Results
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1.
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A novel series of N-(azetidin-3-yl)-2-(heteroarylamino)acetamide CCR2 antagonists. [electronic resource] by
- Subasinghe, Nalin L
- Lanter, James
- Markotan, Thomas
- Opas, Evan
- McKenney, Sandra
- Crysler, Carl
- Hou, Cuifen
- O'Neill, John
- Johnson, Dana
- Sui, Zhihua
Producer: 20131031
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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2.
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Overcoming hERG activity in the discovery of a series of 4-azetidinyl-1-aryl-cyclohexanes as CCR2 antagonists. [electronic resource] by
- Zhang, Xuqing
- Hufnagel, Heather
- Markotan, Thomas
- Lanter, James
- Cai, Chaozhong
- Hou, Cuifen
- Singer, Monica
- Opas, Evan
- McKenney, Sandra
- Crysler, Carl
- Johnson, Dana
- Sui, Zhihua
Producer: 20111219
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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3.
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Oxyguanidines. Part 2: Discovery of a novel orally active thrombin inhibitor through structure-based drug design and parallel synthesis. [electronic resource] by
- Lu, Tianbao
- Markotan, Thomas
- Coppo, Frank
- Tomczuk, Bruce
- Crysler, Carl
- Eisennagel, Stephen
- Spurlino, John
- Gremminger, Lisa
- Soll, Richard M
- Giardino, Edward C
- Bone, Roger
Producer: 20050207
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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4.
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The discovery of novel cyclohexylamide CCR2 antagonists. [electronic resource] by
- Lanter, James C
- Markotan, Thomas P
- Zhang, Xuqing
- Subasinghe, Nalin
- Kang, Fu-An
- Hou, Cuifen
- Singer, Monica
- Opas, Evan
- McKenney, Sandra
- Crysler, Carl
- Johnson, Dana
- Molloy, Christopher J
- Sui, Zhihua
Producer: 20120312
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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5.
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Discovery and clinical evaluation of 1-{N-[2-(amidinoaminooxy)ethyl]amino}carbonylmethyl-6-methyl-3-[2,2-difluoro-2-phenylethylamino]pyrazinone (RWJ-671818), a thrombin inhibitor with an oxyguanidine P1 motif. [electronic resource] by
- Lu, Tianbao
- Markotan, Thomas
- Ballentine, Shelley K
- Giardino, Edward C
- Spurlino, John
- Crysler, Carl S
- Brown, Kathryn
- Maryanoff, Bruce E
- Tomczuk, Bruce E
- Damiano, Bruce P
- Shukla, Umesh
- End, David
- Andrade-Gordon, Patricia
- Bone, Roger F
- Player, Mark R
Producer: 20100323
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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6.
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7-fluoroindazoles as potent and selective inhibitors of factor Xa. [electronic resource] by
- Lee, Yu-Kai
- Parks, Daniel J
- Lu, Tianbao
- Thieu, Tho V
- Markotan, Thomas
- Pan, Wenxi
- McComsey, David F
- Milkiewicz, Karen L
- Crysler, Carl S
- Ninan, Nisha
- Abad, Marta C
- Giardino, Edward C
- Maryanoff, Bruce E
- Damiano, Bruce P
- Player, Mark R
Producer: 20080417
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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7.
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Antibody drug conjugates of cleavable amino-alkyl and aryl maytansinoids. [electronic resource] by
- Nittoli, Thomas
- Kelly, Marcus P
- Delfino, Frank
- Rudge, John
- Kunz, Arthur
- Markotan, Thomas
- Spink, Jan
- Chen, Zhaoyuan
- Shan, Jing
- Navarro, Elizabeth
- Tait, Michele
- Provoncha, Kathleen
- Giurleo, Jason
- Zhao, Feng
- Jiang, Xiaobo
- Hylton, Donna
- Makonnen, Sosina
- Hickey, Carlos
- Kirshner, Jessica R
- Thurston, Gavin
- Papadopoulos, Nicholas
Producer: 20190110
In:
Bioorganic & medicinal chemistry vol. 26
Availability: No items available.
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