Design and Synthesis of Soluble and Cell-Permeable PI3Kδ Inhibitors for Long-Acting Inhaled Administration. [electronic resource]
Producer: 20170811Description: 5057-5071 p. digitalISSN:- 1520-4804
- Administration, Inhalation
- Animals
- Biological Availability
- Chemistry Techniques, Synthetic
- Drug Design
- Drug Evaluation, Preclinical -- methods
- Enzyme Inhibitors -- administration & dosage
- Half-Life
- Isoenzymes -- antagonists & inhibitors
- Mice, Transgenic
- Permeability
- Phosphoinositide-3 Kinase Inhibitors
- Rats
- Solubility
- Structure-Activity Relationship
- Thiazoles -- chemistry
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Publication Type: Journal Article
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