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Oxadiazolone bioisosteres of pregabalin and gabapentin. [electronic resource] by
- Wustrow, David J
- Belliotti, Thomas R
- Capiris, Thomas
- Kneen, Clare O
- Bryans, Justin S
- Field, Mark J
- Williams, Dic
- El-Kattan, Ayman
- Buchholz, Lisa
- Kinsora, Jack J
- Lotarski, Susan M
- Vartanian, Mark G
- Taylor, Charles P
- Donevan, Sean D
- Thorpe, Andrew J
- Schwarz, Jacob B
Producer: 20090128
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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5.
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Rational design of 7-arylquinolines as non-competitive metabotropic glutamate receptor subtype 5 antagonists. [electronic resource] by
- Milbank, Jared B J
- Knauer, Christopher S
- Augelli-Szafran, Corinne E
- Sakkab-Tan, Annette T
- Lin, Kristin K
- Yamagata, Koji
- Hoffman, Jennifer K
- Zhuang, Nian
- Thomas, John
- Galatsis, Paul
- Wendt, John A
- Mickelson, John W
- Schwarz, Roy D
- Kinsora, Jack J
- Lotarski, Susan M
- Stakich, Korana
- Gillespie, Kristen K
- Lam, Wing W
- Mutlib, Abdul E
Producer: 20071121
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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6.
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Design and Synthesis of γ- and δ-Lactam M [electronic resource] by
- Davoren, Jennifer E
- Garnsey, Michelle
- Pettersen, Betty
- Brodney, Michael A
- Edgerton, Jeremy R
- Fortin, Jean-Philippe
- Grimwood, Sarah
- Harris, Anthony R
- Jenkinson, Stephen
- Kenakin, Terry
- Lazzaro, John T
- Lee, Che-Wah
- Lotarski, Susan M
- Nottebaum, Lisa
- O'Neil, Steven V
- Popiolek, Michael
- Ramsey, Simeon
- Steyn, Stefanus J
- Thorn, Catherine A
- Zhang, Lei
- Webb, Damien
Producer: 20170905
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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7.
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Novel cyclopropyl beta-amino acid analogues of pregabalin and gabapentin that target the alpha2-delta protein. [electronic resource] by
- Schwarz, Jacob B
- Gibbons, Sian E
- Graham, Shelley R
- Colbry, Norman L
- Guzzo, Peter R
- Le, Van-Duc
- Vartanian, Mark G
- Kinsora, Jack J
- Lotarski, Susan M
- Li, Zheng
- Dickerson, Melvin R
- Su, Ti-Zhi
- Weber, Mark L
- El-Kattan, Ayman
- Thorpe, Andrew J
- Donevan, Sean D
- Taylor, Charles P
- Wustrow, David J
Producer: 20050524
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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8.
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Carboxylate bioisosteres of gabapentin. [electronic resource] by
- Burgos-Lepley, Carmen E
- Thompson, Lisa R
- Kneen, Clare O
- Osborne, Simon A
- Bryans, Justin S
- Capiris, Thomas
- Suman-Chauhan, Nirmala
- Dooley, David J
- Donovan, Cindy M
- Field, Mark J
- Vartanian, Mark G
- Kinsora, Jack J
- Lotarski, Susan M
- El-Kattan, Ayman
- Walters, Karen
- Cherukury, Madhu
- Taylor, Charles P
- Wustrow, David J
- Schwarz, Jacob B
Producer: 20060626
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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9.
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Carboxylate bioisosteres of pregabalin. [electronic resource] by
- Schwarz, Jacob B
- Colbry, Norman L
- Zhu, Zhijian
- Nichelson, Brian
- Barta, Nancy S
- Lin, Kristin
- Hudack, Raymond A
- Gibbons, Sian E
- Galatsis, Paul
- DeOrazio, Russell J
- Manning, David D
- Vartanian, Mark G
- Kinsora, Jack J
- Lotarski, Susan M
- Li, Zheng
- Dickerson, Melvin R
- El-Kattan, Ayman
- Thorpe, Andrew J
- Donevan, Sean D
- Taylor, Charles P
- Wustrow, David J
Producer: 20060802
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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10.
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Design and optimization of selective azaindole amide M1 positive allosteric modulators. [electronic resource] by
- Davoren, Jennifer E
- O'Neil, Steven V
- Anderson, Dennis P
- Brodney, Michael A
- Chenard, Lois
- Dlugolenski, Keith
- Edgerton, Jeremy R
- Green, Michael
- Garnsey, Michelle
- Grimwood, Sarah
- Harris, Anthony R
- Kauffman, Gregory W
- LaChapelle, Erik
- Lazzaro, John T
- Lee, Che-Wah
- Lotarski, Susan M
- Nason, Deane M
- Obach, R Scott
- Reinhart, Veronica
- Salomon-Ferrer, Romelia
- Steyn, Stefanus J
- Webb, Damien
- Yan, Jiangli
- Zhang, Lei
Producer: 20161011
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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11.
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The discovery and characterization of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor potentiator N-{(3S,4S)-4-[4-(5-cyano-2-thienyl)phenoxy]tetrahydrofuran-3-yl}propane-2-sulfonamide (PF-04958242). [electronic resource] by
- Shaffer, Christopher L
- Patel, Nandini C
- Schwarz, Jacob
- Scialis, Renato J
- Wei, Yunjing
- Hou, Xinjun J
- Xie, Longfei
- Karki, Kapil
- Bryce, Dianne K
- Osgood, Sarah M
- Hoffmann, William E
- Lazzaro, John T
- Chang, Cheng
- McGinnis, Dina F
- Lotarski, Susan M
- Liu, JianHua
- Obach, R Scott
- Weber, Mark L
- Chen, Laigao
- Zasadny, Kenneth R
- Seymour, Patricia A
- Schmidt, Christopher J
- Hajós, Mihály
- Hurst, Raymond S
- Pandit, Jayvardhan
- O'Donnell, Christopher J
Producer: 20150904
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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12.
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Discovery of the Potent and Selective M1 PAM-Agonist N-[(3R,4S)-3-Hydroxytetrahydro-2H-pyran-4-yl]-5-methyl-4-[4-(1,3-thiazol-4-yl)benzyl]pyridine-2-carboxamide (PF-06767832): Evaluation of Efficacy and Cholinergic Side Effects. [electronic resource] by
- Davoren, Jennifer E
- Lee, Che-Wah
- Garnsey, Michelle
- Brodney, Michael A
- Cordes, Jason
- Dlugolenski, Keith
- Edgerton, Jeremy R
- Harris, Anthony R
- Helal, Christopher J
- Jenkinson, Stephen
- Kauffman, Gregory W
- Kenakin, Terrence P
- Lazzaro, John T
- Lotarski, Susan M
- Mao, Yuxia
- Nason, Deane M
- Northcott, Carrie
- Nottebaum, Lisa
- O'Neil, Steven V
- Pettersen, Betty
- Popiolek, Michael
- Reinhart, Veronica
- Salomon-Ferrer, Romelia
- Steyn, Stefanus J
- Webb, Damien
- Zhang, Lei
- Grimwood, Sarah
Producer: 20170529
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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