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4-arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV. [electronic resource] by
- Kaelin, David E
- Smenton, Abigail L
- Eiermann, George J
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Alexsandr
- Scapin, Giovanna
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Duffy, Joseph L
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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8.
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Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-5). [electronic resource] by
- Singh, Sheo B
- Kaelin, David E
- Meinke, Peter T
- Wu, Jin
- Miesel, Lynn
- Tan, Christopher M
- Olsen, David B
- Lagrutta, Armando
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Takeuchi, Tomoko
- Takano, Hisashi
- Ohata, Kohei
- Kurasaki, Haruaki
- Nishimura, Akinori
- Shibata, Takeshi
- Fukuda, Yasumichi
Producer: 20160520
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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9.
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Oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad spectrum antibacterial agents. [electronic resource] by
- Singh, Sheo B
- Kaelin, David E
- Wu, Jin
- Miesel, Lynn
- Tan, Christopher M
- Meinke, Peter T
- Olsen, David
- Lagrutta, Armando
- Bradley, Prudence
- Lu, Jun
- Patel, Sangita
- Rickert, Keith W
- Smith, Robert F
- Soisson, Stephen
- Wei, Changqing
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Fukuda, Yasumichi
Producer: 20140606
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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10.
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Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6). [electronic resource] by
- Singh, Sheo B
- Kaelin, David E
- Wu, Jin
- Miesel, Lynn
- Tan, Christopher M
- Meinke, Peter T
- Olsen, David B
- Lagrutta, Armando
- Wei, Changqing
- Liao, Yonggang
- Peng, Xuanjia
- Wang, Xiu
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Yajima, Masanobu
- Shibue, Taku
- Shibata, Takeshi
- Ohata, Kohei
- Nishimura, Akinori
- Fukuda, Yasumichi
Producer: 20160520
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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11.
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Structure activity relationship of substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-4). [electronic resource] by
- Singh, Sheo B
- Kaelin, David E
- Wu, Jin
- Miesel, Lynn
- Tan, Christopher M
- Meinke, Peter T
- Olsen, David B
- Lagrutta, Armando
- Wei, Changqing
- Peng, Xuanjia
- Wang, Xiu
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Shibata, Takeshi
- Ohata, Kohei
- Takano, Hisashi
- Kurasaki, Haruaki
- Takeuchi, Tomoko
- Nishimura, Akinori
- Fukuda, Yasumichi
Producer: 20160217
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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12.
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In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase. [electronic resource] by
- Tan, Christopher M
- Gill, Charles J
- Wu, Jin
- Toussaint, Nathalie
- Yin, Jingjun
- Tsuchiya, Takayuki
- Garlisi, Charles G
- Kaelin, David
- Meinke, Peter T
- Miesel, Lynn
- Olsen, David B
- Lagrutta, Armando
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Oohata, Kouhei
- Takeuchi, Tomoko
- Shibue, Taku
- Takano, Hisashi
- Nishimura, Akinori
- Fukuda, Yasumichi
- Singh, Sheo B
Producer: 20170912
In:
Antimicrobial agents and chemotherapy vol. 60
Availability: No items available.
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13.
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Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3). [electronic resource] by
- Singh, Sheo B
- Kaelin, David E
- Wu, Jin
- Miesel, Lynn
- Tan, Christopher M
- Gill, Charles
- Black, Todd
- Nargund, Ravi
- Meinke, Peter T
- Olsen, David B
- Lagrutta, Armando
- Wei, Changqing
- Peng, Xuanjia
- Wang, Xiu
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Takeuchi, Tomoko
- Shibue, Taku
- Ohata, Kohei
- Takano, Hisashi
- Ban, Shizuka
- Nishimura, Akinori
- Fukuda, Yasumichi
Producer: 20160223
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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14.
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Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2). [electronic resource] by
- Singh, Sheo B
- Kaelin, David E
- Wu, Jin
- Miesel, Lynn
- Tan, Christopher M
- Black, Todd
- Nargund, Ravi
- Meinke, Peter T
- Olsen, David B
- Lagrutta, Armando
- Lu, Jun
- Patel, Sangita
- Rickert, Keith W
- Smith, Robert F
- Soisson, Stephen
- Sherer, Edward
- Joyce, Leo A
- Wei, Changqing
- Peng, Xuanjia
- Wang, Xiu
- Fukuda, Hideyuki
- Kishii, Ryuta
- Takei, Masaya
- Takano, Hisashi
- Shibasaki, Mitsuhito
- Yajima, Masanobu
- Nishimura, Akinori
- Shibata, Takeshi
- Fukuda, Yasumichi
Producer: 20160219
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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