Synthesis and biological evaluation of imidazo[4,5-b]pyridine and 4-heteroaryl-pyrimidine derivatives as anti-cancer agents. [electronic resource]
Producer: 20130509Description: 311-22 p. digitalISSN:- 1768-3254
- Amines -- chemical synthesis
- Antineoplastic Agents -- chemical synthesis
- Apoptosis -- drug effects
- Caspase 3 -- metabolism
- Caspase 7 -- metabolism
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Cyclin-Dependent Kinase 9 -- antagonists & inhibitors
- Drug Design
- Drug Discovery
- Enzyme Activation -- drug effects
- Humans
- Myeloid Cell Leukemia Sequence 1 Protein
- Protein Kinase Inhibitors -- chemical synthesis
- Proto-Oncogene Proteins c-bcl-2 -- antagonists & inhibitors
- Pyridines -- chemical synthesis
- Pyrimidines -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Journal Article
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