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The discovery of quinoline based single-ligand human H [electronic resource] by
- Procopiou, Panayiotis A
- Ancliff, Rachael A
- Gore, Paul M
- Hancock, Ashley P
- Hodgson, Simon T
- Holmes, Duncan S
- Keeling, Steven P
- Looker, Brian E
- Parr, Nigel A
- Rowedder, James E
- Slack, Robert J
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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3.
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Design of Phthalazinone Amide Histamine H [electronic resource] by
- Procopiou, Panayiotis A
- Ford, Alison J
- Gore, Paul M
- Looker, Brian E
- Hodgson, Simon T
- Holmes, Duncan S
- Vile, Sadie
- Clark, Kenneth L
- Saunders, Ken A
- Slack, Robert J
- Rowedder, James E
- Watts, Clarissa J
Publication details: ACS medicinal chemistry letters May 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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4.
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Identification of selective 8-(piperidin-4-yloxy)quinoline sulfone and sulfonamide histamine H [electronic resource] by
- Procopiou, Panayiotis A
- Ford, Alison J
- Gore, Paul M
- Hancock, Ashley P
- Hodgson, Simon T
- Holmes, Duncan S
- Looker, Brian E
- Vile, Sadie
- Clark, Kenneth L
- Saunders, Ken A
- Slack, Robert J
- Watts, Clarissa J
Producer: 20171206
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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5.
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Discovery of a rapidly metabolized, long-acting β(2) adrenergic receptor agonist with a short onset time incorporating a sulfone group suitable for once-daily dosing. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Biggadike, Keith
- Butchers, Peter R
- Craven, Andrew
- Ford, Alison J
- Guntrip, Stephen B
- Holmes, Duncan S
- Hughes, Sara C
- Jones, Anne E
- Looker, Brian E
- Mutch, Peter J
- Ruston, Mark
- Needham, Deborah
- Smith, Claire E
Producer: 20140310
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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6.
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The discovery of long-acting saligenin β₂ adrenergic receptor agonists incorporating hydantoin or uracil rings. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Bevan, Nicola J
- Butchers, Peter R
- Conroy, Richard
- Emmons, Amanda
- Ford, Alison J
- Jeulin, Séverine
- Looker, Brian E
- Lunniss, Gillian E
- Morrison, Valerie S
- Mutch, Peter J
- Perciaccante, Rossana
- Ruston, Mark
- Smith, Claire E
- Somers, Graham
Producer: 20111220
In:
Bioorganic & medicinal chemistry vol. 19
Availability: No items available.
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7.
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The discovery of phthalazinone-based human H1 and H3 single-ligand antagonists suitable for intranasal administration for the treatment of allergic rhinitis. [electronic resource] by
- Procopiou, Panayiotis A
- Browning, Christopher
- Buckley, Jennifer M
- Clark, Kenneth L
- Fechner, Lise
- Gore, Paul M
- Hancock, Ashley P
- Hodgson, Simon T
- Holmes, Duncan S
- Kranz, Michael
- Looker, Brian E
- Morriss, Karen M L
- Parton, Daniel L
- Russell, Linda J
- Slack, Robert J
- Sollis, Steven L
- Vile, Sadie
- Watts, Clarissa J
Producer: 20110606
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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8.
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4-acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a novel class of non-brain-penetrant histamine H3 receptor antagonists. [electronic resource] by
- Procopiou, Panayiotis A
- Ancliff, Rachael A
- Bamford, Mark J
- Browning, Christopher
- Connor, Helen
- Davies, Susannah
- Fogden, Yvonne C
- Hodgson, Simon T
- Holmes, Duncan S
- Looker, Brian E
- Morriss, Karen M L
- Parr, Christopher A
- Pickup, Elizabeth A
- Sehmi, Sanjeet S
- White, Gemma V
- Watts, Clarissa J
- Wilson, David M
- Woodrow, Michael D
Producer: 20080403
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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9.
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Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating arylsulfonamide groups. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Bevan, Nicola J
- Biggadike, Keith
- Butchers, Peter R
- Coe, Diane M
- Conroy, Richard
- Edney, Dean D
- Field, Rita N
- Ford, Alison J
- Guntrip, Stephen B
- Looker, Brian E
- McLay, Iain M
- Monteith, Michael J
- Morrison, Valerie S
- Mutch, Peter J
- Richards, Stephen A
- Sasse, Rosemary
- Smith, Claire E
Producer: 20090506
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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10.
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Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating metabolic inactivation: an antedrug approach. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Bevan, Nicola J
- Biggadike, Keith
- Box, Philip C
- Butchers, Peter R
- Coe, Diane M
- Conroy, Richard
- Emmons, Amanda
- Ford, Alison J
- Holmes, Duncan S
- Horsley, Helen
- Kerr, Fern
- Li-Kwai-Cheung, Anne-Marie
- Looker, Brian E
- Mann, Inderjit S
- McLay, Iain M
- Morrison, Valerie S
- Mutch, Peter J
- Smith, Claire E
- Tomlin, Paula
Producer: 20100701
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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