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Discovery of potent and selective DP1 receptor antagonists in the azaindole series. [electronic resource] by
- Leblanc, Yves
- Roy, Patrick
- Dufresne, Claude
- Lachance, Nicolas
- Wang, Zhaoyin
- O'Neill, Gary
- Greig, Gillian
- Denis, Danielle
- Mathieu, Marie-Claude
- Slipetz, Deborah
- Sawyer, Nicole
- Tsou, Nancy
Producer: 20090826
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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5.
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Mutual antagonistic relationship between prostaglandin E(2) and IFN-gamma: Implications for rheumatoid arthritis. [electronic resource] by
- Mathieu, Marie-Claude
- Lord-Dufour, Simon
- Bernier, Virginie
- Boie, Yves
- Burch, Jason D
- Clark, Patsy
- Denis, Danielle
- Han, Yongxin
- Mortimer, James R
- Therien, Alex G
Producer: 20080902
In:
European journal of immunology vol. 38
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6.
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MF498 [N-{[4-(5,9-Diethoxy-6-oxo-6,8-dihydro-7H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylbenzyl]sulfonyl}-2-(2-methoxyphenyl)acetamide], a selective E prostanoid receptor 4 antagonist, relieves joint inflammation and pain in rodent models of rheumatoid and osteoarthritis. [electronic resource] by
- Clark, Patsy
- Rowland, Steven E
- Denis, Danielle
- Mathieu, Marie-Claude
- Stocco, Rino
- Poirier, Hugo
- Burch, Jason
- Han, Yongxin
- Audoly, Laurent
- Therien, Alex G
- Xu, Daigen
Producer: 20080519
In:
The Journal of pharmacology and experimental therapeutics vol. 325
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Gene expression profiling following NRF2 and KEAP1 siRNA knockdown in human lung fibroblasts identifies CCL11/Eotaxin-1 as a novel NRF2 regulated gene. [electronic resource] by
- Fourtounis, Jimmy
- Wang, I-Ming
- Mathieu, Marie-Claude
- Claveau, David
- Loo, Tenneille
- Jackson, Aimee L
- Peters, Mette A
- Therien, Alex G
- Boie, Yves
- Crackower, Michael A
Producer: 20130801
In:
Respiratory research vol. 13
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Identification of prostaglandin D2 receptor antagonists based on a tetrahydropyridoindole scaffold. [electronic resource] by
- Beaulieu, Christian
- Guay, Daniel
- Wang, Zhaoyin
- Leblanc, Yves
- Roy, Patrick
- Dufresne, Claude
- Zamboni, Robert
- Berthelette, Carl
- Day, Stephen
- Tsou, Nancy
- Denis, Danielle
- Greig, Gillian
- Mathieu, Marie-Claude
- O'Neill, Gary
Producer: 20080516
In:
Bioorganic & medicinal chemistry letters vol. 18
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The C3a receptor antagonist SB 290157 has agonist activity. [electronic resource] by
- Mathieu, Marie-Claude
- Sawyer, Nicole
- Greig, Gillian M
- Hamel, Martine
- Kargman, Stacia
- Ducharme, Yves
- Lau, Cheuk K
- Friesen, Richard W
- O'Neill, Gary P
- Gervais, Francois G
- Therien, Alex G
Producer: 20060912
In:
Immunology letters vol. 100
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10.
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A novel series of potent and selective EP(4) receptor ligands: facile modulation of agonism and antagonism. [electronic resource] by
- Boyd, Michael J
- Berthelette, Carl
- Chiasson, Jean-François
- Clark, Patsy
- Colucci, John
- Denis, Danielle
- Han, Yongxin
- Lévesque, Jean-Francois
- Mathieu, Marie-Claude
- Stocco, Rino
- Therien, Alex
- Rowland, Steve
- Wrona, Mark
- Xu, Daigen
Producer: 20110414
In:
Bioorganic & medicinal chemistry letters vol. 21
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Structure-function relationships in the neuropeptide S receptor: molecular consequences of the asthma-associated mutation N107I. [electronic resource] by
- Bernier, Virginie
- Stocco, Rino
- Bogusky, Michael J
- Joyce, Joseph G
- Parachoniak, Christine
- Grenier, Karl
- Arget, Michael
- Mathieu, Marie-Claude
- O'Neill, Gary P
- Slipetz, Deborah
- Crackower, Michael A
- Tan, Christopher M
- Therien, Alex G
Producer: 20061106
In:
The Journal of biological chemistry vol. 281
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12.
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Discovery of 4-[1-[([1-[4-(trifluoromethyl)benzyl]-1H-indol-7-yl]carbonyl)amino]cyclopropyl]benzoic acid (MF-766), a highly potent and selective EP4 antagonist for treating inflammatory pain. [electronic resource] by
- Colucci, John
- Boyd, Michael
- Berthelette, Carl
- Chiasson, Jean-Francois
- Wang, Zhaoyin
- Ducharme, Yves
- Friesen, Rick
- Wrona, Mark
- Levesque, Jean-Francois
- Denis, Danielle
- Mathieu, Marie-Claude
- Stocco, Rino
- Therien, Alex G
- Clarke, Patsy
- Rowland, Steve
- Xu, Daigen
- Han, Yongxin
Producer: 20100913
In:
Bioorganic & medicinal chemistry letters vol. 20
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13.
