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	1.	Cyclic guanidines as dual 5-HT5A/5-HT7 receptor ligands: structure-activity relationship elucidation. [electronic resource] by Peters, Jens-Uwe Lübbers, Thomas Alanine, Alexander Kolczewski, Sabine Blasco, Francesca Steward, Lucinda Producer: 20080212 In: Bioorganic & medicinal chemistry letters vol. 18 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	2.	Cyclic guanidines as dual 5-HT5A/5-HT7 receptor ligands: optimising brain penetration. [electronic resource] by Peters, Jens-Uwe Lübbers, Thomas Alanine, Alexander Kolczewski, Sabine Blasco, Francesca Steward, Lucinda Producer: 20080212 In: Bioorganic & medicinal chemistry letters vol. 18 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	3.	Parallel solution- and solid-phase synthesis of spirohydantoin derivatives as neurokinin-1 receptor ligands. [electronic resource] by Bleicher, Konrad H Wüthrich, Yves De Boni, Maxime Kolczewski, Sabine Hoffmann, Torsten Sleight, Andrew J Producer: 20030211 In: Bioorganic & medicinal chemistry letters vol. 12 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	4.	Rational design, synthesis, and structure-activity relationship of benzoxazolones: new potent mglu5 receptor antagonists based on the fenobam structure. [electronic resource] by Ceccarelli, Simona M Jaeschke, Georg Buettelmann, Bernd Huwyler, Jörg Kolczewski, Sabine Peters, Jens-Uwe Prinssen, Eric Porter, Richard Spooren, Will Vieira, Eric Producer: 20070515 In: Bioorganic & medicinal chemistry letters vol. 17 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	5.	Functional heterogeneity of nociceptin/orphanin FQ receptors revealed by (+)-5a Compound and Ro 64-6198 in rat periaqueductal grey slices. [electronic resource] by Liao, Yan-Yu Teng, Shu-Fang Lin, Li-Chun Kolczewski, Sabine Prinssen, Eric P Lee, Li-Jen Ho, Ing-Kang Chiou, Lih-Chu Producer: 20111110 In: The international journal of neuropsychopharmacology vol. 14 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	6.	Novel hexahydrospiro[piperidine-4,1'-pyrrolo[3,4-c]pyrroles]: highly selective small-molecule nociceptin/orphanin FQ receptor agonists. [electronic resource] by Kolczewski, Sabine Adam, Geo Cesura, Andrea M Jenck, François Hennig, Michael Oberhauser, Thomas Poli, Sonia M Rössler, Felix Röver, Stephan Wichmann, Jürgen Dautzenberg, Frank M Producer: 20030204 In: Journal of medicinal chemistry vol. 46 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	7.	Arylmethoxypyridines as novel, potent and orally active mGlu5 receptor antagonists. [electronic resource] by Büttelmann, Bernd Peters, Jens-Uwe Ceccarelli, Simona Kolczewski, Sabine Vieira, Eric Prinssen, Eric P Spooren, Will Schuler, Franz Huwyler, Jörg Porter, Richard H P Jaeschke, Georg Producer: 20060719 In: Bioorganic & medicinal chemistry letters vol. 16 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	8.	3-Amido-3-aryl-piperidines: A Novel Class of Potent, Selective, and Orally Active GlyT1 Inhibitors. [electronic resource] by Pinard, Emmanuel Alberati, Daniela Alvarez-Sanchez, Ruben Brom, Virginie Burner, Serge Fischer, Holger Hauser, Nicole Kolczewski, Sabine Lengyel, Judith Mory, Roland Saladin, Christian Schulz-Gasch, Tanja Stalder, Henri Producer: 20140606 In: ACS medicinal chemistry letters vol. 5 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	9.	Asymmetric synthesis and receptor pharmacology of the group II mGlu receptor ligand (1S,2R,3R,5R,6S)-2-amino-3-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid-HYDIA. [electronic resource] by Woltering, Thomas J Adam, Geo Huguenin, Philipp Wichmann, Jürgen Kolczewski, Sabine Gatti, Silvia Bourson, Anne Kew, James N C Richards, Grayson Kemp, John A Mutel, Vincent Knoflach, Frédéric Producer: 20080723 In: ChemMedChem vol. 3 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	10.	Synthesis and biological evaluation of fenobam analogs as mGlu5 receptor antagonists. [electronic resource] by Jaeschke, Georg Porter, Richard Büttelmann, Bernd Ceccarelli, Simona M Guba, Wolfgang Kuhn, Bernd Kolczewski, Sabine Huwyler, Jörg Mutel, Vincent Peters, Jens-Uwe Ballard, Theresa Prinssen, Eric Vieira, Eric Wichmann, Jürgen Spooren, Will Producer: 20070515 In: Bioorganic & medicinal chemistry letters vol. 17 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	11.	