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Synthesis and biological evaluation of 2-benzylamino-4(5)-(6-methylpyridin-2-yl)-5(4)-([1,2,4]triazolo[1,5-a]-pyridin-6-yl)thiazoles as transforming growth factor-β type 1 receptor kinase inhibitors. [electronic resource] by
- Krishnaiah, Maddeboina
- Jin, Cheng Hua
- Sreenu, Domalapally
- Subrahmanyam, Vura Bala
- Rao, Kota Sudhakar
- Son, Do-Hyun
- Park, Hyun-Ju
- Kim, Seung Won
- Sheen, Yhun Yhong
- Kim, Dae-Kee
Producer: 20130509
In:
European journal of medicinal chemistry vol. 57
Availability: No items available.
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Synthesis and biological evaluation of 1-substituted-3-(6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors. [electronic resource] by
- Jin, Cheng Hua
- Krishnaiah, Maddeboina
- Sreenu, Domalapally
- Subrahmanyam, Vura Bala
- Rao, Kota Sudhakar
- Mohan, Annaji Venkata Nagendra
- Park, Chul-Yong
- Son, Jee-Yeon
- Sheen, Yhun Yhong
- Kim, Dae-Kee
Producer: 20120118
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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Discovery of N-((4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methyl)-2-fluoroaniline (EW-7197): a highly potent, selective, and orally bioavailable inhibitor of TGF-β type I receptor kinase as cancer immunotherapeutic/antifibrotic agent. [electronic resource] by
- Jin, Cheng Hua
- Krishnaiah, Maddeboina
- Sreenu, Domalapally
- Subrahmanyam, Vura B
- Rao, Kota S
- Lee, Hwa Jeong
- Park, So-Jung
- Park, Hyun-Ju
- Lee, Kiho
- Sheen, Yhun Yhong
- Kim, Dae-Kee
Producer: 20140808
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors. [electronic resource] by
- Jin, Cheng Hua
- Sreenu, Domalapally
- Krishnaiah, Maddeboina
- Subrahmanyam, Vura Bala
- Rao, Kota Sudhakar
- Nagendra Mohan, Annaji Venkata
- Park, Chul-Yong
- Son, Jee-Yeon
- Son, Do-Hyun
- Park, Hyun-Ju
- Sheen, Yhun Yhong
- Kim, Dae-Kee
Producer: 20120103
In:
European journal of medicinal chemistry vol. 46
Availability: No items available.
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