Results
|
1.
|
|
|
2.
|
Thieno[3,2-d]pyrimidin-4(3H)-one derivatives as PDK1 inhibitors discovered by fragment-based screening. [electronic resource] by
- Lee, Angeline C-H
- Ramanujulu, Pondy Murugappan
- Poulsen, Anders
- Williams, Meredith
- Blanchard, Stéphanie
- Ma, Diana M
- Bonday, Zahid
- Goh, Kay Lin
- Goh, Kee Chuan
- Goh, Miah Kiat
- Wood, Jeanette
- Dymock, Brian W
Producer: 20120925
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
|
|
3.
|
Synthesis and evaluation of alkenyl indazoles as selective Aurora kinase inhibitors. [electronic resource] by
- Blanchard, Stéphanie
- William, Anthony D
- Lee, Angeline C-H
- Poulsen, Anders
- Teo, Ee Ling
- Deng, Weiping
- Tu, Noah
- Tan, Evelyn
- Goh, Kay Lin
- Ong, Wai Chung
- Ng, Chee Pang
- Goh, Kee Chuan
- Bonday, Zahid
- Sun, Eric T
Producer: 20100812
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
|
|
4.
|
Discovery of the macrocycle (9E)-15-(2-(pyrrolidin-1-yl)ethoxy)-7,12,25-trioxa-19,21,24-triaza-tetracyclo[18.3.1.1(2,5).1(14,18)]hexacosa-1(24),2,4,9,14(26),15,17,20,22-nonaene (SB1578), a potent inhibitor of janus kinase 2/fms-like tyrosine kinase-3 (JAK2/FLT3) for the treatment of rheumatoid arthritis. [electronic resource] by
- William, Anthony D
- Lee, Angeline C-H
- Poulsen, Anders
- Goh, Kee Chuan
- Madan, Babita
- Hart, Stefan
- Tan, Evelyn
- Wang, Haishan
- Nagaraj, Harish
- Chen, Dizhong
- Lee, Chai Ping
- Sun, Eric T
- Jayaraman, Ramesh
- Pasha, Mohammad Khalid
- Ethirajulu, Kantharaj
- Wood, Jeanette M
- Dymock, Brian W
Producer: 20120727
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
|
|
5.
|
Discovery of kinase spectrum selective macrocycle (16E)-14-methyl-20-oxa-5,7,14,26-tetraazatetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8(27),9,11,16,21,23-decaene (SB1317/TG02), a potent inhibitor of cyclin dependent kinases (CDKs), Janus kinase 2 (JAK2), and fms-like tyrosine kinase-3 (FLT3) for the treatment of cancer. [electronic resource] by
- William, Anthony D
- Lee, Angeline C-H
- Goh, Kee Chuan
- Blanchard, Stéphanie
- Poulsen, Anders
- Teo, Ee Ling
- Nagaraj, Harish
- Lee, Chai Ping
- Wang, Haishan
- Williams, Meredith
- Sun, Eric T
- Hu, Changyong
- Jayaraman, Ramesh
- Pasha, Mohammed Khalid
- Ethirajulu, Kantharaj
- Wood, Jeanette M
- Dymock, Brian W
Producer: 20120326
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
|
|
6.
|
Discovery of the macrocycle 11-(2-pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene (SB1518), a potent Janus kinase 2/fms-like tyrosine kinase-3 (JAK2/FLT3) inhibitor for the treatment of myelofibrosis and lymphoma. [electronic resource] by
- William, Anthony D
- Lee, Angeline C-H
- Blanchard, Stéphanie
- Poulsen, Anders
- Teo, Ee Ling
- Nagaraj, Harish
- Tan, Evelyn
- Chen, Dizhong
- Williams, Meredith
- Sun, Eric T
- Goh, Kee Chuan
- Ong, Wai Chung
- Goh, Siok Kun
- Hart, Stefan
- Jayaraman, Ramesh
- Pasha, Mohammed Khalid
- Ethirajulu, Kantharaj
- Wood, Jeanette M
- Dymock, Brian W
Producer: 20110923
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
|