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Scaffold Morphing Identifies 3-Pyridyl Azetidine Ureas as Inhibitors of Nicotinamide Phosphoribosyltransferase (NAMPT). [electronic resource] by
- Palacios, Daniel S
- Meredith, Erik L
- Kawanami, Toshio
- Adams, Christopher M
- Chen, Xin
- Darsigny, Veronique
- Palermo, Mark
- Baird, Daniel
- George, Elizabeth L
- Guy, Chantale
- Hewett, Jeffrey
- Tierney, Laryssa
- Thigale, Sachin
- Wang, Louis
- Weihofen, Wilhelm A
Publication details: ACS medicinal chemistry letters Nov 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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5.
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Discovery of a Novel Piperidine-Based Inhibitor of Cholesteryl Ester Transfer Protein (CETP) That Retains Activity in Hypertriglyceridemic Plasma. [electronic resource] by
- Yamada, Ken
- Brousseau, Margaret
- Honma, Wataru
- Iimura, Akiko
- Imase, Hidetomo
- Iwaki, Yuki
- Kawanami, Toshio
- LaSala, Daniel
- Liang, Guiqing
- Mitani, Hironobu
- Nonomura, Kazuhiko
- Ohmori, Osamu
- Pan, Meihui
- Rigel, Dean F
- Umemura, Ichiro
- Yasoshima, Kayo
- Zhu, Guoming
- Mogi, Muneto
Producer: 20171121
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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Structure based design of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors from a phenotypic screen. [electronic resource] by
- Palacios, Daniel S
- Meredith, Erik
- Kawanami, Toshio
- Adams, Christopher
- Chen, Xin
- Darsigny, Veronique
- Geno, Erin
- Palermo, Mark
- Baird, Daniel
- Boynton, Geoffrey
- Busby, Scott A
- George, Elizabeth L
- Guy, Chantale
- Hewett, Jeffrey
- Tierney, Laryssa
- Thigale, Sachin
- Weihofen, Wilhelm
- Wang, Louis
- White, Nicole
- Yin, Ming
- Argikar, Upendra A
Producer: 20190530
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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Optimization of Allosteric With-No-Lysine (WNK) Kinase Inhibitors and Efficacy in Rodent Hypertension Models. [electronic resource] by
- Yamada, Ken
- Levell, Julian
- Yoon, Taeyong
- Kohls, Darcy
- Yowe, David
- Rigel, Dean F
- Imase, Hidetomo
- Yuan, Jun
- Yasoshima, Kayo
- DiPetrillo, Keith
- Monovich, Lauren
- Xu, Lingfei
- Zhu, Meicheng
- Kato, Mitsunori
- Jain, Monish
- Idamakanti, Neeraja
- Taslimi, Paul
- Kawanami, Toshio
- Argikar, Upendra A
- Kunjathoor, Vidya
- Xie, Xiaoling
- Yagi, Yukiko I
- Iwaki, Yuki
- Robinson, Zachary
- Park, Hyi-Man
Producer: 20170926
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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Discovery and Characterization of Allosteric WNK Kinase Inhibitors. [electronic resource] by
- Yamada, Ken
- Zhang, Ji-Hu
- Xie, Xiaoling
- Reinhardt, Juergen
- Xie, Amy Qiongshu
- LaSala, Daniel
- Kohls, Darcy
- Yowe, David
- Burdick, Debra
- Yoshisue, Hajime
- Wakai, Hiromichi
- Schmidt, Isabel
- Gunawan, Jason
- Yasoshima, Kayo
- Yue, Q Kimberley
- Kato, Mitsunori
- Mogi, Muneto
- Idamakanti, Neeraja
- Kreder, Natasha
- Drueckes, Peter
- Pandey, Pramod
- Kawanami, Toshio
- Huang, Waanjeng
- Yagi, Yukiko I
- Deng, Zhan
- Park, Hyi-Man
Producer: 20170310
In:
ACS chemical biology vol. 11
Availability: No items available.
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Structure-Guided Design of Substituted Biphenyl Butanoic Acid Derivatives as Neprilysin Inhibitors. [electronic resource] by
- Kawanami, Toshio
- Karki, Rajeshri G
- Cody, Emma
- Liu, Qian
- Liang, Guiqing
- Ksander, Gary M
- Rigel, Dean F
- Schiering, Nikolaus
- Gong, Yongjin
- Coppola, Gary M
- Iwaki, Yuki
- Sun, Robert
- Neubert, Alan
- Fan, Li
- Ingles, Sara
- D'Arcy, Allan
- Villard, Frederic
- Ramage, Paul
- Jeng, Arco Y
- Leung-Chu, Jennifer
- Liu, Jing
- Beil, Michael
- Fu, Fumin
- Chen, Wei
- Cumin, Frederic
- Wiesmann, Christian
- Mogi, Muneto
Publication details: ACS medicinal chemistry letters Feb 2020
In:
ACS medicinal chemistry letters vol. 11
Availability: No items available.
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10.
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Discovery of 4-((2 [electronic resource] by
- Mainolfi, Nello
- Ehara, Takeru
- Karki, Rajeshri G
- Anderson, Karen
- Mac Sweeney, Aengus
- Liao, Sha-Mei
- Argikar, Upendra A
- Jendza, Keith
- Zhang, Chun
- Powers, James
- Klosowski, Daniel W
- Crowley, Maura
- Kawanami, Toshio
- Ding, Jian
- April, Myriam
- Forster, Cornelia
- Serrano-Wu, Michael
- Capparelli, Michael
- Ramqaj, Rrezarta
- Solovay, Catherine
- Cumin, Frederic
- Smith, Thomas M
- Ferrara, Luciana
- Lee, Wendy
- Long, Debby
- Prentiss, Melissa
- De Erkenez, Andrea
- Yang, Louis
- Liu, Fang
- Sellner, Holger
- Sirockin, Finton
- Valeur, Eric
- Erbel, Paulus
- Ostermeier, Daniela
- Ramage, Paul
- Gerhartz, Bernd
- Schubart, Anna
- Flohr, Stefanie
- Gradoux, Nathalie
- Feifel, Roland
- Vogg, Barbara
- Wiesmann, Christian
- Maibaum, Jürgen
- Eder, Jörg
- Sedrani, Richard
- Harrison, Richard A
- Mogi, Muneto
- Jaffee, Bruce D
- Adams, Christopher M
Producer: 20201112
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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