Preclinical pharmacokinetic, toxicological and biomarker evaluation of SR16157, a novel dual-acting steroid sulfatase inhibitor and selective estrogen receptor modulator. [electronic resource]
Producer: 20110722Description: 1341-52 p. digitalISSN:- 1432-0843
- Administration, Oral
- Animals
- Antineoplastic Agents, Hormonal -- pharmacokinetics
- Biological Availability
- Biomarkers -- blood
- Dogs
- Dose-Response Relationship, Drug
- Female
- Leukocytes, Mononuclear -- cytology
- Male
- Norpregnatrienes -- pharmacokinetics
- Rats
- Rats, Inbred F344
- Selective Estrogen Receptor Modulators -- pharmacokinetics
- Species Specificity
- Steryl-Sulfatase -- antagonists & inhibitors
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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