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Pyrrolidine-carboxamides and oxadiazoles as potent hNK1 antagonists. [electronic resource] by
- Young, Jonathan R
- Eid, Ronsar
- Turner, Cherilyn
- DeVita, Robert J
- Kurtz, Marc M
- Tsao, Kwei-Lan C
- Chicchi, Gary G
- Wheeldon, Alan
- Carlson, Emma
- Mills, Sander G
Producer: 20071127
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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5.
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NK1 antagonists based on seven membered lactam scaffolds. [electronic resource] by
- Elliott, Jason M
- Carlson, Emma J
- Chicchi, Gary G
- Dirat, Olivier
- Dominguez, Maria
- Gerhard, Ute
- Jelley, Richard
- Jones, A Brian
- Kurtz, Marc M
- Tsao, Kwei lan
- Wheeldon, Alan
Producer: 20060802
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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6.
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Tetrahydroindolizinone NK1 antagonists. [electronic resource] by
- Bao, Jianming
- Lu, Huagang
- Morriello, Gregori J
- Carlson, Emma J
- Wheeldon, Alan
- Chicchi, Gary G
- Kurtz, Marc M
- Tsao, Kwei-Lan C
- Zheng, Song
- Tong, Xinchun
- Mills, Sander G
- DeVita, Robert J
Producer: 20100705
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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7.
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Spirocyclic NK(1) antagonists I: [4.5] and [5.5]-spiroketals. [electronic resource] by
- Seward, Eileen M
- Carlson, Emma
- Harrison, Timothy
- Haworth, Karen R
- Herbert, Richard
- Kelleher, Fintan J
- Kurtz, Marc M
- Moseley, Jonathan
- Owen, Simon N
- Owens, Andrew P
- Sadowski, Sharon J
- Swain, Christopher J
- Williams, Brian J
Producer: 20030211
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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8.
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4,4-Disubstituted cyclohexylamine NK(1) receptor antagonists I. [electronic resource] by
- Elliott, Jason M
- Castro, Jose L
- Chicchi, Gary G
- Cooper, Laura C
- Dinnell, Kevin
- Hollingworth, Gregory J
- Ridgill, Mark P
- Rycroft, Wayne
- Kurtz, Marc M
- Shaw, Duncan E
- Swain, Christopher J
- Tsao, Kwei-Lan
- Yang, Lihu
Producer: 20021119
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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9.
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4,4-Disubstituted cyclohexylamine NK(1) receptor antagonists II. [electronic resource] by
- Cooper, Laura C
- Carlson, Emma J
- Castro, Jose L
- Chicchi, Gary G
- Dinnell, Kevin
- Di Salvo, Jerry
- Elliott, Jason M
- Hollingworth, Gregory J
- Kurtz, Marc M
- Ridgill, Mark P
- Rycroft, Wayne
- Tsao, Kwei-Lan
- Swain, Christopher J
Producer: 20021119
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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10.
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Comparison of the functional blockade of rat substance P (NK1) receptors by GR205171, RP67580, SR140333 and NKP-608. [electronic resource] by
- Rupniak, Nadia M J
- Carlson, Emma J
- Shepheard, Sara
- Bentley, Graham
- Williams, Angela R
- Hill, Alastair
- Swain, Christopher
- Mills, Sander G
- Di Salvo, Jerry
- Kilburn, Ruth
- Cascieri, Margaret A
- Kurtz, Marc M
- Tsao, Kwei-Lan
- Gould, Sandra L
- Chicchi, Gary G
Producer: 20030916
In:
Neuropharmacology vol. 45
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11.
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Novel lactam NK1 antagonists with anti-emetic activity. [electronic resource] by
- Hollingworth, Gregory J
- Carlson, Emma J
- Castro, José L
- Chicchi, Gary G
- Clark, Natalie
- Cooper, Laura C
- Dirat, Olivier
- Salvo, Jerry Di
- Elliott, Jason M
- Kilburn, Ruth
- Kurtz, Marc M
- Rycroft, Wayne
- Tattersall, F David
- Tsao, Kwei-Lan
- Swain, Christopher J
Producer: 20060323
In:
Bioorganic & medicinal chemistry letters vol. 16
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12.
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Fused bicyclic pyrrolizinones as new scaffolds for human NK1 antagonists. [electronic resource] by
- Morriello, Gregori J
- Devita, Robert J
- Mills, Sander G
- Young, Jonathan R
- Lin, Peter
- Doss, George
- Chicchi, Gary G
- Demartino, Julie
- Kurtz, Marc M
- Tsao, Kwei-Lan C
- Carlson, Emma
- Townson, Karen
- Wheeldon, Alan
- Boyce, Susan
- Collinson, Neil
- Rupniak, Nadia
- Moore, Stephen
Producer: 20080514
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
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13.
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Discovery of MK-8722: A Systemic, Direct Pan-Activator of AMP-Activated Protein Kinase. [electronic resource] by
- Feng, Danqing
- Biftu, Tesfaye
- Romero, F Anthony
- Kekec, Ahmet
- Dropinski, James
- Kassick, Andrew
- Xu, Shiyao
- Kurtz, Marc M
- Gollapudi, Anantha
- Shao, Qing
- Yang, Xiaodong
- Lu, Ku
- Zhou, Gaochao
- Kemp, Daniel
- Myers, Robert W
- Guan, Hong-Ping
- Trujillo, Maria E
- Li, Cai
- Weber, Ann
- Sebhat, Iyassu K
Publication details: ACS medicinal chemistry letters Jan 2018
In:
ACS medicinal chemistry letters vol. 9
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14.
