Results
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1.
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Glucocorticoid receptor antagonism by cyproterone acetate and RU486. [electronic resource] by
- Honer, Christian
- Nam, Kiyean
- Fink, Cynthia
- Marshall, Paul
- Ksander, Gary
- Chatelain, Ricardo E
- Cornell, Wendy
- Steele, Ronald
- Schweitzer, Robert
- Schumacher, Christoph
Producer: 20030513
In:
Molecular pharmacology vol. 63
Availability: No items available.
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2.
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Structure of neprilysin in complex with the active metabolite of sacubitril. [electronic resource] by
- Schiering, Nikolaus
- D'Arcy, Allan
- Villard, Frederic
- Ramage, Paul
- Logel, Claude
- Cumin, Frederic
- Ksander, Gary M
- Wiesmann, Christian
- Karki, Rajeshri G
- Mogi, Muneto
Producer: 20180806
In:
Scientific reports vol. 6
Availability: No items available.
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3.
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Dipeptide sulfonamides as endothelin ETA/ETB receptor antagonists. [electronic resource] by
- Ksander, Gary M
- Shetty, Suraj S
- DelGrande, Dominick
- Balwierczak, Joseph L
- Bruseo, Charles W
- Savage, Paula
- deJesus, Reynalda
- Yuan, Andrew
- Webb, Randy L
- Jeng, Arco Y
Producer: 20021210
In:
Canadian journal of physiology and pharmacology vol. 80
Availability: No items available.
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4.
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Pharmacokinetics and pharmacodynamics of LCZ696, a novel dual-acting angiotensin receptor-neprilysin inhibitor (ARNi). [electronic resource] by
- Gu, Jessie
- Noe, Adele
- Chandra, Priya
- Al-Fayoumi, Suliman
- Ligueros-Saylan, Monica
- Sarangapani, Ramesh
- Maahs, Suzanne
- Ksander, Gary
- Rigel, Dean F
- Jeng, Arco Y
- Lin, Tsu-Han
- Zheng, Weiyi
- Dole, William P
Producer: 20100929
In:
Journal of clinical pharmacology vol. 50
Availability: No items available.
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5.
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The discovery of potent inhibitors of aldosterone synthase that exhibit selectivity over 11-beta-hydroxylase. [electronic resource] by
- Adams, Christopher M
- Hu, Chii-Whei
- Jeng, Arco Y
- Karki, Rajeshri
- Ksander, Gary
- Lasala, Dan
- Leung-Chu, Jennifer
- Liang, Guiqing
- Liu, Qian
- Meredith, Erik
- Rao, Chang
- Rigel, Dean F
- Shi, Jie
- Smith, Sherri
- Springer, Clayton
- Zhang, Chun
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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Discovery and in Vivo Evaluation of Potent Dual CYP11B2 (Aldosterone Synthase) and CYP11B1 Inhibitors. [electronic resource] by
- Meredith, Erik L
- Ksander, Gary
- Monovich, Lauren G
- Papillon, Julien P N
- Liu, Qian
- Miranda, Karl
- Morris, Patrick
- Rao, Chang
- Burgis, Robin
- Capparelli, Michael
- Hu, Qi-Ying
- Singh, Alok
- Rigel, Dean F
- Jeng, Arco Y
- Beil, Michael
- Fu, Fumin
- Hu, Chii-Whei
- LaSala, Daniel
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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7.
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Discovery of N-[5-(6-Chloro-3-cyano-1-methyl-1H-indol-2-yl)-pyridin-3-ylmethyl]-ethanesulfonamide, a Cortisol-Sparing CYP11B2 Inhibitor that Lowers Aldosterone in Human Subjects. [electronic resource] by
- Papillon, Julien P N
- Lou, Changgang
- Singh, Alok K
- Adams, Christopher M
- Ksander, Gary M
- Beil, Michael E
- Chen, Wei
- Leung-Chu, Jennifer
- Fu, Fumin
- Gan, Lu
- Hu, Chii-Whei
- Jeng, Arco Y
- LaSala, Daniel
- Liang, Guiqing
- Rigel, Dean F
- Russell, Kerry S
- Vest, John A
- Watson, Catherine
Producer: 20160412
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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8.
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Structure-Activity Relationships, Pharmacokinetics, and in Vivo Activity of CYP11B2 and CYP11B1 Inhibitors. [electronic resource] by
- Papillon, Julien P N
- Adams, Christopher M
- Hu, Qi-Ying
- Lou, Changgang
- Singh, Alok K
- Zhang, Chun
- Carvalho, Jose
- Rajan, Srinivan
- Amaral, Adam
- Beil, Michael E
- Fu, Fumin
- Gangl, Eric
- Hu, Chii-Whei
- Jeng, Arco Y
- LaSala, Daniel
- Liang, Guiqing
- Logman, Michael
- Maniara, Wieslawa M
- Rigel, Dean F
- Smith, Sherri A
- Ksander, Gary M
Producer: 20150928
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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9.
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Structure-Guided Design of Substituted Biphenyl Butanoic Acid Derivatives as Neprilysin Inhibitors. [electronic resource] by
- Kawanami, Toshio
- Karki, Rajeshri G
- Cody, Emma
- Liu, Qian
- Liang, Guiqing
- Ksander, Gary M
- Rigel, Dean F
- Schiering, Nikolaus
- Gong, Yongjin
- Coppola, Gary M
- Iwaki, Yuki
- Sun, Robert
- Neubert, Alan
- Fan, Li
- Ingles, Sara
- D'Arcy, Allan
- Villard, Frederic
- Ramage, Paul
- Jeng, Arco Y
- Leung-Chu, Jennifer
- Liu, Jing
- Beil, Michael
- Fu, Fumin
- Chen, Wei
- Cumin, Frederic
- Wiesmann, Christian
- Mogi, Muneto
Publication details: ACS medicinal chemistry letters Feb 2020
In:
ACS medicinal chemistry letters vol. 11
Availability: No items available.
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