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Structure-based design and parallel synthesis of N-benzyl isatin oximes as JNK3 MAP kinase inhibitors. [electronic resource] by
- Cao, Jingrong
- Gao, Huai
- Bemis, Guy
- Salituro, Francesco
- Ledeboer, Mark
- Harrington, Edmund
- Wilke, Susanne
- Taslimi, Paul
- Pazhanisamy, S
- Xie, Xiaoling
- Jacobs, Marc
- Green, Jeremy
Producer: 20090629
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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4.
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A novel chemotype of kinase inhibitors: Discovery of 3,4-ring fused 7-azaindoles and deazapurines as potent JAK2 inhibitors. [electronic resource] by
- Wang, Tiansheng
- Ledeboer, Mark W
- Duffy, John P
- Salituro, Francesco G
- Pierce, Albert C
- Zuccola, Harmon J
- Block, Eric
- Shlyakter, Dina
- Hogan, James K
- Bennani, Youssef L
Producer: 20100506
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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5.
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Discovery of a Potent and Selective TRPC5 Inhibitor, Efficacious in a Focal Segmental Glomerulosclerosis Model. [electronic resource] by
- Yu, Maolin
- Ledeboer, Mark W
- Daniels, Matthew
- Malojcic, Goran
- Tibbitts, Thomas T
- Coeffet-Le Gal, Marie
- Pan-Zhou, Xin-Ru
- Westerling-Bui, Amy
- Beconi, Maria
- Reilly, John F
- Mundel, Peter
- Harmange, Jean-Christophe
Publication details: ACS medicinal chemistry letters Nov 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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Isosteric replacements of the carboxylic acid of drug candidate VX-787: Effect of charge on antiviral potency and kinase activity of azaindole-based influenza PB2 inhibitors. [electronic resource] by
- Boyd, Michael J
- Bandarage, Upul K
- Bennett, Hamilton
- Byrn, Randal R
- Davies, Ioana
- Gu, Wenxin
- Jacobs, Marc
- Ledeboer, Mark W
- Ledford, Brian
- Leeman, Joshua R
- Perola, Emanuele
- Wang, Tiansheng
- Bennani, Youssef
- Clark, Michael P
- Charifson, Paul S
Producer: 20160219
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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7.
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Preclinical activity of VX-787, a first-in-class, orally bioavailable inhibitor of the influenza virus polymerase PB2 subunit. [electronic resource] by
- Byrn, Randal A
- Jones, Steven M
- Bennett, Hamilton B
- Bral, Chris
- Clark, Michael P
- Jacobs, Marc D
- Kwong, Ann D
- Ledeboer, Mark W
- Leeman, Joshua R
- McNeil, Colleen F
- Murcko, Mark A
- Nezami, Azin
- Perola, Emanuele
- Rijnbrand, Rene
- Saxena, Kumkum
- Tsai, Alice W
- Zhou, Yi
- Charifson, Paul S
Producer: 20151202
In:
Antimicrobial agents and chemotherapy vol. 59
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Discovery of Highly Isoform Selective Thiazolopiperidine Inhibitors of Phosphoinositide 3-Kinase γ. [electronic resource] by
- Collier, Philip N
- Messersmith, David
- Le Tiran, Arnaud
- Bandarage, Upul K
- Boucher, Christina
- Come, Jon
- Cottrell, Kevin M
- Damagnez, Veronique
- Doran, John D
- Griffith, James P
- Khare-Pandit, Suvarna
- Krueger, Elaine B
- Ledeboer, Mark W
- Ledford, Brian
- Liao, Yusheng
- Mahajan, Sudipta
- Moody, Cameron S
- Roday, Setu
- Wang, Tiansheng
- Xu, Jinwang
- Aronov, Alex M
Producer: 20151012
In:
Journal of medicinal chemistry vol. 58
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9.
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2-Aminopyrazolo[1,5-a]pyrimidines as potent and selective inhibitors of JAK2. [electronic resource] by
- Ledeboer, Mark W
- Pierce, Albert C
- Duffy, John P
- Gao, Huai
- Messersmith, David
- Salituro, Francesco G
- Nanthakumar, Suganthini
- Come, Jon
- Zuccola, Harmon J
- Swenson, Lora
- Shlyakter, Dina
- Mahajan, Sudipta
- Hoock, Thomas
- Fan, Bin
- Tsai, Wan-Jung
- Kolaczkowski, Elaine
- Carrier, Scott
- Hogan, James K
- Zessis, Richard
- Pazhanisamy, S
- Bennani, Youssef L
Producer: 20100119
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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10.
