Results
|
1.
|
|
|
2.
|
|
|
3.
|
|
|
4.
|
Structural basis for pharmacological modulation of the TRPC6 channel. [electronic resource] by
- Bai, Yonghong
- Yu, Xinchao
- Chen, Hao
- Horne, Daniel
- White, Ryan
- Wu, Xiaosu
- Lee, Paul
- Gu, Yan
- Ghimire-Rijal, Sudipa
- Lin, Daniel C-H
- Huang, Xin
Producer: 20210402
In:
eLife vol. 9
Availability: No items available.
|
|
5.
|
Discovery of AM-6226: A Potent and Orally Bioavailable GPR40 Full Agonist That Displays Efficacy in Nonhuman Primates. [electronic resource] by
- Brown, Sean P
- Dransfield, Paul
- Vimolratana, Marc
- Zhu, Liusheng
- Luo, Jian
- Zhang, Jane
- Jiao, XianYun
- Pattaropong, Vatee
- Wong, Simon
- Zhuang, Run
- Swaminath, Gayathri
- Houze, Jonathan B
- Lin, Daniel C-H
Publication details: ACS medicinal chemistry letters Jul 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
|
|
6.
|
Evaluating insulin secretagogues in a humanized mouse model with functional human islets. [electronic resource] by
- Luo, Jian
- Nguyen, Kathy
- Chen, Michael
- Tran, Than
- Hao, Jianqiang
- Tian, Bole
- Rulifson, Ingrid C
- Zhang, Ying
- Tian, Lei
- Zhang, Yu
- Lopez, Edwin
- Lin, Daniel C-H
- Wang, Yingcai
- Ma, Zhihua
- Houze, Jonathan
- Guo, Zhiguang
Producer: 20130503
In:
Metabolism: clinical and experimental vol. 62
Availability: No items available.
|
|
7.
|
Identification and pharmacological characterization of multiple allosteric binding sites on the free fatty acid 1 receptor. [electronic resource] by
- Lin, Daniel C-H
- Guo, Qi
- Luo, Jian
- Zhang, Jane
- Nguyen, Kathy
- Chen, Michael
- Tran, Thanh
- Dransfield, Paul J
- Brown, Sean P
- Houze, Jonathan
- Vimolratana, Marc
- Jiao, Xian Yun
- Wang, Yingcai
- Birdsall, Nigel J M
- Swaminath, Gayathri
Producer: 20130212
In:
Molecular pharmacology vol. 82
Availability: No items available.
|
|
8.
|
A potent class of GPR40 full agonists engages the enteroinsular axis to promote glucose control in rodents. [electronic resource] by
- Luo, Jian
- Swaminath, Gayathri
- Brown, Sean P
- Zhang, Jane
- Guo, Qi
- Chen, Michael
- Nguyen, Kathy
- Tran, Thanhvien
- Miao, Lynn
- Dransfield, Paul J
- Vimolratana, Marc
- Houze, Jonathan B
- Wong, Simon
- Toteva, Maria
- Shan, Bei
- Li, Frank
- Zhuang, Run
- Lin, Daniel C-H
Producer: 20130611
In:
PloS one vol. 7
Availability: No items available.
|
|
9.
|
Discovery of AM-1638: A Potent and Orally Bioavailable GPR40/FFA1 Full Agonist. [electronic resource] by
- Brown, Sean P
- Dransfield, Paul J
- Vimolratana, Marc
- Jiao, XianYun
- Zhu, Liusheng
- Pattaropong, Vatee
- Sun, Ying
- Liu, Jinqian
- Luo, Jian
- Zhang, Jane
- Wong, Simon
- Zhuang, Run
- Guo, Qi
- Li, Frank
- Medina, Julio C
- Swaminath, Gayathri
- Lin, Daniel C-H
- Houze, Jonathan B
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
|
|
10.
|
Discovery of the imidazole-derived GPR40 agonist AM-3189. [electronic resource] by
- Ma, Zhihua
- Lin, Daniel C-H
- Sharma, Rajiv
- Liu, Jinqian
- Zhu, Liusheng
- Li, An-Rong
- Kohn, Todd
- Wang, Yingcai
- Liu, Jiwen Jim
- Bartberger, Michael D
- Medina, Julio C
- Zhuang, Run
- Li, Frank
- Zhang, Jane
- Luo, Jian
- Wong, Simon
- Tonn, George R
- Houze, Jonathan B
Producer: 20160727
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
|
|
11.
|
Activation of FFA1 mediates GLP-1 secretion in mice. Evidence for allosterism at FFA1. [electronic resource] by
- Xiong, Yumei
- Swaminath, Gayathri
- Cao, Qiong
- Yang, Li
- Guo, Qi
- Salomonis, Heather
- Lu, Jenny
- Houze, Jonathan B
- Dransfield, Paul J
- Wang, Yingcai
- Liu, Jiwen Jim
- Wong, Simon
- Schwandner, Ralf
- Steger, Franziska
- Baribault, Helene
- Liu, Lily
- Coberly, Suzanne
- Miao, Lynn
- Zhang, Jane
- Lin, Daniel C-H
- Schwarz, Margrit
Producer: 20130916
In:
Molecular and cellular endocrinology vol. 369
Availability: No items available.
