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Synthesis and SAR of potent LXR agonists containing an indole pharmacophore. [electronic resource] by
- Washburn, David G
- Hoang, Tram H
- Campobasso, Nino
- Smallwood, Angela
- Parks, Derek J
- Webb, Christine L
- Frank, Kelly A
- Nord, Melanie
- Duraiswami, Chaya
- Evans, Christopher
- Jaye, Michael
- Thompson, Scott K
Producer: 20090310
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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8.
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Rational design of orally-active, pyrrolidine-based progesterone receptor partial agonists. [electronic resource] by
- Thompson, Scott K
- Washburn, David G
- Frazee, James S
- Madauss, Kevin P
- Hoang, Tram H
- Lapinski, Leahann
- Grygielko, Eugene T
- Glace, Lindsay E
- Trizna, Walter
- Williams, Shawn P
- Duraiswami, Chaya
- Bray, Jeffrey D
- Laping, Nicholas J
Producer: 20091013
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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9.
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Synthesis and SAR of amino acid-derived heterocyclic progesterone receptor full and partial agonists. [electronic resource] by
- Hammond, Marlys
- Patterson, Jaclyn R
- Manns, Sharada
- Hoang, Tram H
- Washburn, David G
- Trizna, Walter
- Glace, Lindsay
- Grygielko, Eugene T
- Nagilla, Rakesh
- Nord, Melanie
- Fries, Harvey E
- Minick, Douglas J
- Laping, Nicholas J
- Bray, Jeffrey D
- Thompson, Scott K
Producer: 20090629
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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10.
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Discovery of orally active, pyrrolidinone-based progesterone receptor partial agonists. [electronic resource] by
- Washburn, David G
- Hoang, Tram H
- Frazee, James S
- Johnson, Latisha
- Hammond, Marlys
- Manns, Sharada
- Madauss, Kevin P
- Williams, Shawn P
- Duraiswami, Chaya
- Tran, Thuy B
- Stewart, Eugene L
- Grygielko, Eugene T
- Glace, Lindsay E
- Trizna, Walter
- Nagilla, Rakesh
- Bray, Jeffrey D
- Thompson, Scott K
Producer: 20091013
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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11.
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Discovery of GSK2798745: A Clinical Candidate for Inhibition of Transient Receptor Potential Vanilloid 4 (TRPV4). [electronic resource] by
- Brooks, Carl A
- Barton, Linda S
- Behm, David J
- Eidam, Hilary S
- Fox, Ryan M
- Hammond, Marlys
- Hoang, Tram H
- Holt, Dennis A
- Hilfiker, Mark A
- Lawhorn, Brian G
- Patterson, Jaclyn R
- Stoy, Patrick
- Roethke, Theresa J
- Ye, Guosen
- Zhao, Steve
- Thorneloe, Kevin S
- Goodman, Krista B
- Cheung, Mui
Publication details: ACS medicinal chemistry letters Aug 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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12.
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Reverse Hydroxamate Inhibitors of Bone Morphogenetic Protein 1. [electronic resource] by
- Kallander, Lara S
- Washburn, David
- Hilfiker, Mark A
- Eidam, Hilary Schenck
- Lawhorn, Brian G
- Prendergast, Joanne
- Fox, Ryan
- Dowdell, Sarah
- Manns, Sharada
- Hoang, Tram
- Zhao, Steve
- Ye, Guosen
- Hammond, Marlys
- Holt, Dennis A
- Roethke, Theresa
- Hong, Xuan
- Reid, Robert A
- Gampe, Robert
- Zhang, Hong
- Diaz, Elsie
- Rendina, Alan R
- Quinn, Amy M
- Willette, Bob
Publication details: ACS medicinal chemistry letters Jul 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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13.
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Improving the developability profile of pyrrolidine progesterone receptor partial agonists. [electronic resource] by
- Kallander, Lara S
- Washburn, David G
- Hoang, Tram H
- Frazee, James S
- Stoy, Patrick
- Johnson, Latisha
- Lu, Qing
- Hammond, Marlys
- Barton, Linda S
- Patterson, Jaclyn R
- Azzarano, Leonard M
- Nagilla, Rakesh
- Madauss, Kevin P
- Williams, Shawn P
- Stewart, Eugene L
- Duraiswami, Chaya
- Grygielko, Eugene T
- Xu, Xiaoping
- Laping, Nicholas J
- Bray, Jeffrey D
- Thompson, Scott K
Producer: 20100506
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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14.
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Histone deacetylase 3 coordinates commensal-bacteria-dependent intestinal homeostasis. [electronic resource] by
- Alenghat, Theresa
- Osborne, Lisa C
- Saenz, Steven A
- Kobuley, Dmytro
- Ziegler, Carly G K
- Mullican, Shannon E
- Choi, Inchan
- Grunberg, Stephanie
- Sinha, Rohini
- Wynosky-Dolfi, Meghan
- Snyder, Annelise
- Giacomin, Paul R
- Joyce, Karen L
- Hoang, Tram B
- Bewtra, Meenakshi
- Brodsky, Igor E
- Sonnenberg, Gregory F
- Bushman, Frederic D
- Won, Kyoung-Jae
- Lazar, Mitchell A
- Artis, David
Producer: 20131227
In:
Nature vol. 504
Availability: No items available.
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