Fenobam: a clinically validated nonbenzodiazepine anxiolytic is a potent, selective, and noncompetitive mGlu5 receptor antagonist with inverse agonist activity. [electronic resource] by Porter, Richard H P Jaeschke, Georg Spooren, Will Ballard, Theresa M Büttelmann, Bernd Kolczewski, Sabine Peters, Jens-Uwe Prinssen, Eric Wichmann, Jürgen Vieira, Eric Mühlemann, Andreas Gatti, Silvia Mutel, Vincent Malherbe, Pari Producer: 20060112 In: The Journal of pharmacology and experimental therapeutics vol. 315 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	12.	CTEP: a novel, potent, long-acting, and orally bioavailable metabotropic glutamate receptor 5 inhibitor. [electronic resource] by Lindemann, Lothar Jaeschke, Georg Michalon, Aubin Vieira, Eric Honer, Michael Spooren, Will Porter, Richard Hartung, Thomas Kolczewski, Sabine Büttelmann, Bernd Flament, Christophe Diener, Catherine Fischer, Christophe Gatti, Silvia Prinssen, Eric P Parrott, Neil Hoffmann, Gerhard Wettstein, Joseph G Producer: 20120116 In: The Journal of pharmacology and experimental therapeutics vol. 339 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	13.	Metabolite identification via LC-SPE-NMR-MS of the in vitro biooxidation products of a lead mGlu5 allosteric antagonist and impact on the improvement of metabolic stability in the series. [electronic resource] by Ceccarelli, Simona M Schlotterbeck, Götz Boissin, Patrick Binder, Martin Buettelmann, Bernd Hanlon, Steven Jaeschke, Georg Kolczewski, Sabine Kupfer, Ernst Peters, Jens-Uwe Porter, Richard H P Prinssen, Eric P Rueher, Marianne Ruf, Iris Spooren, Will Stämpfli, Andreas Vieira, Eric Producer: 20080730 In: ChemMedChem vol. 3 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	14.	Zebrafish behavioral profiling identifies multitarget antipsychotic-like compounds. [electronic resource] by Bruni, Giancarlo Rennekamp, Andrew J Velenich, Andrea McCarroll, Matthew Gendelev, Leo Fertsch, Ethan Taylor, Jack Lakhani, Parth Lensen, Dennis Evron, Tama Lorello, Paul J Huang, Xi-Ping Kolczewski, Sabine Carey, Galen Caldarone, Barbara J Prinssen, Eric Roth, Bryan L Keiser, Michael J Peterson, Randall T Kokel, David Producer: 20170515 In: Nature chemical biology vol. 12 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	15.	G protein-coupled receptor transmembrane binding pockets and their applications in GPCR research and drug discovery: a survey. [electronic resource] by Kratochwil, Nicole A Gatti-McArthur, Silvia Hoener, Marius C Lindemann, Lothar Christ, Andreas D Green, Luke G Guba, Wolfgang Martin, Rainer E Malherbe, Pari Porter, Richard H P Slack, Jay P Winnig, Marcel Dehmlow, Henrietta Grether, Uwe Hertel, Cornelia Narquizian, Robert Panousis, Constantinos G Kolczewski, Sabine Steward, Lucinda Producer: 20120224 In: Current topics in medicinal chemistry vol. 11 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	16.	Pharmacology of basimglurant (RO4917523, RG7090), a unique metabotropic glutamate receptor 5 negative allosteric modulator in clinical development for depression. [electronic resource] by Lindemann, Lothar Porter, Richard H Scharf, Sebastian H Kuennecke, Basil Bruns, Andreas von Kienlin, Markus Harrison, Anthony C Paehler, Axel Funk, Christoph Gloge, Andreas Schneider, Manfred Parrott, Neil J Polonchuk, Liudmila Niederhauser, Urs Morairty, Stephen R Kilduff, Thomas S Vieira, Eric Kolczewski, Sabine Wichmann, Juergen Hartung, Thomas Honer, Michael Borroni, Edilio Moreau, Jean-Luc Prinssen, Eric Spooren, Will Wettstein, Joseph G Jaeschke, Georg Producer: 20150509 In: The Journal of pharmacology and experimental therapeutics vol. 353 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	17.	Metabotropic glutamate receptor 5 negative allosteric modulators: discovery of 2-chloro-4-[1-(4-fluorophenyl)-2,5-dimethyl-1H-imidazol-4-ylethynyl]pyridine (basimglurant, RO4917523), a promising novel medicine for psychiatric diseases. [electronic resource] by Jaeschke, Georg Kolczewski, Sabine Spooren, Will Vieira, Eric Bitter-Stoll, Nadia Boissin, Patrick Borroni, Edilio Büttelmann, Bernd Ceccarelli, Simona Clemann, Nicole David, Beatrice Funk, Christoph Guba, Wolfgang Harrison, Anthony Hartung, Thomas Honer, Michael Huwyler, Jörg Kuratli, Martin Niederhauser, Urs Pähler, Axel Peters, Jens-Uwe Petersen, Ann Prinssen, Eric Ricci, Antonio Rueher, Daniel Rueher, Marianne Schneider, Manfred Spurr, Paul Stoll, Theodor Tännler, Daniel Wichmann, Jürgen Porter, Richard H Wettstein, Joseph G Lindemann, Lothar Producer: 20150414 In: Journal of medicinal chemistry vol. 58 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)