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The discovery of potent, selective, and orally bioavailable hNK1 antagonists derived from pyrrolidine. [electronic resource] by
- Lin, Peter
- Chang, Lehua
- Devita, Robert J
- Young, Jonathan R
- Eid, Ronsar
- Tong, Xinchun
- Zheng, Song
- Ball, Richard G
- Tsou, Nancy N
- Chicchi, Gary G
- Kurtz, Marc M
- Tsao, Kwei-Lan C
- Wheeldon, Alan
- Carlson, Emma J
- Eng, Waisi
- Burns, H Donald
- Hargreaves, Richard J
- Mills, Sander G
Producer: 20071227
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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15.
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High-throughput simultaneous analysis of RNA, protein, and lipid biomarkers in heterogeneous tissue samples. [electronic resource] by
- Reiser, Vladimír
- Smith, Ryan C
- Xue, Jiyan
- Kurtz, Marc M
- Liu, Rong
- Legrand, Cheryl
- He, Xuanmin
- Yu, Xiang
- Wong, Peggy
- Hinchcliffe, John S
- Tanen, Michael R
- Lazar, Gloria
- Zieba, Renata
- Ichetovkin, Marina
- Chen, Zhu
- O'Neill, Edward A
- Tanaka, Wesley K
- Marton, Matthew J
- Liao, Jason
- Morris, Mark
- Hailman, Eric
- Tokiwa, George Y
- Plump, Andrew S
Producer: 20111215
In:
Clinical chemistry vol. 57
Availability: No items available.
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16.
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Potent, brain-penetrant, hydroisoindoline-based human neurokinin-1 receptor antagonists. [electronic resource] by
- Jiang, Jinlong
- Bunda, Jaime L
- Doss, Geoge A
- Chicchi, Gary G
- Kurtz, Marc M
- Tsao, Kwei-Lan C
- Tong, Xinchun
- Zheng, Song
- Upthagrove, Alana
- Samuel, Koppara
- Tschirret-Guth, Richard
- Kumar, Sanjeev
- Wheeldon, Alan
- Carlson, Emma J
- Hargreaves, Richard
- Burns, Donald
- Hamill, Terence
- Ryan, Christine
- Krause, Stephen M
- Eng, WaiSi
- DeVita, Robert J
- Mills, Sander G
Producer: 20090602
In:
Journal of medicinal chemistry vol. 52
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17.
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Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver. [electronic resource] by
- Muise, Eric S
- Guan, Hong-Ping
- Liu, Jinqi
- Nawrocki, Andrea R
- Yang, Xiaodong
- Wang, Chuanlin
- Rodríguez, Carlos G
- Zhou, Dan
- Gorski, Judith N
- Kurtz, Marc M
- Feng, Danqing
- Leavitt, Kenneth J
- Wei, Lan
- Wilkening, Robert R
- Apgar, James M
- Xu, Shiyao
- Lu, Ku
- Feng, Wen
- Li, Ying
- He, Huaibing
- Previs, Stephen F
- Shen, Xiaolan
- van Heek, Margaret
- Souza, Sandra C
- Rosenbach, Mark J
- Biftu, Tesfaye
- Erion, Mark D
- Kelley, David E
- Kemp, Daniel M
- Myers, Robert W
- Sebhat, Iyassu K
Producer: 20191202
In:
PloS one vol. 14
Availability: No items available.
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18.
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Systemic pan-AMPK activator MK-8722 improves glucose homeostasis but induces cardiac hypertrophy. [electronic resource] by
- Myers, Robert W
- Guan, Hong-Ping
- Ehrhart, Juliann
- Petrov, Aleksandr
- Prahalada, Srinivasa
- Tozzo, Effie
- Yang, Xiaodong
- Kurtz, Marc M
- Trujillo, Maria
- Gonzalez Trotter, Dinko
- Feng, Danqing
- Xu, Shiyao
- Eiermann, George
- Holahan, Marie A
- Rubins, Daniel
- Conarello, Stacey
- Niu, Xiaoda
- Souza, Sandra C
- Miller, Corin
- Liu, Jinqi
- Lu, Ku
- Feng, Wen
- Li, Ying
- Painter, Ronald E
- Milligan, James A
- He, Huaibing
- Liu, Franklin
- Ogawa, Aimie
- Wisniewski, Douglas
- Rohm, Rory J
- Wang, Liyang
- Bunzel, Michelle
- Qian, Ying
- Zhu, Wei
- Wang, Hongwu
- Bennet, Bindu
- LaFranco Scheuch, Lisa
- Fernandez, Guillermo E
- Li, Cai
- Klimas, Michael
- Zhou, Gaochao
- van Heek, Margaret
- Biftu, Tesfaye
- Weber, Ann
- Kelley, David E
- Thornberry, Nancy
- Erion, Mark D
- Kemp, Daniel M
- Sebhat, Iyassu K
Producer: 20180108
In:
Science (New York, N.Y.) vol. 357
Availability: No items available.
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