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A novel inhibitor of I-kappaB kinase beta ameliorates experimental arthritis through downregulation of proinflammatory cytokines in arthritic joints. [electronic resource] by
- Tanaka, Shinji
- Toki, Tadashi
- Yokoyama, Mika
- Shimizu, Hiroki
- Yamasaki, Tomonori
- Yoneda, Yoshiyuki
- Muro, Fumihito
- Yasukochi, Takanori
- Iimura, Shin
- Morishita, Kaoru
Producer: 20140826
In:
Biological & pharmaceutical bulletin vol. 37
Availability: No items available.
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7.
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Discovery of imidazo[1,2-b]pyridazines as IKKβ inhibitors. Part 2: improvement of potency in vitro and in vivo. [electronic resource] by
- Shimizu, Hiroki
- Yasumatsu, Isao
- Hamada, Tomoaki
- Yoneda, Yoshiyuki
- Yamasaki, Tomonori
- Tanaka, Shinji
- Toki, Tadashi
- Yokoyama, Mika
- Morishita, Kaoru
- Iimura, Shin
Producer: 20110502
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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8.
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A novel and potent VLA-4 antagonist based on trans-4-substituted cyclohexanecarboxylic acid. [electronic resource] by
- Muro, Fumihito
- Iimura, Shin
- Yoneda, Yoshiyuki
- Chiba, Jun
- Watanabe, Toshiyuki
- Setoguchi, Masaki
- Takayama, Gensuke
- Yokoyama, Mika
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20090415
In:
Bioorganic & medicinal chemistry vol. 17
Availability: No items available.
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9.
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Discovery of imidazo[1,2-b]pyridazines as IKKβ inhibitors. Part 3: exploration of effective compounds in arthritis models. [electronic resource] by
- Shimizu, Hiroki
- Yamasaki, Tomonori
- Yoneda, Yoshiyuki
- Muro, Fumihito
- Hamada, Tomoaki
- Yasukochi, Takanori
- Tanaka, Shinji
- Toki, Tadashi
- Yokoyama, Mika
- Morishita, Kaoru
- Iimura, Shin
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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10.
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A novel inhibitor stabilizes the inactive conformation of MAPK-interacting kinase 1. [electronic resource] by
- Matsui, Yumi
- Yasumatsu, Isao
- Yoshida, Ken Ichi
- Iimura, Shin
- Ikeno, Yutaka
- Nawano, Takako
- Fukano, Hajime
- Ubukata, Osamu
- Hanzawa, Hiroyuki
- Tanzawa, Fumie
- Isoyama, Takeshi
Producer: 20190201
In:
Acta crystallographica. Section F, Structural biology communications vol. 74
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11.
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Identification of 4-[1-[3-chloro-4-[N'-(5-fluoro-2-methylphenyl)ureido]phenylacetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]benzoic acid as a potent, orally active VLA-4 antagonist. [electronic resource] by
- Muro, Fumihito
- Iimura, Shin
- Yoneda, Yoshiyuki
- Chiba, Jun
- Watanabe, Toshiyuki
- Setoguchi, Masaki
- Iigou, Yutaka
- Takayama, Gensuke
- Yokoyama, Mika
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20090109
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
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12.
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Synthesis and biological evaluation of benzoic acid derivatives as potent, orally active VLA-4 antagonists. [electronic resource] by
- Chiba, Jun
- Iimura, Shin
- Yoneda, Yoshiyuki
- Watanabe, Toshiyuki
- Muro, Fumito
- Tsubokawa, Masao
- Iigou, Yutaka
- Satoh, Atsushi
- Takayama, Gensuke
- Yokoyama, Mika
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20070403
In:
Bioorganic & medicinal chemistry vol. 15
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13.
