Combinatorial target-guided ligand assembly: identification of potent subtype-selective c-Src inhibitors. [electronic resource]
Producer: 20000425Description: 2419-24 p. digitalISSN:- 0027-8424
- Adenosine Triphosphate -- metabolism
- CSK Tyrosine-Protein Kinase
- Combinatorial Chemistry Techniques
- Drug Design
- Inhibitory Concentration 50
- Ligands
- Magnetic Resonance Spectroscopy
- Models, Chemical
- Peptide Library
- Phosphorylation
- Protein Binding
- Protein-Tyrosine Kinases -- antagonists & inhibitors
- src-Family Kinases
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Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
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