew P
- Lokey, R Scott
Producer: 20111222
In:
Nature chemical biology vol. 7
Availability: No items available.
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19.
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Decreasing the rate of metabolic ketone reduction in the discovery of a clinical acetyl-CoA carboxylase inhibitor for the treatment of diabetes. [electronic resource] by
- Griffith, David A
- Kung, Daniel W
- Esler, William P
- Amor, Paul A
- Bagley, Scott W
- Beysen, Carine
- Carvajal-Gonzalez, Santos
- Doran, Shawn D
- Limberakis, Chris
- Mathiowetz, Alan M
- McPherson, Kirk
- Price, David A
- Ravussin, Eric
- Sonnenberg, Gabriele E
- Southers, James A
- Sweet, Laurel J
- Turner, Scott M
- Vajdos, Felix F
Producer: 20150310
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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20.
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Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists. [electronic resource] by
- Hoang, Huy N
- Song, Kun
- Hill, Timothy A
- Derksen, David R
- Edmonds, David J
- Kok, W Mei
- Limberakis, Chris
- Liras, Spiros
- Loria, Paula M
- Mascitti, Vincent
- Mathiowetz, Alan M
- Mitchell, Justin M
- Piotrowski, David W
- Price, David A
- Stanton, Robert V
- Suen, Jacky Y
- Withka, Jane M
- Griffith, David A
- Fairlie, David P
Producer: 20150806
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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