Results
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1.
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Design, synthesis and antifungal activity of a novel water soluble prodrug of antifungal triazole. [electronic resource] by
- Ohwada, Jun
- Tsukazaki, Masao
- Hayase, Tadakatsu
- Oikawa, Nobuhiro
- Isshiki, Yoshiaki
- Fukuda, Hiroshi
- Mizuguchi, Eisaku
- Sakaitani, Masahiro
- Shiratori, Yasuhiko
- Yamazaki, Toshikazu
- Ichihara, Shigeyasu
- Umeda, Isao
- Shimma, Nobuo
Producer: 20030717
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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2.
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Development of a Novel Human Parathyroid Hormone Receptor 1 (hPTHR1) Agonist (CH5447240), a Potent and Orally Available Small Molecule for Treatment of Hypoparathyroidism. [electronic resource] by
- Nishimura, Yoshikazu
- Esaki, Toru
- Isshiki, Yoshiaki
- Okamoto, Naoki
- Furuta, Yoshiyuki
- Kotake, Tomoya
- Watanabe, Yoshiaki
- Ohta, Masateru
- Nakagawa, Toshito
- Noda, Hiroshi
- Shimizu, Masaru
- Saito, Hitoshi
- Tamura, Tatsuya
- Sato, Haruhiko
Producer: 20190624
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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3.
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Design and synthesis of novel prodrugs of 2'-deoxy-2'-methylidenecytidine activated by membrane dipeptidase overexpressed in tumor tissues. [electronic resource] by
- Kohchi, Yasunori
- Hattori, Kazuo
- Oikawa, Nobuhiro
- Mizuguchi, Eisaku
- Isshiki, Yoshiaki
- Aso, Kohsuke
- Yoshinari, Kiyoshi
- Shirai, Haruyoshi
- Miwa, Masanori
- Inagaki, Yukiko
- Ura, Masako
- Ogawa, Kotaroh
- Okabe, Hisafumi
- Ishitsuka, Hideo
- Shimma, Nobuo
Producer: 20070530
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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4.
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Lead Optimization and Avoidance of Reactive Metabolite Leading to PCO371, a Potent, Selective, and Orally Available Human Parathyroid Hormone Receptor 1 (hPTHR1) Agonist. [electronic resource] by
- Nishimura, Yoshikazu
- Esaki, Toru
- Isshiki, Yoshiaki
- Furuta, Yoshiyuki
- Mizutani, Akemi
- Kotake, Tomoya
- Emura, Takashi
- Watanabe, Yoshiaki
- Ohta, Masateru
- Nakagawa, Toshito
- Ogawa, Kotaro
- Arai, Shinichi
- Noda, Hiroshi
- Kitamura, Hidetomo
- Shimizu, Masaru
- Tamura, Tatsuya
- Sato, Haruhiko
Producer: 20201023
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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5.
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Design and synthesis of 2-amino-6-(1H,3H-benzo[de]isochromen-6-yl)-1,3,5-triazines as novel Hsp90 inhibitors. [electronic resource] by
- Suda, Atsushi
- Kawasaki, Ken-ichi
- Komiyama, Susumu
- Isshiki, Yoshiaki
- Yoon, Dong-Oh
- Kim, Sung-Jin
- Na, Young-Jun
- Hasegawa, Kiyoshi
- Fukami, Takaaki A
- Sato, Shigeo
- Miura, Takaaki
- Ono, Naomi
- Yamazaki, Toshikazu
- Saitoh, Ryoichi
- Shimma, Nobuo
- Shiratori, Yasuhiko
- Tsukuda, Takuo
Producer: 20141124
In:
Bioorganic & medicinal chemistry vol. 22
Availability: No items available.
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6.
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Halogen bonding at the active sites of human cathepsin L and MEK1 kinase: efficient interactions in different environments. [electronic resource] by
- Hardegger, Leo A
- Kuhn, Bernd
- Spinnler, Beat
- Anselm, Lilli
- Ecabert, Robert
- Stihle, Martine
- Gsell, Bernard
- Thoma, Ralf
- Diez, Joachim
- Benz, Jörg
- Plancher, Jean-Marc
- Hartmann, Guido
- Isshiki, Yoshiaki
- Morikami, Kenji
- Shimma, Nobuo
- Haap, Wolfgang
- Banner, David W
- Diederich, François
Producer: 20120413
In:
ChemMedChem vol. 6
Availability: No items available.
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7.
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Design and synthesis of novel allosteric MEK inhibitor CH4987655 as an orally available anticancer agent. [electronic resource] by
- Isshiki, Yoshiaki
- Kohchi, Yasunori
- Iikura, Hitoshi
- Matsubara, Yasuaki
- Asoh, Kohsuke
- Murata, Takeshi
- Kohchi, Masami
- Mizuguchi, Eisaku
- Tsujii, Shinji
- Hattori, Kazuo
- Miura, Takaaki
- Yoshimura, Yasushi
- Aida, Satoshi
- Miwa, Masanori
- Saitoh, Ryoichi
- Murao, Naoaki
- Okabe, Hisafumi
- Belunis, Charles
- Janson, Cheryl
- Lukacs, Christine
- Schück, Verena
- Shimma, Nobuo
Producer: 20110705
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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