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Identification of potent and reversible cruzipain inhibitors for the treatment of Chagas disease. [electronic resource] by
- Beaulieu, Christian
- Isabel, Elise
- Fortier, Angélique
- Massé, Frédéric
- Mellon, Christophe
- Méthot, Nathalie
- Ndao, Momar
- Nicoll-Griffith, Deborah
- Lee, Doris
- Park, Hyeram
- Black, W Cameron
Producer: 20110314
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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7.
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Reversible cysteine protease inhibitors show promise for a Chagas disease cure. [electronic resource] by
- Ndao, Momar
- Beaulieu, Christian
- Black, W Cameron
- Isabel, Elise
- Vasquez-Camargo, Fabio
- Nath-Chowdhury, Milli
- Massé, Frédéric
- Mellon, Christophe
- Methot, Nathalie
- Nicoll-Griffith, Deborah A
Producer: 20140922
In:
Antimicrobial agents and chemotherapy vol. 58
Availability: No items available.
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8.
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Lysosomotropism of basic cathepsin K inhibitors contributes to increased cellular potencies against off-target cathepsins and reduced functional selectivity. [electronic resource] by
- Falgueyret, Jean-Pierre
- Desmarais, Sylvie
- Oballa, Renata
- Black, W Cameron
- Cromlish, Wanda
- Khougaz, Karine
- Lamontagne, Sonia
- Massé, Frederic
- Riendeau, Denis
- Toulmond, Sylvie
- Percival, M David
Producer: 20060209
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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9.
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A role for the malonyl-CoA/long-chain acyl-CoA pathway of lipid signaling in the regulation of insulin secretion in response to both fuel and nonfuel stimuli. [electronic resource] by
- Roduit, Raphaël
- Nolan, Christopher
- Alarcon, Cristina
- Moore, Patrick
- Barbeau, Annie
- Delghingaro-Augusto, Viviane
- Przybykowski, Ewa
- Morin, Johane
- Massé, Frédéric
- Massie, Bernard
- Ruderman, Neil
- Rhodes, Christopher
- Poitout, Vincent
- Prentki, Marc
Producer: 20040520
In:
Diabetes vol. 53
Availability: No items available.
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10.
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The discovery of setileuton, a potent and selective 5-lipoxygenase inhibitor. [electronic resource] by
- Ducharme, Yves
- Blouin, Marc
- Brideau, Christine
- Châteauneuf, Anne
- Gareau, Yves
- Grimm, Erich L
- Juteau, Hélène
- Laliberté, Sébastien
- MacKay, Bruce
- Massé, Frédéric
- Ouellet, Marc
- Salem, Myriam
- Styhler, Angela
- Friesen, Richard W
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
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11.
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Synthesis and biological activity of a potent and orally bioavailable SCD inhibitor (MF-438). [electronic resource] by
- Léger, Serge
- Black, W Cameron
- Deschenes, Denis
- Dolman, Sarah
- Falgueyret, Jean-Pierre
- Gagnon, Marc
- Guiral, Sébastien
- Huang, Zheng
- Guay, Jocelyne
- Leblanc, Yves
- Li, Chun-Sing
- Massé, Frédéric
- Oballa, Renata
- Zhang, Lei
Producer: 20100420
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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12.
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Beta-substituted cyclohexanecarboxamide cathepsin K inhibitors: modification of the 1,2-disubstituted aromatic core. [electronic resource] by
- Robichaud, Joël
- Bayly, Christopher I
- Black, W Cameron
- Desmarais, Sylvie
- Léger, Serge
- Massé, Frédéric
- McKay, Daniel J
- Oballa, Renata M
- Pâquet, Julie
- Percival, M David
- Truchon, Jean-François
- Wesolowski, Gregg
- Crane, Sheldon N
Producer: 20070807
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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13.
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Trifluoroethylamines as amide isosteres in inhibitors of cathepsin K. [electronic resource] by
- Black, W Cameron
- Bayly, Christopher I
- Davis, Dana E
- Desmarais, Sylvie
- Falgueyret, Jean-Pierre
- Léger, Serge
- Li, Chun Sing
- Massé, Frédéric
- McKay, Daniel J
- Palmer, James T
- Percival, M David
- Robichaud, Joël
- Tsou, Nancy
- Zamboni, Robert
Producer: 20051223
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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14.
