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Discovery of GS-9973, a selective and orally efficacious inhibitor of spleen tyrosine kinase. [electronic resource] by
- Currie, Kevin S
- Kropf, Jeffrey E
- Lee, Tony
- Blomgren, Peter
- Xu, Jianjun
- Zhao, Zhongdong
- Gallion, Steve
- Whitney, J Andrew
- Maclin, Deborah
- Lansdon, Eric B
- Maciejewski, Patricia
- Rossi, Ann Marie
- Rong, Hong
- Macaluso, Jennifer
- Barbosa, James
- Di Paolo, Julie A
- Mitchell, Scott A
Producer: 20140710
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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Imidazo[1,2-a]pyrazine diaryl ureas: inhibitors of the receptor tyrosine kinase EphB4. [electronic resource] by
- Mitchell, Scott A
- Danca, Mihaela Diana
- Blomgren, Peter A
- Darrow, James W
- Currie, Kevin S
- Kropf, Jeffrey E
- Lee, Seung H
- Gallion, Steven L
- Xiong, Jin-Ming
- Pippin, Douglas A
- DeSimone, Robert W
- Brittelli, David R
- Eustice, David C
- Bourret, Aaron
- Hill-Drzewi, Melissa
- Maciejewski, Patricia M
- Elkin, Lisa L
Producer: 20100209
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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Discovery of Lanraplenib (GS-9876): A Once-Daily Spleen Tyrosine Kinase Inhibitor for Autoimmune Diseases. [electronic resource] by
- Blomgren, Peter
- Chandrasekhar, Jayaraman
- Di Paolo, Julie A
- Fung, Wanchi
- Geng, Guoju
- Ip, Carmen
- Jones, Randall
- Kropf, Jeffrey E
- Lansdon, Eric B
- Lee, Seung
- Lo, Jennifer R
- Mitchell, Scott A
- Murray, Bernard
- Pohlmeyer, Chris
- Schmitt, Aaron
- Suekawa-Pirrone, Kimberly
- Wise, Sarah
- Xiong, Jin-Ming
- Xu, Jianjun
- Yu, Helen
- Zhao, Zhongdong
- Currie, Kevin S
Publication details: ACS medicinal chemistry letters Apr 2020
In:
ACS medicinal chemistry letters vol. 11
Availability: No items available.
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Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation. [electronic resource] by
- Farand, Julie
- Kropf, Jeffrey E
- Blomgren, Peter
- Xu, Jianjun
- Schmitt, Aaron C
- Newby, Zachary E
- Wang, Ting
- Murakami, Eisuke
- Barauskas, Ona
- Sudhamsu, Jawahar
- Feng, Joy Y
- Niedziela-Majka, Anita
- Schultz, Brian E
- Schwartz, Karen
- Viatchenko-Karpinski, Serge
- Kornyeyev, Dmytro
- Kashishian, Adam
- Fan, Peidong
- Chen, Xiaowu
- Lansdon, Eric B
- Ports, Michael O
- Currie, Kevin S
- Watkins, William J
- Notte, Gregory T
Publication details: ACS medicinal chemistry letters Mar 2020
In:
ACS medicinal chemistry letters vol. 11
Availability: No items available.
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Potent and selective Bruton's tyrosine kinase inhibitors: discovery of GDC-0834. [electronic resource] by
- Young, Wendy B
- Barbosa, James
- Blomgren, Peter
- Bremer, Meire C
- Crawford, James J
- Dambach, Donna
- Gallion, Steve
- Hymowitz, Sarah G
- Kropf, Jeffrey E
- Lee, Seung H
- Liu, Lichuan
- Lubach, Joseph W
- Macaluso, Jen
- Maciejewski, Pat
- Maurer, Brigitte
- Mitchell, Scott A
- Ortwine, Daniel F
- Di Paolo, Julie
- Reif, Karin
- Scheerens, Heleen
- Schmitt, Aaron
- Sowell, C Gregory
- Wang, Xiaojing
- Wong, Harvey
- Xiong, Jin-Ming
- Xu, Jianjun
- Zhao, Zhongdong
- Currie, Kevin S
Producer: 20151228
In:
Bioorganic & medicinal chemistry letters vol. 25
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Discovery of highly potent and selective Bruton's tyrosine kinase inhibitors: Pyridazinone analogs with improved metabolic stability. [electronic resource] by
- Young, Wendy B
- Barbosa, James
- Blomgren, Peter
- Bremer, Meire C
- Crawford, James J
- Dambach, Donna
- Eigenbrot, Charles
- Gallion, Steve
- Johnson, Adam R
- Kropf, Jeffrey E
- Lee, Seung H
- Liu, Lichuan
- Lubach, Joseph W
- Macaluso, Jen
- Maciejewski, Pat
- Mitchell, Scott A
- Ortwine, Daniel F
- Di Paolo, Julie
- Reif, Karin
- Scheerens, Heleen
- Schmitt, Aaron
- Wang, Xiaojing
- Wong, Harvey
- Xiong, Jin-Ming
- Xu, Jianjun
- Yu, Christine
- Zhao, Zhongdong
- Currie, Kevin S
Producer: 20161011
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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9.
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Discovery of Potent and Selective Tricyclic Inhibitors of Bruton's Tyrosine Kinase with Improved Druglike Properties. [electronic resource] by
- Wang, Xiaojing
- Barbosa, James
- Blomgren, Peter
- Bremer, Meire C
- Chen, Jacob
- Crawford, James J
- Deng, Wei
- Dong, Liming
- Eigenbrot, Charles
- Gallion, Steve
- Hau, Jonathon
- Hu, Huiyong
- Johnson, Adam R
- Katewa, Arna
- Kropf, Jeffrey E
- Lee, Seung H
- Liu, Lichuan
- Lubach, Joseph W
- Macaluso, Jen
- Maciejewski, Pat
- Mitchell, Scott A
- Ortwine, Daniel F
- DiPaolo, Julie
- Reif, Karin
- Scheerens, Heleen
- Schmitt, Aaron
- Wong, Harvey
- Xiong, Jin-Ming
- Xu, Jianjun
- Zhao, Zhongdong
- Zhou, Fusheng
- Currie, Kevin S
- Young, Wendy B
Publication details: ACS medicinal chemistry letters Jun 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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Specific Btk inhibition suppresses B cell- and myeloid cell-mediated arthritis. [electronic resource] by
- Di Paolo, Julie A
- Huang, Tao
- Balazs, Mercedesz
- Barbosa, James
- Barck, Kai H
- Bravo, Brandon J
- Carano, Richard A D
- Darrow, James
- Davies, Douglas R
- DeForge, Laura E
- Diehl, Lauri
- Ferrando, Ronald
- Gallion, Steven L
- Giannetti, Anthony M
- Gribling, Peter
- Hurez, Vincent
- Hymowitz, Sarah G
- Jones, Randall
- Kropf, Jeffrey E
- Lee, Wyne P
- Maciejewski, Patricia M
- Mitchell, Scott A
- Rong, Hong
- Staker, Bart L
- Whitney, J Andrew
- Yeh, Sherry
- Young, Wendy B
- Yu, Christine
- Zhang, Juan
- Reif, Karin
- Currie, Kevin S
Producer: 20110118
In:
Nature chemical biology vol. 7
Availability: No items available.
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