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Identification of triazinoindol-benzimidazolones as nanomolar inhibitors of the Mycobacterium tuberculosis enzyme TDP-6-deoxy-d-xylo-4-hexopyranosid-4-ulose 3,5-epimerase (RmlC). [electronic resource] by
- Sivendran, Sharmila
- Jones, Victoria
- Sun, Dianqing
- Wang, Yi
- Grzegorzewicz, Anna E
- Scherman, Michael S
- Napper, Andrew D
- McCammon, J Andrew
- Lee, Richard E
- Diamond, Scott L
- McNeil, Michael
Producer: 20100427
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
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Novel insights into the mechanism of inhibition of MmpL3, a target of multiple pharmacophores in Mycobacterium tuberculosis. [electronic resource] by
- Li, Wei
- Upadhyay, Ashutosh
- Fontes, Fabio L
- North, E Jeffrey
- Wang, Yuehong
- Crans, Debbie C
- Grzegorzewicz, Anna E
- Jones, Victoria
- Franzblau, Scott G
- Lee, Richard E
- Crick, Dean C
- Jackson, Mary
Producer: 20150803
In:
Antimicrobial agents and chemotherapy vol. 58
Availability: No items available.
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9.
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Covalent modification of the [electronic resource] by
- Grzegorzewicz, Anna E
- Eynard, Nathalie
- Quémard, Annaïk
- North, E Jeffrey
- Margolis, Alyssa
- Lindenberger, Jared J
- Jones, Victoria
- Korduláková, Jana
- Brennan, Patrick J
- Lee, Richard E
- Ronning, Donald R
- McNeil, Michael R
- Jackson, Mary
Publication details: ACS infectious diseases Feb 2015
In:
ACS infectious diseases vol. 1
Availability: No items available.
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Screening a library of 1600 adamantyl ureas for anti-Mycobacterium tuberculosis activity in vitro and for better physical chemical properties for bioavailability. [electronic resource] by
- Scherman, Michael S
- North, Elton J
- Jones, Victoria
- Hess, Tamara N
- Grzegorzewicz, Anna E
- Kasagami, Takeo
- Kim, In-Hae
- Merzlikin, Oleg
- Lenaerts, Anne J
- Lee, Richard E
- Jackson, Mary
- Morisseau, Christophe
- McNeil, Michael R
Producer: 20120810
In:
Bioorganic & medicinal chemistry vol. 20
Availability: No items available.
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Inhibition of mycolic acid transport across the Mycobacterium tuberculosis plasma membrane. [electronic resource] by
- Grzegorzewicz, Anna E
- Pham, Ha
- Gundi, Vijay A K B
- Scherman, Michael S
- North, Elton J
- Hess, Tamara
- Jones, Victoria
- Gruppo, Veronica
- Born, Sarah E M
- Korduláková, Jana
- Chavadi, Sivagami Sundaram
- Morisseau, Christophe
- Lenaerts, Anne J
- Lee, Richard E
- McNeil, Michael R
- Jackson, Mary
Producer: 20120521
In:
Nature chemical biology vol. 8
Availability: No items available.
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Assembling of the Mycobacterium tuberculosis Cell Wall Core. [electronic resource] by
- Grzegorzewicz, Anna E
- de Sousa-d'Auria, Célia
- McNeil, Michael R
- Huc-Claustre, Emilie
- Jones, Victoria
- Petit, Cécile
- Angala, Shiva Kumar
- Zemanová, Júlia
- Wang, Qinglan
- Belardinelli, Juan Manuel
- Gao, Qian
- Ishizaki, Yoshimasa
- Mikušová, Katarína
- Brennan, Patrick J
- Ronning, Donald R
- Chami, Mohamed
- Houssin, Christine
- Jackson, Mary
Producer: 20170512
In:
The Journal of biological chemistry vol. 291
Availability: No items available.
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13.
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A common mechanism of inhibition of the Mycobacterium tuberculosis mycolic acid biosynthetic pathway by isoxyl and thiacetazone. [electronic resource] by
- Grzegorzewicz, Anna E
- Korduláková, Jana
- Jones, Victoria
- Born, Sarah E M
- Belardinelli, Juan M
- Vaquié, Adrien
- Gundi, Vijay A K B
- Madacki, Jan
- Slama, Nawel
- Laval, Françoise
- Vaubourgeix, Julien
- Crew, Rebecca M
- Gicquel, Brigitte
- Daffé, Mamadou
- Morbidoni, Hector R
- Brennan, Patrick J
- Quémard, Annaik
- McNeil, Michael R
- Jackson, Mary
Producer: 20130131
In:
The Journal of biological chemistry vol. 287
Availability: No items available.
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