Results
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Diastereoselective synthesis and configuration-dependent activity of (3-substituted-cycloalkyl)glycine pyrrolidides and thiazolidides as dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Ashton, Wallace T
- Dong, Hong
- Sisco, Rosemary M
- Doss, George A
- Leiting, Barbara
- Patel, Reshma A
- Wu, Joseph K
- Marsilio, Frank
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20040928
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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5.
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Discovery of new binding elements in DPP-4 inhibition and their applications in novel DPP-4 inhibitor design. [electronic resource] by
- Liang, Gui-Bai
- Qian, Xiaoxia
- Biftu, Tesfaye
- Singh, Suresh
- Gao, Ying-Duo
- Scapin, Giovanna
- Patel, Sangita
- Leiting, Barbara
- Patel, Reshma
- Wu, Joseph
- Zhang, Xiaoping
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20080916
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetes. [electronic resource] by
- Chen, Ping
- Caldwell, Charles G
- Mathvink, Robert J
- Leiting, Barbara
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- He, Huaibing
- Lyons, Kathryn A
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Xu, Jinyou
- Wei, Lan
- Mathvink, Robert
- He, Jiafang
- Park, You-Jung
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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8.
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Dipeptidyl peptidase IV inhibitors derived from beta-aminoacylpiperidines bearing a fused thiazole, oxazole, isoxazole, or pyrazole. [electronic resource] by
- Ashton, Wallace T
- Sisco, Rosemary M
- Dong, Hong
- Lyons, Kathryn A
- He, Huaibing
- Doss, George A
- Leiting, Barbara
- Patel, Reshma A
- Wu, Joseph K
- Marsilio, Frank
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20050930
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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Optimization of 1,4-diazepan-2-one containing dipeptidyl peptidase IV inhibitors for the treatment of type 2 diabetes. [electronic resource] by
- Liang, Gui-Bai
- Qian, Xiaoxia
- Feng, Dennis
- Biftu, Tesfaye
- Eiermann, George
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathy
- Petrov, Aleksandr
- Sinha-Roy, Ranabir
- Zhang, Bei
- Wu, Joseph
- Zhang, Xiaoping
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20070725
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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10.
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Design, synthesis, and biological evaluation of triazolopiperazine-based beta-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors. [electronic resource] by
- Kowalchick, Jennifer E
- Leiting, Barbara
- Pryor, KellyAnn D
- Marsilio, Frank
- Wu, Joseph K
- He, Huaibing
- Lyons, Kathryn A
- Eiermann, George J
- Petrov, Aleksandr
- Scapin, Giovanna
- Patel, Reshma A
- Thornberry, Nancy A
- Weber, Ann E
- Kim, Dooseop
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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11.
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Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Cox, Jason M
- Harper, Bart
- Mastracchio, Anthony
- Leiting, Barbara
- Sinha Roy, Ranabir
- Patel, Reshma A
- Wu, Joseph K
- Lyons, Kathryn A
- He, Huaibing
- Xu, Shiyao
- Zhu, Bing
- Thornberry, Nancy A
- Weber, Ann E
- Edmondson, Scott D
Producer: 20071121
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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12.
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Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: close analogs of JANUVIA (sitagliptin phosphate). [electronic resource] by
- Kim, Dooseop
- Kowalchick, Jennifer E
- Edmondson, Scott D
- Mastracchio, Anthony
- Xu, Jinyou
- Eiermann, George J
- Leiting, Barbara
- Wu, Joseph K
- Pryor, KellyAnn D
- Patel, Reshma A
- He, Huaibing
- Lyons, Kathryn A
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20070830
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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13.
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Substituted piperazines as novel dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Brockunier, Linda L
- He, Jiafang
- Colwell, Lawrence F
- Habulihaz, Bahanu
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Teffera, Yohannes
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Parmee, Emma R
Producer: 20050307
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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14.
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Fluoropyrrolidine amides as dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Caldwell, Charles G
- Chen, Ping
- He, Jiafang
- Parmee, Emma R
- Leiting, Barbara
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Eiermann, George J
- Petrov, Aleksandr
- He, Huaibing
- Lyons, Kathryn A
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20041012
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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15.
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4-arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV. [electronic resource] by
- Kaelin, David E
- Smenton, Abigail L
- Eiermann, George J
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Alexsandr
- Scapin, Giovanna
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Duffy, Joseph L
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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16.
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4-aminophenylalanine and 4-aminocyclohexylalanine derivatives as potent, selective, and orally bioavailable inhibitors of dipeptidyl peptidase IV. [electronic resource] by
- Duffy, Joseph L
- Kirk, Brian A
- Wang, Liping
- Eiermann, George J
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Alexsandr
- Scapin, Giovanna
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20070730
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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17.
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Discovery of potent and selective beta-homophenylalanine based dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Xu, Jinyou
- Ok, Hyun O
- Gonzalez, Edward J
- Colwell, Lawrence F
- Habulihaz, Bahanu
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Parmee, Emma R
Producer: 20050307
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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18.
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Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors. [electronic resource] by
- Xu, Jinyou
- Wei, Lan
- Mathvink, Robert
- Edmondson, Scott D
- Mastracchio, Anthony
- Eiermann, George J
- He, Huaibing
- Leone, Joseph F
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Petrov, Aleksandr
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20060323
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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19.
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Discovery of potent and selective orally bioavailable beta-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Edmondson, Scott D
- Mastracchio, Anthony
- Duffy, Joseph L
- Eiermann, George J
- He, Huaibing
- Ita, Ida
- Leiting, Barbara
- Leone, Joseph F
- Lyons, Kathryn A
- Makarewicz, Amanda M
- Patel, Reshma A
- Petrov, Aleksandr
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20050919
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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20.
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Potent and selective proline derived dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Edmondson, Scott D
- Mastracchio, Anthony
- Beconi, Maria
- Colwell, Lawrence F
- Habulihaz, Bahanu
- He, Huaibing
- Kumar, Sanjeev
- Leiting, Barbara
- Lyons, Kathryn A
- Mao, Ann
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Zhu, Lan
- Thornberry, Nancy A
- Weber, Ann E
- Parmee, Emma R
Producer: 20050404
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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