Preclinical evaluation of the antifolate QN254, 5-chloro- N'6'-(2,5-dimethoxy-benzyl)-quinazoline-2,4,6-triamine, as an antimalarial drug candidate. [electronic resource]
Producer: 20100914Description: 2603-10 p. digitalISSN:- 1098-6596
- Administration, Oral
- Animals
- Antimalarials -- administration & dosage
- Biological Availability
- Drug Resistance
- Female
- Folic Acid Antagonists -- administration & dosage
- Humans
- In Vitro Techniques
- Malaria -- drug therapy
- Malaria, Falciparum -- drug therapy
- Male
- Mice
- Models, Molecular
- Mutation
- Parasitic Sensitivity Tests
- Plasmodium berghei -- drug effects
- Plasmodium falciparum -- drug effects
- Pyrimethamine -- pharmacology
- Quinazolines -- administration & dosage
- Rats
- Rats, Wistar
- Tetrahydrofolate Dehydrogenase -- chemistry
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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