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Differential mechanisms of acquired resistance to insulin-like growth factor-i receptor antibody therapy or to a small-molecule inhibitor, BMS-754807, in a human rhabdomyosarcoma model. [electronic resource] by
- Huang, Fei
- Hurlburt, Warren
- Greer, Ann
- Reeves, Karen A
- Hillerman, Stephen
- Chang, Han
- Fargnoli, Joseph
- Graf Finckenstein, Friedrich
- Gottardis, Marco M
- Carboni, Joan M
Producer: 20101019
In:
Cancer research vol. 70
Availability: No items available.
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4.
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IRS2 copy number gain, KRAS and BRAF mutation status as predictive biomarkers for response to the IGF-1R/IR inhibitor BMS-754807 in colorectal cancer cell lines. [electronic resource] by
- Huang, Fei
- Chang, Han
- Greer, Ann
- Hillerman, Stephen
- Reeves, Karen A
- Hurlburt, Warren
- Cogswell, John
- Patel, Dharmesh
- Qi, Zhenhao
- Fairchild, Craig
- Ryseck, Rolf-Peter
- Wong, Tai W
- Finckenstein, Friedrich G
- Jackson, Jeffrey
- Carboni, Joan M
Producer: 20151103
In:
Molecular cancer therapeutics vol. 14
Availability: No items available.
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5.
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The mechanisms of differential sensitivity to an insulin-like growth factor-1 receptor inhibitor (BMS-536924) and rationale for combining with EGFR/HER2 inhibitors. [electronic resource] by
- Huang, Fei
- Greer, Ann
- Hurlburt, Warren
- Han, Xia
- Hafezi, Rameh
- Wittenberg, Gayle M
- Reeves, Karen
- Chen, Jiwen
- Robinson, Douglas
- Li, Aixin
- Lee, Francis Y
- Gottardis, Marco M
- Clark, Edwin
- Helman, Lee
- Attar, Ricardo M
- Dongre, Ashok
- Carboni, Joan M
Producer: 20090130
In:
Cancer research vol. 69
Availability: No items available.
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BMS-754807, a small molecule inhibitor of insulin-like growth factor-1R/IR. [electronic resource] by
- Carboni, Joan M
- Wittman, Mark
- Yang, Zheng
- Lee, Francis
- Greer, Ann
- Hurlburt, Warren
- Hillerman, Stephen
- Cao, Carolyn
- Cantor, Glenn H
- Dell-John, Janet
- Chen, Cliff
- Discenza, Lorell
- Menard, Krista
- Li, Aixin
- Trainor, George
- Vyas, Dolatrai
- Kramer, Robert
- Attar, Ricardo M
- Gottardis, Marco M
Producer: 20100324
In:
Molecular cancer therapeutics vol. 8
Availability: No items available.
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7.
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Discovery and evaluation of 4-(2-(4-chloro-1H-pyrazol-1-yl)ethylamino)-3-(6-(1-(3-fluoropropyl)piperidin-4-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one (BMS-695735), an orally efficacious inhibitor of insulin-like growth factor-1 receptor kinase with broad spectrum in vivo antitumor activity. [electronic resource] by
- Velaparthi, Upender
- Wittman, Mark
- Liu, Peiying
- Carboni, Joan M
- Lee, Francis Y
- Attar, Ricardo
- Balimane, Praveen
- Clarke, Wendy
- Sinz, Michael W
- Hurlburt, Warren
- Patel, Karishma
- Discenza, Lorell
- Kim, Sean
- Gottardis, Marco
- Greer, Ann
- Li, Aixin
- Saulnier, Mark
- Yang, Zheng
- Zimmermann, Kurt
- Trainor, George
- Vyas, Dolatrai
Producer: 20081030
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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8.
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Tumor development by transgenic expression of a constitutively active insulin-like growth factor I receptor. [electronic resource] by
- Carboni, Joan M
- Lee, Adrian V
- Hadsell, Darryl L
- Rowley, Bruce R
- Lee, Francis Y
- Bol, David K
- Camuso, Amy E
- Gottardis, Marco
- Greer, Ann F
- Ho, Ching Ping
- Hurlburt, Warren
- Li, Aixin
- Saulnier, Mark
- Velaparthi, Upender
- Wang, Cindy
- Wen, Mei-Li
- Westhouse, Richard A
- Wittman, Mark
- Zimmermann, Kurt
- Rupnow, Brent A
- Wong, Tai W
Producer: 20050615
In:
Cancer research vol. 65
Availability: No items available.
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9.
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Discovery of a (1H-benzoimidazol-2-yl)-1H-pyridin-2-one (BMS-536924) inhibitor of insulin-like growth factor I receptor kinase with in vivo antitumor activity. [electronic resource] by
- Wittman, Mark
- Carboni, Joan
- Attar, Ricardo
- Balasubramanian, Balu
- Balimane, Praveen
- Brassil, Patrick
- Beaulieu, Francis
- Chang, Chiehying
- Clarke, Wendy
- Dell, Janet
- Eummer, Jeffrey
- Frennesson, David
- Gottardis, Marco
- Greer, Ann
- Hansel, Steven
- Hurlburt, Warren
- Jacobson, Bruce
- Krishnananthan, Subramaniam
- Lee, Francis Y
- Li, Aixin
- Lin, Tai-An
- Liu, Peiying
- Ouellet, Carl
- Sang, Xiaopeng
- Saulnier, Mark G
- Stoffan, Karen
- Sun, Yax
- Velaparthi, Upender
- Wong, Henry
- Yang, Zheng
- Zimmermann, Kurt
- Zoeckler, Mary
- Vyas, Dolatrai
Producer: 20051101
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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10.
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Discovery of a 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitor (BMS-754807) of insulin-like growth factor receptor (IGF-1R) kinase in clinical development. [electronic resource] by
- Wittman, Mark D
- Carboni, Joan M
- Yang, Zheng
- Lee, Francis Y
- Antman, Melissa
- Attar, Ricardo
- Balimane, Praveen
- Chang, Chiehying
- Chen, Cliff
- Discenza, Lorell
- Frennesson, David
- Gottardis, Marco M
- Greer, Ann
- Hurlburt, Warren
- Johnson, Walter
- Langley, David R
- Li, Aixin
- Li, Jianqing
- Liu, Peiying
- Mastalerz, Harold
- Mathur, Arvind
- Menard, Krista
- Patel, Karishma
- Sack, John
- Sang, Xiaopeng
- Saulnier, Mark
- Smith, Daniel
- Stefanski, Kevin
- Trainor, George
- Velaparthi, Upender
- Zhang, Guifen
- Zimmermann, Kurt
- Vyas, Dolatrai M
Producer: 20091231
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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