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Discovery of alpha-amidosulfones as potent and selective agonists of CB2: synthesis, SAR, and pharmacokinetic properties. [electronic resource] by
- Marx, Isaac E
- DiMauro, Erin F
- Cheng, Alan
- Emkey, Renee
- Hitchcock, Stephen A
- Huang, Liyue
- Huang, Ming Y
- Human, Jason
- Lee, Josie H
- Li, Xingwen
- Martin, Matthew W
- White, Ryan D
- Fremeau, Robert T
- Patel, Vinod F
Producer: 20090128
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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Inhibitors of β-site amyloid precursor protein cleaving enzyme (BACE1): identification of (S)-7-(2-fluoropyridin-3-yl)-3-((3-methyloxetan-3-yl)ethynyl)-5'H-spiro[chromeno[2,3-b]pyridine-5,4'-oxazol]-2'-amine (AMG-8718). [electronic resource] by
- Dineen, Thomas A
- Chen, Kui
- Cheng, Alan C
- Derakhchan, Katayoun
- Epstein, Oleg
- Esmay, Joel
- Hickman, Dean
- Kreiman, Chuck E
- Marx, Isaac E
- Wahl, Robert C
- Wen, Paul H
- Weiss, Matthew M
- Whittington, Douglas A
- Wood, Stephen
- Fremeau, Robert T
- White, Ryan D
- Patel, Vinod F
Producer: 20150226
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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4.
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Lead optimization and modulation of hERG activity in a series of aminooxazoline xanthene β-site amyloid precursor protein cleaving enzyme (BACE1) inhibitors. [electronic resource] by
- Epstein, Oleg
- Bryan, Marian C
- Cheng, Alan C
- Derakhchan, Katayoun
- Dineen, Thomas A
- Hickman, Dean
- Hua, Zihao
- Human, Jason B
- Kreiman, Charles
- Marx, Isaac E
- Weiss, Matthew M
- Wahl, Robert C
- Wen, Paul H
- Whittington, Douglas A
- Wood, Stephen
- Zheng, Xiao Mei
- Fremeau, Robert T
- White, Ryan D
- Patel, Vinod F
Producer: 20150226
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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5.
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Sulfonamides as Selective Na [electronic resource] by
- Marx, Isaac E
- Dineen, Thomas A
- Able, Jessica
- Bode, Christiane
- Bregman, Howard
- Chu-Moyer, Margaret
- DiMauro, Erin F
- Du, Bingfan
- Foti, Robert S
- Fremeau, Robert T
- Gao, Hua
- Gunaydin, Hakan
- Hall, Brian E
- Huang, Liyue
- Kornecook, Thomas
- Kreiman, Charles R
- La, Daniel S
- Ligutti, Joseph
- Lin, Min-Hwa Jasmine
- Liu, Dong
- McDermott, Jeff S
- Moyer, Bryan D
- Peterson, Emily A
- Roberts, Jonathan T
- Rose, Paul
- Wang, Jean
- Youngblood, Beth D
- Yu, Violeta
- Weiss, Matthew M
Publication details: ACS medicinal chemistry letters Dec 2016
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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6.
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Correction to "Sulfonamides as Selective Na [electronic resource] by
- Marx, Isaac E
- Dineen, Thomas A
- Able, Jessica
- Bode, Christiane
- Bregman, Howard
- Chu-Moyer, Margaret
- DiMauro, Erin F
- Du, Bingfan
- Foti, Robert S
- Fremeau, Robert T
- Gao, Hua
- Gunaydin, Hakan
- Hall, Brian E
- Huang, Liyue
- Kornecook, Thomas
- Kreiman, Charles R
- La, Daniel S
- Ligutti, Joseph
- Lin, Min-Hwa Jasmine
- Liu, Dong
- McDermott, Jeff S
- Moyer, Bryan D
- Nguyen, Hanh N
- Peterson, Emily A
- Roberts, Jonathan T
- Rose, Paul
- Wang, Jean
- Youngblood, Beth D
- Yu, Violeta
- Weiss, Matthew M
Publication details: ACS medicinal chemistry letters Mar 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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7.
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Sulfonamides as Selective Na [electronic resource] by
- Weiss, Matthew M
- Dineen, Thomas A
- Marx, Isaac E
- Altmann, Steven
- Boezio, Alessandro
- Bregman, Howard
- Chu-Moyer, Margaret
- DiMauro, Erin F
- Feric Bojic, Elma
- Foti, Robert S
- Gao, Hua
- Graceffa, Russell
- Gunaydin, Hakan
- Guzman-Perez, Angel
- Huang, Hongbing
- Huang, Liyue
- Jarosh, Michael
- Kornecook, Thomas
- Kreiman, Charles R
- Ligutti, Joseph
- La, Daniel S
- Lin, Min-Hwa Jasmine
- Liu, Dong
- Moyer, Bryan D
- Nguyen, Hanh N
- Peterson, Emily A
- Rose, Paul E
- Taborn, Kristin
- Youngblood, Beth D
- Yu, Violeta
- Fremeau, Robert T
Producer: 20170905
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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8.
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Sulfonamides as Selective Na [electronic resource] by
- Graceffa, Russell F
- Boezio, Alessandro A
- Able, Jessica
- Altmann, Steven
- Berry, Loren M
- Boezio, Christiane
- Butler, John R
- Chu-Moyer, Margaret
- Cooke, Melanie
- DiMauro, Erin F
- Dineen, Thomas A
- Feric Bojic, Elma
- Foti, Robert S
- Fremeau, Robert T
- Guzman-Perez, Angel
- Gao, Hua
- Gunaydin, Hakan
- Huang, Hongbing
- Huang, Liyue
- Ilch, Christopher
- Jarosh, Michael
- Kornecook, Thomas
- Kreiman, Charles R
- La, Daniel S
- Ligutti, Joseph
- Milgram, Benjamin C
- Lin, Min-Hwa Jasmine
- Marx, Isaac E
- Nguyen, Hanh N
- Peterson, Emily A
- Rescourio, Gwen
- Roberts, John
- Schenkel, Laurie
- Shimanovich, Roman
- Sparling, Brian A
- Stellwagen, John
- Taborn, Kristin
- Vaida, Karina R
- Wang, Jean
- Yeoman, John
- Yu, Violeta
- Zhu, Dawn
- Moyer, Bryan D
- Weiss, Matthew M
Producer: 20170905
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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