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The identification of potent, selective, and bioavailable cathepsin S inhibitors. [electronic resource] by
- Gauthier, Jacques Yves
- Black, W Cameron
- Courchesne, Isabelle
- Cromlish, Wanda
- Desmarais, Sylvie
- Houle, Robert
- Lamontagne, Sonia
- Li, Chun Sing
- Massé, Frédéric
- McKay, Daniel J
- Ouellet, Marc
- Robichaud, Joël
- Truchon, Jean-François
- Truong, Vouy-Linh
- Wang, Qingping
- Percival, M David
Producer: 20071120
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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15.
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Substituted phenanthrene imidazoles as potent, selective, and orally active mPGES-1 inhibitors. [electronic resource] by
- Côté, Bernard
- Boulet, Louise
- Brideau, Christine
- Claveau, David
- Ethier, Diane
- Frenette, Richard
- Gagnon, Marc
- Giroux, André
- Guay, Jocelyne
- Guiral, Sébastien
- Mancini, Joseph
- Martins, Evelyn
- Massé, Frédéric
- Méthot, Nathalie
- Riendeau, Denis
- Rubin, Joel
- Xu, Daigen
- Yu, Hongping
- Ducharme, Yves
- Friesen, Richard W
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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16.
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Discovery of disubstituted phenanthrene imidazoles as potent, selective and orally active mPGES-1 inhibitors. [electronic resource] by
- Giroux, André
- Boulet, Louise
- Brideau, Christine
- Chau, Anh
- Claveau, David
- Côté, Bernard
- Ethier, Diane
- Frenette, Richard
- Gagnon, Marc
- Guay, Jocelyne
- Guiral, Sébastien
- Mancini, Joseph
- Martins, Evelyn
- Massé, Frédéric
- Méthot, Nathalie
- Riendeau, Denis
- Rubin, Joel
- Xu, Daigen
- Yu, Hongping
- Ducharme, Yves
- Friesen, Richard W
Producer: 20100105
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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17.
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Trisubstituted ureas as potent and selective mPGES-1 inhibitors. [electronic resource] by
- Chiasson, Jean-François
- Boulet, Louise
- Brideau, Christine
- Chau, Anh
- Claveau, David
- Côté, Bernard
- Ethier, Diane
- Giroux, André
- Guay, Jocelyne
- Guiral, Sébastien
- Mancini, Joseph
- Massé, Frédéric
- Méthot, Nathalie
- Riendeau, Denis
- Roy, Patrick
- Rubin, Joel
- Xu, Daigen
- Yu, Hongping
- Ducharme, Yves
- Friesen, Richard W
Producer: 20110614
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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18.
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Identification of a nonbasic, nitrile-containing cathepsin K inhibitor (MK-1256) that is efficacious in a monkey model of osteoporosis. [electronic resource] by
- Robichaud, Jöel
- Black, W Cameron
- Thérien, Michel
- Paquet, Julie
- Oballa, Renata M
- Bayly, Christopher I
- McKay, Daniel J
- Wang, Qingping
- Isabel, Elise
- Léger, Serge
- Mellon, Christophe
- Kimmel, Donald B
- Wesolowski, Gregg
- Percival, M David
- Massé, Fréderic
- Desmarais, Sylvie
- Falgueyret, Jean-Pierre
- Crane, Sheldon N
Producer: 20081113
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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19.
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Beta-substituted cyclohexanecarboxamide: a nonpeptidic framework for the design of potent inhibitors of cathepsin K. [electronic resource] by
- Crane, Sheldon N
- Black, W Cameron
- Palmer, James T
- Davis, Dana E
- Setti, Eduardo
- Robichaud, Joel
- Paquet, Julie
- Oballa, Renata M
- Bayly, Christopher I
- McKay, Daniel J
- Somoza, John R
- Chauret, Natalie
- Seto, Carmai
- Scheigetz, John
- Wesolowski, Greg
- Massé, Frederic
- Desmarais, Sylvie
- Ouellet, Marc
Producer: 20060329
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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20.
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Identification of a potent and selective non-basic cathepsin K inhibitor. [electronic resource] by
- Li, Chun Sing
- Deschenes, Denis
- Desmarais, Sylvie
- Falgueyret, Jean-Pierre
- Gauthier, Jacques Yves
- Kimmel, Donald B
- Léger, Serge
- Massé, Frédéric
- McGrath, Mary E
- McKay, Daniel J
- Percival, M David
- Riendeau, Denis
- Rodan, Sevgi B
- Thérien, Michel
- Truong, Vouy-Linh
- Wesolowski, Gregg
- Zamboni, Robert
- Black, W Cameron
Producer: 20060719
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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