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Inhibition of 3-phosphoglycerate dehydrogenase (PHGDH) by indole amides abrogates de novo serine synthesis in cancer cells. [electronic resource] by
- Mullarky, Edouard
- Xu, Jiayi
- Robin, Anita D
- Huggins, David J
- Jennings, Andy
- Noguchi, Naoyoshi
- Olland, Andrea
- Lakshminarasimhan, Damodharan
- Miller, Michael
- Tomita, Daisuke
- Michino, Mayako
- Su, Taojunfeng
- Zhang, Guoan
- Stamford, Andrew W
- Meinke, Peter T
- Kargman, Stacia
- Cantley, Lewis C
Producer: 20200915
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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6.
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Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. [electronic resource] by
- Kharenko, Olesya A
- Patel, Reena G
- Brown, S David
- Calosing, Cyrus
- White, Andre
- Lakshminarasimhan, Damodharan
- Suto, Robert K
- Duffy, Bryan C
- Kitchen, Douglas B
- McLure, Kevin G
- Hansen, Henrik C
- van der Horst, Edward H
- Young, Peter R
Producer: 20191014
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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7.
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Discovery of a new chemical series of BRD4(1) inhibitors using protein-ligand docking and structure-guided design. [electronic resource] by
- Duffy, Bryan C
- Liu, Shuang
- Martin, Gregory S
- Wang, Ruifang
- Hsia, Ming Min
- Zhao, He
- Guo, Cheng
- Ellis, Michael
- Quinn, John F
- Kharenko, Olesya A
- Norek, Karen
- Gesner, Emily M
- Young, Peter R
- McLure, Kevin G
- Wagner, Gregory S
- Lakshminarasimhan, Damodharan
- White, Andre
- Suto, Robert K
- Hansen, Henrik C
- Kitchen, Douglas B
Producer: 20160307
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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8.
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Exploiting an Asp-Glu "switch" in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia. [electronic resource] by
- Wagner, Florence F
- Benajiba, Lina
- Campbell, Arthur J
- Weïwer, Michel
- Sacher, Joshua R
- Gale, Jennifer P
- Ross, Linda
- Puissant, Alexandre
- Alexe, Gabriela
- Conway, Amy
- Back, Morgan
- Pikman, Yana
- Galinsky, Ilene
- DeAngelo, Daniel J
- Stone, Richard M
- Kaya, Taner
- Shi, Xi
- Robers, Matthew B
- Machleidt, Thomas
- Wilkinson, Jennifer
- Hermine, Olivier
- Kung, Andrew
- Stein, Adam J
- Lakshminarasimhan, Damodharan
- Hemann, Michael T
- Scolnick, Edward
- Zhang, Yan-Ling
- Pan, Jen Q
- Stegmaier, Kimberly
- Holson, Edward B
Producer: 20190923
In:
Science translational medicine vol. 10
Availability: No items available.
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9.
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Non-homeostatic body weight regulation through a brainstem-restricted receptor for GDF15. [electronic resource] by
- Hsu, Jer-Yuan
- Crawley, Suzanne
- Chen, Michael
- Ayupova, Dina A
- Lindhout, Darrin A
- Higbee, Jared
- Kutach, Alan
- Joo, William
- Gao, Zhengyu
- Fu, Diana
- To, Carmen
- Mondal, Kalyani
- Li, Betty
- Kekatpure, Avantika
- Wang, Marilyn
- Laird, Teresa
- Horner, Geoffrey
- Chan, Jackie
- McEntee, Michele
- Lopez, Manuel
- Lakshminarasimhan, Damodharan
- White, Andre
- Wang, Sheng-Ping
- Yao, Jun
- Yie, Junming
- Matern, Hugo
- Solloway, Mark
- Haldankar, Raj
- Parsons, Thomas
- Tang, Jie
- Shen, Wenyan D
- Alice Chen, Yu
- Tian, Hui
- Allan, Bernard B
Producer: 20180227
In:
Nature vol. 550
Availability: No items available.
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10.
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Erratum: Non-homeostatic body weight regulation through a brainstem-restricted receptor for GDF15. [electronic resource] by
- Hsu, Jer-Yuan
- Crawley, Suzanne
- Chen, Michael
- Ayupova, Dina A
- Lindhout, Darrin A
- Higbee, Jared
- Kutach, Alan
- Joo, William
- Gao, Zhengyu
- Fu, Diana
- To, Carmen
- Mondal, Kalyani
- Li, Betty
- Kekatpure, Avantika
- Wang, Marilyn
- Laird, Teresa
- Horner, Geoffrey
- Chan, Jackie
- McEntee, Michele
- Lopez, Manuel
- Lakshminarasimhan, Damodharan
- White, Andre
- Wang, Sheng-Ping
- Yao, Jun
- Yie, Junming
- Matern, Hugo
- Solloway, Mark
- Haldankar, Raj
- Parsons, Thomas
- Tang, Jie
- Shen, Wenyan D
- Alice Chen, Yu
- Tian, Hui
- Allan, Bernard B
Publication details: Nature 11 2017
In:
Nature vol. 551
Availability: No items available.
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