Results
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Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors. [electronic resource] by
- Sutton, James C
- Bolton, Scott A
- Davis, Malcolm E
- Hartl, Karen S
- Jacobson, Bruce
- Mathur, Arvind
- Ogletree, Martin L
- Slusarchyk, William A
- Zahler, Robert
- Seiler, Steven M
- Bisacchi, Gregory S
Producer: 20041222
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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4.
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Synthesis of potent and highly selective nonguanidine azetidinone inhibitors of human tryptase. [electronic resource] by
- Bisacchi, Gregory S
- Slusarchyk, William A
- Bolton, Scott A
- Hartl, Karen S
- Jacobs, Glenn
- Mathur, Arvind
- Meng, Wei
- Ogletree, Martin L
- Pi, Zulan
- Sutton, James C
- Treuner, Uwe
- Zahler, Robert
- Zhao, Guohua
- Seiler, Steven M
Producer: 20041222
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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5.
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Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors. [electronic resource] by
- Sutton, James C
- Bolton, Scott A
- Hartl, Karen S
- Huang, Ming-Hsing
- Jacobs, Glenn
- Meng, Wei
- Ogletree, Martin L
- Pi, Zulan
- Schumacher, William A
- Seiler, Steven M
- Slusarchyk, William A
- Treuner, Uwe
- Zahler, Robert
- Zhao, Guohua
- Bisacchi, Gregory S
Producer: 20030318
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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6.
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Synthesis of potent and highly selective inhibitors of human tryptase. [electronic resource] by
- Slusarchyk, William A
- Bolton, Scott A
- Hartl, Karen S
- Huang, Ming-Hsing
- Jacobs, Glenn
- Meng, Wei
- Ogletree, Martin L
- Pi, Zulan
- Schumacher, William A
- Seiler, Steven M
- Sutton, James C
- Treuner, Uwe
- Zahler, Robert
- Zhao, Guohua
- Bisacchi, Gregory S
Producer: 20030318
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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7.
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Design, structure-activity relationships, X-ray crystal structure, and energetic contributions of a critical P1 pharmacophore: 3-chloroindole-7-yl-based factor Xa inhibitors. [electronic resource] by
- Shi, Yan
- Sitkoff, Doree
- Zhang, Jing
- Klei, Herbert E
- Kish, Kevin
- Liu, Eddie C-K
- Hartl, Karen S
- Seiler, Steve M
- Chang, Ming
- Huang, Christine
- Youssef, Sonia
- Steinbacher, Thomas E
- Schumacher, William A
- Grazier, Nyeemah
- Pudzianowski, Andrew
- Apedo, Atsu
- Discenza, Lorell
- Yanchunas, Joseph
- Stein, Philip D
- Atwal, Karnail S
Producer: 20090403
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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8.
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Cyanoguanidine-based lactam derivatives as a novel class of orally bioavailable factor Xa inhibitors. [electronic resource] by
- Shi, Yan
- Zhang, Jing
- Shi, Mengxiao
- O'Connor, Stephen P
- Bisaha, Sharon N
- Li, Chi
- Sitkoff, Doree
- Pudzianowski, Andrew T
- Chong, Saeho
- Klei, Herbert E
- Kish, Kevin
- Yanchunas, Joseph
- Liu, Eddie C-K
- Hartl, Karen S
- Seiler, Steve M
- Steinbacher, Thomas E
- Schumacher, William A
- Atwal, Karnail S
- Stein, Philip D
Producer: 20091207
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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9.
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Discovery of nonbenzamidine factor VIIa inhibitors using a biaryl acid scaffold. [electronic resource] by
- Bolton, Scott A
- Sutton, James C
- Anumula, Rushith
- Bisacchi, Gregory S
- Jacobson, Bruce
- Slusarchyk, William A
- Treuner, Uwe D
- Wu, Shung C
- Zhao, Guohua
- Pi, Zulan
- Sheriff, Steven
- Smirk, Rebecca A
- Bisaha, Sharon
- Cheney, Daniel L
- Wei, Anzhi
- Schumacher, William A
- Hartl, Karen S
- Liu, Eddie
- Zahler, Robert
- Seiler, Steven M
Producer: 20140331
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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10.
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Aroylguanidine-based factor Xa inhibitors: the discovery of BMS-344577. [electronic resource] by
- Shi, Yan
- Li, Chi
- O'Connor, Stephen P
- Zhang, Jing
- Shi, Mengxiao
- Bisaha, Sharon N
- Wang, Ying
- Sitkoff, Doree
- Pudzianowski, Andrew T
- Huang, Christine
- Klei, Herbert E
- Kish, Kevin
- Yanchunas, Joseph
- Liu, Eddie C-K
- Hartl, Karen S
- Seiler, Steve M
- Steinbacher, Thomas E
- Schumacher, William A
- Atwal, Karnail S
- Stein, Philip D
Producer: 20100209
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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11.
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Ketene aminal-based lactam derivatives as a novel class of orally active FXa inhibitors. [electronic resource] by
- Shi, Yan
- Zhang, Jing
- Stein, Philip D
- Shi, Mengxiao
- O'Connor, Stephen P
- Bisaha, Sharon N
- Li, Chi
- Atwal, Karnail S
- Bisacchi, Gregory S
- Sitkoff, Doree
- Pudzianowski, Andrew T
- Liu, Eddie C
- Hartl, Karen S
- Seiler, Steven M
- Youssef, Sonia
- Steinbacher, Thomas E
- Schumacher, William A
- Rendina, Alan R
- Bozarth, Jeffrey M
- Peterson, Tara L
- Zhang, Ge
- Zahler, Robert
Producer: 20060627
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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12.
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Discovery of Potent Protease-Activated Receptor 4 Antagonists with in Vivo Antithrombotic Efficacy. [electronic resource] by
- Miller, Michael M
- Banville, Jacques
- Friends, Todd J
- Gagnon, Mark
- Hangeland, Jon J
- Lavallée, Jean-François
- Martel, Alain
- O'Grady, Harold
- Rémillard, Roger
- Ruediger, Edward
- Tremblay, François
- Posy, Shana L
- Allegretto, Nick J
- Guarino, Victor R
- Harden, David G
- Harper, Timothy W
- Hartl, Karen
- Josephs, Jonathan
- Malmstrom, Sarah
- Watson, Carol
- Yang, Yanou
- Zhang, Ge
- Wong, Pancras
- Yang, Jing
- Bouvier, Michel
- Seiffert, Dietmar A
- Wexler, Ruth R
- Lawrence, R Michael
- Priestley, E Scott
- Marinier, Anne
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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