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A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies. [electronic resource] by
- Griglio, Alessia
- Torre, Enza
- Serafini, Marta
- Bianchi, Alice
- Schmid, Roberta
- Coda Zabetta, Giulia
- Massarotti, Alberto
- Sorba, Giovanni
- Pirali, Tracey
- Fallarini, Silvia
Producer: 20181008
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders. [electronic resource] by
- Serafini, Marta
- Griglio, Alessia
- Aprile, Silvio
- Seiti, Fabio
- Travelli, Cristina
- Pattarino, Franco
- Grosa, Giorgio
- Sorba, Giovanni
- Genazzani, Armando A
- Gonzalez-Rodriguez, Sara
- Butron, Laura
- Devesa, Isabel
- Fernandez-Carvajal, Asia
- Pirali, Tracey
- Ferrer-Montiel, Antonio
Producer: 20190603
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to [electronic resource] by
- Serafini, Marta
- Torre, Enza
- Aprile, Silvio
- Grosso, Erika Del
- Gesù, Alessandro
- Griglio, Alessia
- Colombo, Giorgia
- Travelli, Cristina
- Paiella, Salvatore
- Adamo, Annalisa
- Orecchini, Elena
- Coletti, Alice
- Pallotta, Maria Teresa
- Ugel, Stefano
- Massarotti, Alberto
- Pirali, Tracey
- Fallarini, Silvia
Producer: 20200902
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs. [electronic resource] by
- Pirali, Tracey
- Ciraolo, Elisa
- Aprile, Silvio
- Massarotti, Alberto
- Berndt, Alex
- Griglio, Alessia
- Serafini, Marta
- Mercalli, Valentina
- Landoni, Clarissa
- Campa, Carlo Cosimo
- Margaria, Jean Piero
- Silva, Rangel L
- Grosa, Giorgio
- Sorba, Giovanni
- Williams, Roger
- Hirsch, Emilio
- Tron, Gian Cesare
Producer: 20171009
In:
ChemMedChem vol. 12
Availability: No items available.
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Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis. [electronic resource] by
- Riva, Beatrice
- Griglio, Alessia
- Serafini, Marta
- Cordero-Sanchez, Celia
- Aprile, Silvio
- Di Paola, Rosanna
- Gugliandolo, Enrico
- Alansary, Dalia
- Biocotino, Isabella
- Lim, Dmitry
- Grosa, Giorgio
- Galli, Ubaldina
- Niemeyer, Barbara
- Sorba, Giovanni
- Canonico, Pier Luigi
- Cuzzocrea, Salvatore
- Genazzani, Armando A
- Pirali, Tracey
Producer: 20190919
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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