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Identification of trans-4-[1-[[7-fluoro-2-(1-methyl-3-indolyl)-6-benzoxazolyl]acetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid as a potent, orally active VLA-4 antagonist. [electronic resource] by
- Setoguchi, Masaki
- Iimura, Shin
- Sugimoto, Yuuichi
- Yoneda, Yoshiyuki
- Chiba, Jun
- Watanabe, Toshiyuki
- Muro, Fumihito
- Iigo, Yutaka
- Takayama, Gensuke
- Yokoyama, Mika
- Taira, Tomoe
- Aonuma, Misato
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20120516
In:
Bioorganic & medicinal chemistry vol. 20
Availability: No items available.
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14.
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A novel, potent, and orally active VLA-4 antagonist with good aqueous solubility: trans-4-[1-[[2-(5-Fluoro-2-methylphenylamino)-7-fluoro-6-benzoxazolyl]acetyl]-(5S)-[methoxy(methyl)amino]methyl-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid. [electronic resource] by
- Setoguchi, Masaki
- Iimura, Shin
- Sugimoto, Yuuichi
- Yoneda, Yoshiyuki
- Chiba, Jun
- Watanabe, Toshiyuki
- Muro, Fumihito
- Iigo, Yutaka
- Takayama, Gensuke
- Yokoyama, Mika
- Taira, Tomoe
- Aonuma, Misato
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20130521
In:
Bioorganic & medicinal chemistry vol. 21
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15.
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Discovery of Novel Pyrido-pyridazinone Derivatives as FER Tyrosine Kinase Inhibitors with Antitumor Activity. [electronic resource] by
- Taniguchi, Toru
- Inagaki, Hiroaki
- Baba, Daichi
- Yasumatsu, Isao
- Toyota, Akiko
- Kaneta, Yasuyuki
- Kiga, Masaki
- Iimura, Shin
- Odagiri, Takashi
- Shibata, Yoshihiro
- Ueda, Kiyono
- Seo, Maki
- Shimizu, Hiroki
- Imaoka, Tomoki
- Nakayama, Kiyoshi
Publication details: ACS medicinal chemistry letters May 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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16.
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Discovery of trans-4-[1-[[2,5-Dichloro-4-(1-methyl-3-indolylcarboxamido)phenyl]acetyl]-(4S)-methoxy-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid: an orally active, selective very late antigen-4 antagonist. [electronic resource] by
- Muro, Fumihito
- Iimura, Shin
- Sugimoto, Yuuichi
- Yoneda, Yoshiyuki
- Chiba, Jun
- Watanabe, Toshiyuki
- Setoguchi, Masaki
- Iigou, Yutaka
- Matsumoto, Keiko
- Satoh, Atsushi
- Takayama, Gensuke
- Taira, Tomoe
- Yokoyama, Mika
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20100106
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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17.
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4-(Pyrrolidinyl)methoxybenzoic acid derivatives as a potent, orally active VLA-4 antagonist. [electronic resource] by
- Chiba, Jun
- Iimura, Shin
- Yoneda, Yoshiyuki
- Sugimoto, Yuichi
- Horiuchi, Takao
- Muro, Fumito
- Ochiai, Yuichi
- Ogasawara, Tomomi
- Tsubokawa, Masao
- Iigou, Yutaka
- Takayama, Gensuke
- Taira, Tomoe
- Takata, Yoshimi
- Yokoyama, Mika
- Takashi, Tohru
- Nakayama, Atsushi
- Machinaga, Nobuo
Producer: 20070208
In:
Chemical & pharmaceutical bulletin vol. 54
Availability: No items available.
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18.
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Discovery of 3-(3-(4-(1-Aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine (ARQ 092): An Orally Bioavailable, Selective, and Potent Allosteric AKT Inhibitor. [electronic resource] by
- Lapierre, Jean-Marc
- Eathiraj, Sudharshan
- Vensel, David
- Liu, Yanbin
- Bull, Cathy O
- Cornell-Kennon, Susan
- Iimura, Shin
- Kelleher, Eugene W
- Kizer, Darin E
- Koerner, Steffi
- Makhija, Sapna
- Matsuda, Akihisa
- Moussa, Magdi
- Namdev, Nivedita
- Savage, Ronald E
- Szwaya, Jeff
- Volckova, Erika
- Westlund, Neil
- Wu, Hui
- Schwartz, Brian
Producer: 20170529
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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