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Novel 2-Substituted 7-Azaindole and 7-Azaindazole Analogues as Potential Antiviral Agents for the Treatment of Influenza. [electronic resource] by
- Bandarage, Upul K
- Clark, Michael P
- Perola, Emanuele
- Gao, Huai
- Jacobs, Marc D
- Tsai, Alice
- Gillespie, Jeffery
- Kennedy, Joseph M
- Maltais, François
- Ledeboer, Mark W
- Davies, Ioana
- Gu, Wenxin
- Byrn, Randal A
- Nti Addae, Kwame
- Bennett, Hamilton
- Leeman, Joshua R
- Jones, Steven M
- O'Brien, Colleen
- Memmott, Christine
- Bennani, Youssef
- Charifson, Paul S
Publication details: ACS medicinal chemistry letters Feb 2017
In:
ACS medicinal chemistry letters vol. 8
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11.
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Janus kinase 2 inhibitors. Synthesis and characterization of a novel polycyclic azaindole. [electronic resource] by
- Wang, Tiansheng
- Duffy, John P
- Wang, Jian
- Halas, Summer
- Salituro, Francesco G
- Pierce, Albert C
- Zuccola, Harmon J
- Black, James R
- Hogan, James K
- Jepson, Scott
- Shlyakter, Dina
- Mahajan, Sudipta
- Gu, Yong
- Hoock, Thomas
- Wood, Mark
- Furey, Brinley F
- Frantz, J Daniel
- Dauffenbach, Lisa M
- Germann, Ursula A
- Fan, Bin
- Namchuk, Mark
- Bennani, Youssef L
- Ledeboer, Mark W
Producer: 20100106
In:
Journal of medicinal chemistry vol. 52
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12.
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Discovery of Novel, Orally Bioavailable β-Amino Acid Azaindole Inhibitors of Influenza PB2. [electronic resource] by
- Farmer, Luc J
- Clark, Michael P
- Boyd, Michael J
- Perola, Emanuele
- Jones, Steven M
- Tsai, Alice
- Jacobs, Marc D
- Bandarage, Upul K
- Ledeboer, Mark W
- Wang, Tiansheng
- Deng, Hongbo
- Ledford, Brian
- Gu, Wenxin
- Duffy, John P
- Bethiel, Randy S
- Shannon, Dean
- Byrn, Randal A
- Leeman, Joshua R
- Rijnbrand, Rene
- Bennett, Hamilton B
- O'Brien, Colleen
- Memmott, Christine
- Nti-Addae, Kwame
- Bennani, Youssef L
- Charifson, Paul S
Publication details: ACS medicinal chemistry letters Feb 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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13.
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Discovery of a novel, first-in-class, orally bioavailable azaindole inhibitor (VX-787) of influenza PB2. [electronic resource] by
- Clark, Michael P
- Ledeboer, Mark W
- Davies, Ioana
- Byrn, Randal A
- Jones, Steven M
- Perola, Emanuele
- Tsai, Alice
- Jacobs, Marc
- Nti-Addae, Kwame
- Bandarage, Upul K
- Boyd, Michael J
- Bethiel, Randy S
- Court, John J
- Deng, Hongbo
- Duffy, John P
- Dorsch, Warren A
- Farmer, Luc J
- Gao, Huai
- Gu, Wenxin
- Jackson, Katrina
- Jacobs, Dylan H
- Kennedy, Joseph M
- Ledford, Brian
- Liang, Jianglin
- Maltais, François
- Murcko, Mark
- Wang, Tiansheng
- Wannamaker, M Woods
- Bennett, Hamilton B
- Leeman, Joshua R
- McNeil, Colleen
- Taylor, William P
- Memmott, Christine
- Jiang, Min
- Rijnbrand, Rene
- Bral, Christopher
- Germann, Ursula
- Nezami, Azin
- Zhang, Yuegang
- Salituro, Francesco G
- Bennani, Youssef L
- Charifson, Paul S
Producer: 20150207
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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14.
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Discovery of VX-509 (Decernotinib): A Potent and Selective Janus Kinase 3 Inhibitor for the Treatment of Autoimmune Diseases. [electronic resource] by
- Farmer, Luc J
- Ledeboer, Mark W
- Hoock, Thomas
- Arnost, Michael J
- Bethiel, Randy S
- Bennani, Youssef L
- Black, James J
- Brummel, Christopher L
- Chakilam, Ananthsrinivas
- Dorsch, Warren A
- Fan, Bin
- Cochran, John E
- Halas, Summer
- Harrington, Edmund M
- Hogan, James K
- Howe, David
- Huang, Hui
- Jacobs, Dylan H
- Laitinen, Leena M
- Liao, Shengkai
- Mahajan, Sudipta
- Marone, Valerie
- Martinez-Botella, Gabriel
- McCarthy, Pamela
- Messersmith, David
- Namchuk, Mark
- Oh, Luke
- Penney, Marina S
- Pierce, Albert C
- Raybuck, Scott A
- Rugg, Arthur
- Salituro, Francesco G
- Saxena, Kumkum
- Shannon, Dean
- Shlyakter, Dina
- Swenson, Lora
- Tian, Shi-Kai
- Town, Christopher
- Wang, Jian
- Wang, Tiansheng
- Wannamaker, M Woods
- Winquist, Raymond J
- Zuccola, Harmon J
Producer: 20151229
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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