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Naphthalene/quinoline amides and sulfonylureas as potent and selective antagonists of the EP4 receptor. [electronic resource] by
- Burch, Jason D
- Farand, Julie
- Colucci, John
- Sturino, Claudio
- Ducharme, Yves
- Friesen, Richard W
- Lévesque, Jean-François
- Gagné, Sébastien
- Wrona, Mark
- Therien, Alex G
- Mathieu, Marie-Claude
- Denis, Danielle
- Vigneault, Erika
- Xu, Daigen
- Clark, Patsy
- Rowland, Steve
- Han, Yongxin
Producer: 20110502
In:
Bioorganic & medicinal chemistry letters vol. 21
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Adenovirus IL-13-induced airway disease in mice: a corticosteroid-resistant model of severe asthma. [electronic resource] by
- Therien, Alex G
- Bernier, Virginie
- Weicker, Sean
- Tawa, Paul
- Falgueyret, Jean-Pierre
- Mathieu, Marie-Claude
- Honsberger, Jeanne
- Pomerleau, Véronique
- Robichaud, Annette
- Stocco, Rino
- Dufresne, Lynn
- Houshyar, Hani
- Lafleur, Josiane
- Ramachandran, Chidambaram
- O'Neill, Gary P
- Slipetz, Deborah
- Tan, Christopher M
Producer: 20080801
In:
American journal of respiratory cell and molecular biology vol. 39
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15.
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Structure-activity relationships and pharmacokinetic parameters of quinoline acylsulfonamides as potent and selective antagonists of the EP(4) receptor. [electronic resource] by
- Burch, Jason D
- Belley, Michel
- Fortin, Réjean
- Deschênes, Denis
- Girard, Mario
- Colucci, John
- Farand, Julie
- Therien, Alex G
- Mathieu, Marie-Claude
- Denis, Danielle
- Vigneault, Erika
- Lévesque, Jean-François
- Gagné, Sébastien
- Wrona, Mark
- Xu, Daigen
- Clark, Patsy
- Rowland, Steve
- Han, Yongxin
Producer: 20080609
In:
Bioorganic & medicinal chemistry letters vol. 18
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16.
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The discovery of 4-{1-[({2,5-dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}carbonyl)amino]cyclopropyl}benzoic acid (MK-2894), a potent and selective prostaglandin E2 subtype 4 receptor antagonist. [electronic resource] by
- Blouin, Marc
- Han, Yongxin
- Burch, Jason
- Farand, Julie
- Mellon, Christophe
- Gaudreault, Mireille
- Wrona, Mark
- Lévesque, Jean-François
- Denis, Danielle
- Mathieu, Marie-Claude
- Stocco, Rino
- Vigneault, Erika
- Therien, Alex
- Clark, Patsy
- Rowland, Steve
- Xu, Daigen
- O'Neill, Gary
- Ducharme, Yves
- Friesen, Rick
Producer: 20100401
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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17.
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Identification of an indole series of prostaglandin D2 receptor antagonists. [electronic resource] by
- Sturino, Claudio F
- Lachance, Nicolas
- Boyd, Michael
- Berthelette, Carl
- Labelle, Marc
- Li, Lianhai
- Roy, Bruno
- Scheigetz, John
- Tsou, Nancy
- Brideau, Christine
- Cauchon, Elizabeth
- Carriere, Marie-Claude
- Denis, Danielle
- Greig, Gillian
- Kargman, Stacia
- Lamontagne, Sonia
- Mathieu, Marie-Claude
- Sawyer, Nicole
- Slipetz, Deborah
- O'Neill, Gary
- Wang, Zhaoyin
- Zamboni, Robert
- Metters, Kathleen M
- Young, Robert N
Producer: 20060802
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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18.
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Discovery of a potent and selective prostaglandin D2 receptor antagonist, [(3R)-4-(4-chloro-benzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]-acetic acid (MK-0524). [electronic resource] by
- Sturino, Claudio F
- O'Neill, Gary
- Lachance, Nicolas
- Boyd, Michael
- Berthelette, Carl
- Labelle, Marc
- Li, Lianhai
- Roy, Bruno
- Scheigetz, John
- Tsou, Nancy
- Aubin, Yves
- Bateman, Kevin P
- Chauret, Nathalie
- Day, Stephen H
- Lévesque, Jean-François
- Seto, Carmai
- Silva, Jose H
- Trimble, Laird A
- Carriere, Marie-Claude
- Denis, Danielle
- Greig, Gillian
- Kargman, Stacia
- Lamontagne, Sonia
- Mathieu, Marie-Claude
- Sawyer, Nicole
- Slipetz, Deborah
- Abraham, William M
- Jones, Tom
- McAuliffe, Malia
- Piechuta, Hana
- Nicoll-Griffith, Deborah A
- Wang, Zhaoyin
- Zamboni, Robert
- Young, Robert N
- Metters, Kathleen M
Producer: 20070327
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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