|
|
12.
|
Optimization of GPR40 Agonists for Type 2 Diabetes. [electronic resource] by
- Liu, Jiwen Jim
- Wang, Yingcai
- Ma, Zhihua
- Schmitt, Mike
- Zhu, Liusheng
- Brown, Sean P
- Dransfield, Paul J
- Sun, Ying
- Sharma, Rajiv
- Guo, Qi
- Zhuang, Run
- Zhang, Jane
- Luo, Jian
- Tonn, George R
- Wong, Simon
- Swaminath, Gayathri
- Medina, Julio C
- Lin, Daniel C-H
- Houze, Jonathan B
Producer: 20140606
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
|
|
13.
|
AMG 837: a novel GPR40/FFA1 agonist that enhances insulin secretion and lowers glucose levels in rodents. [electronic resource] by
- Lin, Daniel C-H
- Zhang, Jane
- Zhuang, Run
- Li, Frank
- Nguyen, Kathy
- Chen, Michael
- Tran, Thanhvien
- Lopez, Edwin
- Lu, Jenny Ying Lin
- Li, Xiaoyan Nina
- Tang, Liang
- Tonn, George R
- Swaminath, Gayathri
- Reagan, Jeff D
- Chen, Jin-Long
- Tian, Hui
- Lin, Yi-Jyun
- Houze, Jonathan B
- Luo, Jian
Producer: 20120518
In:
PloS one vol. 6
Availability: No items available.
|
|
14.
|
Aminopyrazole-Phenylalanine Based GPR142 Agonists: Discovery of Tool Compound and in Vivo Efficacy Studies. [electronic resource] by
- Yu, Ming
- Lizarzaburu, Mike
- Motani, Alykhan
- Fu, Zice
- Du, Xiaohui
- Liu, Jiwen Jim
- Jiao, Xianyun
- Lai, SuJen
- Fan, Peter
- Fu, Angela
- Liu, Qingxiang
- Murakoshi, Michiko
- Nara, Futoshi
- Oda, Kozo
- Okuyama, Ryo
- Reagan, Jeff D
- Watanabe, Nobuaki
- Yamazaki, Mami
- Xiong, Yumei
- Zhang, Ying
- Zhuang, Run
- Lin, Daniel C-H
- Houze, Jonathan B
- Medina, Julio C
- Li, Leping
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
|
|
15.
|
AMG 837: a potent, orally bioavailable GPR40 agonist. [electronic resource] by
- Houze, Jonathan B
- Zhu, Liusheng
- Sun, Ying
- Akerman, Michelle
- Qiu, Wei
- Zhang, Alex J
- Sharma, Rajiv
- Schmitt, Michael
- Wang, Yingcai
- Liu, Jiwen
- Liu, Jinqian
- Medina, Julio C
- Reagan, Jeff D
- Luo, Jian
- Tonn, George
- Zhang, Jane
- Lu, Jenny Ying-Lin
- Chen, Michael
- Lopez, Edwin
- Nguyen, Kathy
- Yang, Li
- Tang, Liang
- Tian, Hui
- Shuttleworth, Steven J
- Lin, Daniel C-H
Producer: 20120824
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
|
|
16.
|
Improving the Pharmacokinetics of GPR40/FFA1 Full Agonists. [electronic resource] by
- Du, Xiaohui
- Dransfield, Paul J
- Lin, Daniel C-H
- Wong, Simon
- Wang, Yingcai
- Wang, Zhongyu
- Kohn, Todd
- Yu, Ming
- Brown, Sean P
- Vimolratana, Marc
- Zhu, Liusheng
- Li, An-Rong
- Su, Yongli
- Jiao, Xianyun
- Liu, Jiwen Jim
- Swaminath, Gayathri
- Tran, Thanhvien
- Luo, Jian
- Zhuang, Run
- Zhang, Jane
- Guo, Qi
- Li, Frank
- Connors, Richard
- Medina, Julio C
- Houze, Jonathan B
Producer: 20140606
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
|
|
17.
|
Discovery and Optimization of Potent GPR40 Full Agonists Containing Tricyclic Spirocycles. [electronic resource] by
- Wang, Yingcai
- Liu, Jiwen Jim
- Dransfield, Paul J
- Zhu, Liusheng
- Wang, Zhongyu
- Du, Xiaohui
- Jiao, Xianyun
- Su, Yongli
- Li, An-Rong
- Brown, Sean P
- Kasparian, Annie
- Vimolratana, Marc
- Yu, Ming
- Pattaropong, Vatee
- Houze, Jonathan B
- Swaminath, Gayathri
- Tran, Thanhvien
- Nguyen, Khanh
- Guo, Qi
- Zhang, Jane
- Zhuang, Run
- Li, Frank
- Miao, Lynn
- Bartberger, Michael D
- Correll, Tiffany L
- Chow, David
- Wong, Simon
- Luo, Jian
- Lin, Daniel C-H
- Medina, Julio C
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
|