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A novel and potent poly(ADP-ribose) polymerase-1 inhibitor, FR247304 (5-chloro-2-[3-(4-phenyl-3,6-dihydro-1(2H)-pyridinyl)propyl]-4(3H)-quinazolinone), attenuates neuronal damage in in vitro and in vivo models of cerebral ischemia. [electronic resource] by
- Iwashita, Akinori
- Tojo, Nobuteru
- Matsuura, Shigeru
- Yamazaki, Syunji
- Kamijo, Kazunori
- Ishida, Junya
- Yamamoto, Hirofumi
- Hattori, Kouji
- Matsuoka, Nobuya
- Mutoh, Seitaro
Producer: 20050328
In:
The Journal of pharmacology and experimental therapeutics vol. 310
Availability: No items available.
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Discovery of quinazolinone and quinoxaline derivatives as potent and selective poly(ADP-ribose) polymerase-1/2 inhibitors. [electronic resource] by
- Iwashita, Akinori
- Hattori, Kouji
- Yamamoto, Hirofumi
- Ishida, Junya
- Kido, Yoshiyuki
- Kamijo, Kazunori
- Murano, Kenji
- Miyake, Hiroshi
- Kinoshita, Takayoshi
- Warizaya, Masaichi
- Ohkubo, Mitsuru
- Matsuoka, Nobuya
- Mutoh, Seitaro
Producer: 20050401
In:
FEBS letters vol. 579
Availability: No items available.
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10.
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Discovery of potent and selective PARP-1 and PARP-2 inhibitors: SBDD analysis via a combination of X-ray structural study and homology modeling. [electronic resource] by
- Ishida, Junya
- Yamamoto, Hirofumi
- Kido, Yoshiyuki
- Kamijo, Kazunori
- Murano, Kenji
- Miyake, Hiroshi
- Ohkubo, Mitsuru
- Kinoshita, Takayoshi
- Warizaya, Masaichi
- Iwashita, Akinori
- Mihara, Kayoko
- Matsuoka, Nobuya
- Hattori, Kouji
Producer: 20060502
In:
Bioorganic & medicinal chemistry vol. 14
Availability: No items available.
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Rational approaches to discovery of orally active and brain-penetrable quinazolinone inhibitors of poly(ADP-ribose)polymerase. [electronic resource] by
- Hattori, Kouji
- Kido, Yoshiyuki
- Yamamoto, Hirofumi
- Ishida, Junya
- Kamijo, Kazunori
- Murano, Kenji
- Ohkubo, Mitsuru
- Kinoshita, Takayoshi
- Iwashita, Akinori
- Mihara, Kayoko
- Yamazaki, Syunji
- Matsuoka, Nobuya
- Teramura, Yoshinori
- Miyake, Hiroshi
Producer: 20040830
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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