Results
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1.
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Isocitrate dehydrogenase (IDH) mutations promote a reversible ZEB1/microRNA (miR)-200-dependent epithelial-mesenchymal transition (EMT). [electronic resource] by
- Grassian, Alexandra R
- Lin, Fallon
- Barrett, Rosemary
- Liu, Yue
- Jiang, Wei
- Korpal, Manav
- Astley, Holly
- Gitterman, Daniel
- Henley, Thomas
- Howes, Rob
- Levell, Julian
- Korn, Joshua M
- Pagliarini, Raymond
Producer: 20130212
In:
The Journal of biological chemistry vol. 287
Availability: No items available.
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2.
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Patient-derived glioblastoma cultures as a tool for small-molecule drug discovery. [electronic resource] by
- Ye, Ling F
- Reznik, Eduard
- Korn, Joshua M
- Lin, Fallon
- Yang, Guizhi
- Malesky, Kimberly
- Gao, Hui
- Loo, Alice
- Pagliarini, Raymond
- Mikkelsen, Tom
- Lo, Donald C
- deCarvalho, Ana C
- Stockwell, Brent R
Publication details: Oncotarget Jan 2020
In:
Oncotarget vol. 11
Availability: No items available.
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3.
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A small molecule that binds and inhibits the ETV1 transcription factor oncoprotein. [electronic resource] by
- Pop, Marius S
- Stransky, Nicolas
- Garvie, Colin W
- Theurillat, Jean-Philippe
- Hartman, Emily C
- Lewis, Timothy A
- Zhong, Cheng
- Culyba, Elizabeth K
- Lin, Fallon
- Daniels, Douglas S
- Pagliarini, Raymond
- Ronco, Lucienne
- Koehler, Angela N
- Garraway, Levi A
Producer: 20150219
In:
Molecular cancer therapeutics vol. 13
Availability: No items available.
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4.
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Allosteric Mutant IDH1 Inhibitors Reveal Mechanisms for IDH1 Mutant and Isoform Selectivity. [electronic resource] by
- Xie, Xiaoling
- Baird, Daniel
- Bowen, Kimberly
- Capka, Vladimir
- Chen, Jinyun
- Chenail, Gregg
- Cho, YoungShin
- Dooley, Julia
- Farsidjani, Ali
- Fortin, Pascal
- Kohls, Darcy
- Kulathila, Raviraj
- Lin, Fallon
- McKay, Daniel
- Rodrigues, Lindsey
- Sage, David
- Touré, B Barry
- van der Plas, Simon
- Wright, Kirk
- Xu, Ming
- Yin, Hong
- Levell, Julian
- Pagliarini, Raymond A
Producer: 20170823
In:
Structure (London, England : 1993) vol. 25
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5.
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ERG signaling in prostate cancer is driven through PRMT5-dependent methylation of the Androgen Receptor. [electronic resource] by
- Mounir, Zineb
- Korn, Joshua M
- Westerling, Thomas
- Lin, Fallon
- Kirby, Christina A
- Schirle, Markus
- McAllister, Gregg
- Hoffman, Greg
- Ramadan, Nadire
- Hartung, Anke
- Feng, Yan
- Kipp, David Randal
- Quinn, Christopher
- Fodor, Michelle
- Baird, Jason
- Schoumacher, Marie
- Meyer, Ronald
- Deeds, James
- Buchwalter, Gilles
- Stams, Travis
- Keen, Nicholas
- Sellers, William R
- Brown, Myles
- Pagliarini, Raymond A
Producer: 20171117
In:
eLife vol. 5
Availability: No items available.
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6.
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IDH1 mutations alter citric acid cycle metabolism and increase dependence on oxidative mitochondrial metabolism. [electronic resource] by
- Grassian, Alexandra R
- Parker, Seth J
- Davidson, Shawn M
- Divakaruni, Ajit S
- Green, Courtney R
- Zhang, Xiamei
- Slocum, Kelly L
- Pu, Minying
- Lin, Fallon
- Vickers, Chad
- Joud-Caldwell, Carol
- Chung, Franklin
- Yin, Hong
- Handly, Erika D
- Straub, Christopher
- Growney, Joseph D
- Vander Heiden, Matthew G
- Murphy, Anne N
- Pagliarini, Raymond
- Metallo, Christian M
Producer: 20140808
In:
Cancer research vol. 74
Availability: No items available.
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7.
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Optimization of 3-Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1. [electronic resource] by
- Levell, Julian R
- Caferro, Thomas
- Chenail, Gregg
- Dix, Ina
- Dooley, Julia
- Firestone, Brant
- Fortin, Pascal D
- Giraldes, John
- Gould, Ty
- Growney, Joseph D
- Jones, Michael D
- Kulathila, Raviraj
- Lin, Fallon
- Liu, Gang
- Mueller, Arne
- van der Plas, Simon
- Slocum, Kelly
- Smith, Troy
- Terranova, Remi
- Touré, B Barry
- Tyagi, Viraj
- Wagner, Trixie
- Xie, Xiaoling
- Xu, Ming
- Yang, Fan S
- Zhou, Liping X
- Pagliarini, Raymond
- Cho, Young Shin
Publication details: ACS medicinal chemistry letters Feb 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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8.
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Disordered methionine metabolism in MTAP/CDKN2A-deleted cancers leads to dependence on PRMT5. [electronic resource] by
- Mavrakis, Konstantinos J
- McDonald, E Robert
- Schlabach, Michael R
- Billy, Eric
- Hoffman, Gregory R
- deWeck, Antoine
- Ruddy, David A
- Venkatesan, Kavitha
- Yu, Jianjun
- McAllister, Gregg
- Stump, Mark
- deBeaumont, Rosalie
- Ho, Samuel
- Yue, Yingzi
- Liu, Yue
- Yan-Neale, Yan
- Yang, Guizhi
- Lin, Fallon
- Yin, Hong
- Gao, Hui
- Kipp, D Randal
- Zhao, Songping
- McNamara, Joshua T
- Sprague, Elizabeth R
- Zheng, Bing
- Lin, Ying
- Cho, Young Shin
- Gu, Justin
- Crawford, Kenneth
- Ciccone, David
- Vitari, Alberto C
- Lai, Albert
- Capka, Vladimir
- Hurov, Kristen
- Porter, Jeffery A
- Tallarico, John
- Mickanin, Craig
- Lees, Emma
- Pagliarini, Raymond
- Keen, Nicholas
- Schmelzle, Tobias
- Hofmann, Francesco
- Stegmeier, Frank
- Sellers, William R
Producer: 20160331
In:
Science (New York, N.Y.) vol. 351
Availability: No items available.
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