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Synthesis and biological activity of a novel series of indole-derived PPARgamma agonists. [electronic resource] by
- Henke, B R
- Adkison, K K
- Blanchard, S G
- Leesnitzer, L M
- Mook, R A
- Plunket, K D
- Ray, J A
- Roberson, C
- Unwalla, R
- Willson, T M
Producer: 20000113
In:
Bioorganic & medicinal chemistry letters vol. 9
Availability: No items available.
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Identification of a series of PPAR gamma/delta dual agonists via solid-phase parallel synthesis. [electronic resource] by
- Liu, K G
- Lambert, M H
- Leesnitzer, L M
- Oliver, W
- Ott, R J
- Plunket, K D
- Stuart, L W
- Brown, P J
- Willson, T M
- Sternbach, D D
Producer: 20020115
In:
Bioorganic & medicinal chemistry letters vol. 11
Availability: No items available.
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6.
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Synthesis and biological activity of L-tyrosine-based PPARgamma agonists with reduced molecular weight. [electronic resource] by
- Liu, K G
- Lambert, M H
- Ayscue, A H
- Henke, B R
- Leesnitzer, L M
- Oliver, W R
- Plunket, K D
- Xu, H E
- Sternbach, D D
- Willson, T M
Producer: 20020226
In:
Bioorganic & medicinal chemistry letters vol. 11
Availability: No items available.
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7.
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A synthetic triterpenoid, 2-cyano-3,12-dioxooleana-1,9-dien-28-oic acid (CDDO), is a ligand for the peroxisome proliferator-activated receptor gamma. [electronic resource] by
- Wang, Y
- Porter, W W
- Suh, N
- Honda, T
- Gribble, G W
- Leesnitzer, L M
- Plunket, K D
- Mangelsdorf, D J
- Blanchard, S G
- Willson, T M
- Sporn, M B
Producer: 20010208
In:
Molecular endocrinology (Baltimore, Md.) vol. 14
Availability: No items available.
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A unique PPARgamma ligand with potent insulin-sensitizing yet weak adipogenic activity. [electronic resource] by
- Rocchi, S
- Picard, F
- Vamecq, J
- Gelman, L
- Potier, N
- Zeyer, D
- Dubuquoy, L
- Bac, P
- Champy, M F
- Plunket, K D
- Leesnitzer, L M
- Blanchard, S G
- Desreumaux, P
- Moras, D
- Renaud, J P
- Auwerx, J
Producer: 20011207
In:
Molecular cell vol. 8
Availability: No items available.
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N-(2-Benzoylphenyl)-L-tyrosine PPARgamma agonists. 2. Structure-activity relationship and optimization of the phenyl alkyl ether moiety. [electronic resource] by
- Collins, J L
- Blanchard, S G
- Boswell, G E
- Charifson, P S
- Cobb, J E
- Henke, B R
- Hull-Ryde, E A
- Kazmierski, W M
- Lake, D H
- Leesnitzer, L M
- Lehmann, J
- Lenhard, J M
- Orband-Miller, L A
- Gray-Nunez, Y
- Parks, D J
- Plunkett, K D
- Tong, W Q
Producer: 19990107
In:
Journal of medicinal chemistry vol. 41
Availability: No items available.
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10.
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N-(2-Benzoylphenyl)-L-tyrosine PPARgamma agonists. 1. Discovery of a novel series of potent antihyperglycemic and antihyperlipidemic agents. [electronic resource] by
- Henke, B R
- Blanchard, S G
- Brackeen, M F
- Brown, K K
- Cobb, J E
- Collins, J L
- Harrington, W W
- Hashim, M A
- Hull-Ryde, E A
- Kaldor, I
- Kliewer, S A
- Lake, D H
- Leesnitzer, L M
- Lehmann, J M
- Lenhard, J M
- Orband-Miller, L A
- Miller, J F
- Mook, R A
- Noble, S A
- Oliver, W
- Parks, D J
- Plunket, K D
- Szewczyk, J R
- Willson, T M
Producer: 19990107
In:
Journal of medicinal chemistry vol. 41
Availability: No items available.
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