Results
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1.
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Substituted phenyl as a steroid A-ring mimetic: providing agonist activity to a class of arylsulfonamide nonsteroidal glucocorticoid ligands. [electronic resource] by
- DiSalvo, Darren
- Kuzmich, Daniel
- Bentzien, Jörg
- Regan, John
- Kukulka, Alison
- Fadra-Khan, Tazmeen
- Nelson, Richard
- Harcken, Christian
- Thomson, David
- Nabozny, Gerald
Producer: 20140725
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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2.
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Function-regulating pharmacophores in a sulfonamide class of glucocorticoid receptor agonists. [electronic resource] by
- Kuzmich, Daniel
- Bentzien, Jörg
- Betageri, Raj
- DiSalvo, Darren
- Fadra-Khan, Tazmeen
- Harcken, Christian
- Kukulka, Alison
- Nabozny, Gerald
- Nelson, Richard
- Pack, Edward
- Souza, Donald
- Thomson, David
Producer: 20140725
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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3.
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Identification of dissociated non-steroidal glucocorticoid receptor agonists. [electronic resource] by
- Kuzmich, Daniel
- Kirrane, Tom
- Proudfoot, John
- Bekkali, Younes
- Zindell, Renee
- Beck, Laura
- Nelson, Richard
- Shih, Cheng-Kon
- Kukulka, Alison J
- Paw, Zofia
- Reilly, Patty
- Deleon, Rodney
- Cardozo, Mario
- Nabozny, Gerald
- Thomson, David
Producer: 20071227
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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4.
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Trifluoromethyl group as a pharmacophore: effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand. [electronic resource] by
- Betageri, Raj
- Zhang, Yan
- Zindell, Renee M
- Kuzmich, Daniel
- Kirrane, Thomas M
- Bentzien, Jörg
- Cardozo, Mario
- Capolino, Alison J
- Fadra, Tazmeen N
- Nelson, Richard M
- Paw, Zofia
- Shih, Daw-Tsun
- Shih, Cheng-Kon
- Zuvela-Jelaska, Ljiljana
- Nabozny, Gerald
- Thomson, David S
Producer: 20051223
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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5.
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Identification of highly efficacious glucocorticoid receptor agonists with a potential for reduced clinical bone side effects. [electronic resource] by
- Harcken, Christian
- Riether, Doris
- Kuzmich, Daniel
- Liu, Pingrong
- Betageri, Raj
- Ralph, Mark
- Emmanuel, Michel
- Reeves, Jonathan T
- Berry, Angela
- Souza, Donald
- Nelson, Richard M
- Kukulka, Alison
- Fadra, Tazmeen N
- Zuvela-Jelaska, Ljiljana
- Dinallo, Roger
- Bentzien, Jörg
- Nabozny, Gerald H
- Thomson, David S
Producer: 20140429
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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6.
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Nonsteroidal dissociated glucocorticoid agonists containing azaindoles as steroid A-ring mimetics. [electronic resource] by
- Riether, Doris
- Harcken, Christian
- Razavi, Hossein
- Kuzmich, Daniel
- Gilmore, Thomas
- Bentzien, Jörg
- Pack, Edward J
- Souza, Donald
- Nelson, Richard M
- Kukulka, Alison
- Fadra, Tazmeen N
- Zuvela-Jelaska, Ljiljana
- Pelletier, Josephine
- Dinallo, Roger
- Panzenbeck, Mark
- Torcellini, Carol
- Nabozny, Gerald H
- Thomson, David S
Producer: 20101011
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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7.
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Quinol-4-ones as steroid A-ring mimetics in nonsteroidal dissociated glucocorticoid agonists. [electronic resource] by
- Regan, John
- Lee, Thomas W
- Zindell, Renée M
- Bekkali, Younes
- Bentzien, Jörg
- Gilmore, Thomas
- Hammach, Abdelhakim
- Kirrane, Thomas M
- Kukulka, Alison J
- Kuzmich, Daniel
- Nelson, Richard M
- Proudfoot, John R
- Ralph, Mark
- Pelletier, Josephine
- Souza, Donald
- Zuvela-Jelaska, Lijiljana
- Nabozny, Gerald
- Thomson, David S
Producer: 20070202
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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8.
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G protein-coupled bile acid receptor 1 stimulation mediates arterial vasodilation through a K(Ca)1.1 (BK(Ca))-dependent mechanism. [electronic resource] by
- Fryer, Ryan M
- Ng, Khing Jow
- Nodop Mazurek, Suzanne G
- Patnaude, Lori
- Skow, Donna J
- Muthukumarana, Akalushi
- Gilpin, Kyle E
- Dinallo, Roger M
- Kuzmich, Daniel
- Lord, John
- Sanyal, Sulagna
- Yu, Hui
- Harcken, Christian
- Cerny, Matthew A
- Cerny, Matthew C
- Hickey, Eugene R
- Modis, Louise K
Producer: 20140402
In:
The Journal of pharmacology and experimental therapeutics vol. 348
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9.
