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Novel reversible methionine aminopeptidase-2 (MetAP-2) inhibitors based on purine and related bicyclic templates. [electronic resource] by
- Heinrich, Timo
- Buchstaller, Hans-Peter
- Cezanne, Bertram
- Rohdich, Felix
- Bomke, Jörg
- Friese-Hamim, Manja
- Krier, Mireille
- Knöchel, Thorsten
- Musil, Djordje
- Leuthner, Birgitta
- Zenke, Frank
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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Discovery and Optimization of 2-Arylquinazolin-4-ones into a Potent and Selective Tankyrase Inhibitor Modulating Wnt Pathway Activity. [electronic resource] by
- Buchstaller, Hans-Peter
- Anlauf, Uwe
- Dorsch, Dieter
- Kuhn, Daniel
- Lehmann, Martin
- Leuthner, Birgitta
- Musil, Djordje
- Radtki, Daniela
- Ritzert, Claudio
- Rohdich, Felix
- Schneider, Richard
- Esdar, Christina
Producer: 20200629
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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5.
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Discovery and Structure-Based Optimization of Next-Generation Reversible Methionine Aminopeptidase-2 (MetAP-2) Inhibitors. [electronic resource] by
- Heinrich, Timo
- Seenisamy, Jeyaprakashnarayanan
- Blume, Beatrix
- Bomke, Jörg
- Calderini, Michel
- Eckert, Uwe
- Friese-Hamim, Manja
- Kohl, Rainer
- Lehmann, Martin
- Leuthner, Birgitta
- Musil, Djordje
- Rohdich, Felix
- Zenke, Frank T
Producer: 20200615
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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Identification of Methionine Aminopeptidase-2 (MetAP-2) Inhibitor [electronic resource] by
- Heinrich, Timo
- Seenisamy, Jeyaprakashnarayanan
- Becker, Frank
- Blume, Beatrix
- Bomke, Jörg
- Dietz, Melanie
- Eckert, Uwe
- Friese-Hamim, Manja
- Gunera, Jakub
- Hansen, Kerrin
- Leuthner, Birgitta
- Musil, Djordje
- Pfalzgraf, Jens
- Rohdich, Felix
- Siegl, Christian
- Spuck, Dieter
- Wegener, Ansgar
- Zenke, Frank T
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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A novel tankyrase inhibitor, MSC2504877, enhances the effects of clinical CDK4/6 inhibitors. [electronic resource] by
- Menon, Malini
- Elliott, Richard
- Bowers, Leandra
- Balan, Nicolae
- Rafiq, Rumana
- Costa-Cabral, Sara
- Munkonge, Felix
- Trinidade, Ines
- Porter, Roderick
- Campbell, Andrew D
- Johnson, Emma R
- Esdar, Christina
- Buchstaller, Hans-Peter
- Leuthner, Birgitta
- Rohdich, Felix
- Schneider, Richard
- Sansom, Owen
- Wienke, Dirk
- Ashworth, Alan
- Lord, Christopher J
Producer: 20200430
In:
Scientific reports vol. 9
Availability: No items available.
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Discovery of potent, orally bioavailable, small-molecule inhibitors of WNT signaling from a cell-based pathway screen. [electronic resource] by
- Mallinger, Aurélie
- Crumpler, Simon
- Pichowicz, Mark
- Waalboer, Dennis
- Stubbs, Mark
- Adeniji-Popoola, Olajumoke
- Wood, Bozena
- Smith, Elizabeth
- Thai, Ching
- Henley, Alan T
- Georgi, Katrin
- Court, William
- Hobbs, Steve
- Box, Gary
- Ortiz-Ruiz, Maria-Jesus
- Valenti, Melanie
- De Haven Brandon, Alexis
- TePoele, Robert
- Leuthner, Birgitta
- Workman, Paul
- Aherne, Wynne
- Poeschke, Oliver
- Dale, Trevor
- Wienke, Dirk
- Esdar, Christina
- Rohdich, Felix
- Raynaud, Florence
- Clarke, Paul A
- Eccles, Suzanne A
- Stieber, Frank
- Schiemann, Kai
- Blagg, Julian
Producer: 20150507
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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