Results
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2.
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Benzothiophene piperazine and piperidine urea inhibitors of fatty acid amide hydrolase (FAAH). [electronic resource] by
- Johnson, Douglas S
- Ahn, Kay
- Kesten, Suzanne
- Lazerwith, Scott E
- Song, Yuntao
- Morris, Mark
- Fay, Lorraine
- Gregory, Tracy
- Stiff, Cory
- Dunbar, James B
- Liimatta, Marya
- Beidler, David
- Smith, Sarah
- Nomanbhoy, Tyzoon K
- Cravatt, Benjamin F
Producer: 20090629
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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3.
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A small-molecule inhibitor of hepatitis C virus infectivity. [electronic resource] by
- Bush, Caroline O
- Pokrovskii, Maria V
- Saito, Roland
- Morganelli, Philip
- Canales, Eda
- Clarke, Michael O
- Lazerwith, Scott E
- Golde, Justin
- Reid, Brian G
- Babaoglu, Kerim
- Pagratis, Nikos
- Zhong, Weidong
- Delaney, William E
- Paulson, Matthew S
- Beran, Rudolf K F
Producer: 20140918
In:
Antimicrobial agents and chemotherapy vol. 58
Availability: No items available.
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4.
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Discovery of PF-04457845: A Highly Potent, Orally Bioavailable, and Selective Urea FAAH Inhibitor. [electronic resource] by
- Johnson, Douglas S
- Stiff, Cory
- Lazerwith, Scott E
- Kesten, Suzanne R
- Fay, Lorraine K
- Morris, Mark
- Beidler, David
- Liimatta, Marya B
- Smith, Sarah E
- Dudley, David T
- Sadagopan, Nalini
- Bhattachar, Shobha N
- Kesten, Stephen J
- Nomanbhoy, Tyzoon K
- Cravatt, Benjamin F
- Ahn, Kay
Publication details: ACS medicinal chemistry letters Feb 2011
In:
ACS medicinal chemistry letters vol. 2
Availability: No items available.
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5.
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Antiviral Activity of Bictegravir (GS-9883), a Novel Potent HIV-1 Integrase Strand Transfer Inhibitor with an Improved Resistance Profile. [electronic resource] by
- Tsiang, Manuel
- Jones, Gregg S
- Goldsmith, Joshua
- Mulato, Andrew
- Hansen, Derek
- Kan, Elaine
- Tsai, Luong
- Bam, Rujuta A
- Stepan, George
- Stray, Kirsten M
- Niedziela-Majka, Anita
- Yant, Stephen R
- Yu, Helen
- Kukolj, George
- Cihlar, Tomas
- Lazerwith, Scott E
- White, Kirsten L
- Jin, Haolun
Producer: 20170919
In:
Antimicrobial agents and chemotherapy vol. 60
Availability: No items available.
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6.
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Optimization of Pharmacokinetics through Manipulation of Physicochemical Properties in a Series of HCV Inhibitors. [electronic resource] by
- Lazerwith, Scott E
- Bahador, Gina
- Canales, Eda
- Cheng, Guofeng
- Chong, Lee
- Clarke, Michael O
- Doerffler, Edward
- Eisenberg, Eugene J
- Hayes, Jaclyn
- Lu, Bing
- Liu, Qi
- Matles, Mike
- Mertzman, Michael
- Mitchell, Michael L
- Morganelli, Philip
- Murray, Bernard P
- Robinson, Margaret
- Strickley, Robert G
- Tessler, Megan
- Tirunagari, Neeraj
- Wang, Jianhong
- Wang, Yujin
- Zhang, Jennifer R
- Zheng, Xubin
- Zhong, Weidong
- Watkins, William J
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 2
Availability: No items available.
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7.
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Discovery of GS-9669, a thumb site II non-nucleoside inhibitor of NS5B for the treatment of genotype 1 chronic hepatitis C infection. [electronic resource] by
- Lazerwith, Scott E
- Lew, Willard
- Zhang, Jennifer
- Morganelli, Philip
- Liu, Qi
- Canales, Eda
- Clarke, Michael O
- Doerffler, Edward
- Byun, Daniel
- Mertzman, Michael
- Ye, Hong
- Chong, Lee
- Xu, Lianhong
- Appleby, Todd
- Chen, Xiaowu
- Fenaux, Martijn
- Hashash, Ahmad
- Leavitt, Stephanie A
- Mabery, Eric
- Matles, Mike
- Mwangi, Judy W
- Tian, Yang
- Lee, Yu-Jen
- Zhang, Jingyu
- Zhu, Christine
- Murray, Bernard P
- Watkins, William J
Producer: 20140515
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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8.
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Preclinical characterization of GS-9669, a thumb site II inhibitor of the hepatitis C virus NS5B polymerase. [electronic resource] by
- Fenaux, Martijn
- Eng, Stacey
- Leavitt, Stephanie A
- Lee, Yu-Jen
- Mabery, Eric M
- Tian, Yang
- Byun, Daniel
- Canales, Eda
- Clarke, Michael O
- Doerffler, Edward
- Lazerwith, Scott E
- Lew, Willard
- Liu, Qi
- Mertzman, Michael
- Morganelli, Philip
- Xu, Lianhong
- Ye, Hong
- Zhang, Jennifer
- Matles, Mike
- Murray, Bernard P
- Mwangi, Judy
- Zhang, Jingyu
- Hashash, Ahmad
- Krawczyk, Steve H
- Bidgood, Alison M
- Appleby, Todd C
- Watkins, William J
Producer: 20130729
In:
Antimicrobial agents and chemotherapy vol. 57
Availability: No items available.
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