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A GPBAR1 (TGR5) small molecule agonist shows specific inhibitory effects on myeloid cell activation in vitro and reduces experimental autoimmune encephalitis (EAE) in vivo. [electronic resource] by
- Lewis, Nuruddeen D
- Patnaude, Lori A
- Pelletier, Josephine
- Souza, Donald J
- Lukas, Susan M
- King, F James
- Hill, Jonathan D
- Stefanopoulos, Dimitria E
- Ryan, Kelli
- Desai, Sudha
- Skow, Donna
- Kauschke, Stefan G
- Broermann, Andre
- Kuzmich, Daniel
- Harcken, Christian
- Hickey, Eugene R
- Modis, Louise K
Producer: 20151007
In:
PloS one vol. 9
Availability: No items available.
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10.
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Identification of novel azaindazole CCR1 antagonist clinical candidates. [electronic resource] by
- Harcken, Christian
- Kuzmich, Daniel
- Cook, Brain
- Mao, Can
- Disalvo, Darren
- Razavi, Hossein
- Swinamer, Alan
- Liu, Pingrong
- Zhang, Qiang
- Kukulka, Alison
- Skow, Donna
- Patel, Mita
- Patel, Monica
- Fletcher, Kimberly
- Sherry, Tara
- Joseph, David
- Smith, Dustin
- Canfield, Melissa
- Souza, Donald
- Bogdanffy, Matthew
- Berg, Karen
- Brown, Maryanne
Producer: 20191209
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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11.
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CCR1 plays a critical role in modulating pain through hematopoietic and non-hematopoietic cells. [electronic resource] by
- Lewis, Nuruddeen D
- Muthukumarana, Akalushi
- Fogal, Steven E
- Corradini, Laura
- Stefanopoulos, Dimitria E
- Adusumalli, Prathima
- Pelletier, Josephine
- Panzenbeck, Mark
- Berg, Karen
- Canfield, Melissa
- Cook, Brian N
- Razavi, Hossein
- Kuzmich, Daniel
- Anderson, Shawn
- Allard, Devan
- Harrison, Paul
- Grimaldi, Christine
- Souza, Donald
- Harcken, Christian
- Fryer, Ryan M
- Modis, Louise K
- Brown, Maryanne L
Producer: 20150626
In:
PloS one vol. 9
Availability: No items available.
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12.
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Second-generation lymphocyte function-associated antigen-1 inhibitors: 1H-imidazo[1,2-alpha]imidazol-2-one derivatives. [electronic resource] by
- Wu, Jiang-Ping
- Emeigh, Jonathan
- Gao, Donghong A
- Goldberg, Daniel R
- Kuzmich, Daniel
- Miao, Clara
- Potocki, Ian
- Qian, Kevin C
- Sorcek, Ronald J
- Jeanfavre, Deborah D
- Kishimoto, Kei
- Mainolfi, Elizabeth A
- Nabozny, Gerald
- Peng, Charline
- Reilly, Patricia
- Rothlein, Robert
- Sellati, Rosemarie H
- Woska, Joseph R
- Chen, Shirlynn
- Gunn, Jocelyn A
- O'Brien, Drane
- Norris, Stephen H
- Kelly, Terence A
Producer: 20041203
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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13.
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Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores. [electronic resource] by
- Betageri, Raj
- Gilmore, Thomas
- Kuzmich, Daniel
- Kirrane, Thomas M
- Bentzien, Jörg
- Wiedenmayer, Dieter
- Bekkali, Younes
- Regan, John
- Berry, Angela
- Latli, Bachir
- Kukulka, Alison J
- Fadra, Tazmeen N
- Nelson, Richard M
- Goldrick, Susan
- Zuvela-Jelaska, Ljiljana
- Souza, Don
- Pelletier, Josephine
- Dinallo, Roger
- Panzenbeck, Mark
- Torcellini, Carol
- Lee, Heewon
- Pack, Edward
- Harcken, Christian
- Nabozny, Gerald
- Thomson, David S
Producer: 20120213
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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14.
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Late-stage optimization of a tercyclic class of S1P3-sparing, S1P1 receptor agonists. [electronic resource] by
- Horan, Joshua C
- Kuzmich, Daniel
- Liu, Pingrong
- DiSalvo, Darren
- Lord, John
- Mao, Can
- Hopkins, Tamara D
- Yu, Hui
- Harcken, Christian
- Betageri, Raj
- Hill-Drzewi, Melissa
- Patenaude, Lori
- Patel, Monica
- Fletcher, Kimberly
- Terenzzio, Donna
- Linehan, Brian
- Xia, Heather
- Patel, Mita
- Studwell, Debbie
- Miller, Craig
- Hickey, Eugene
- Levin, Jeremy I
- Smith, Dustin
- Kemper, Raymond A
- Modis, Louise K
- Bannen, Lynne C
- Chan, Diva S
- Mac, Morrison B
- Ng, Stephanie
- Wang, Yong
- Xu, Wei
- Lemieux, René M
Producer: 20170116
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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