Results
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2.
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Discovery of a potent class I selective ketone histone deacetylase inhibitor with antitumor activity in vivo and optimized pharmacokinetic properties. [electronic resource] by
- Kinzel, Olaf
- Llauger-Bufi, Laura
- Pescatore, Giovanna
- Rowley, Michael
- Schultz-Fademrecht, Carsten
- Monteagudo, Edith
- Fonsi, Massimiliano
- Gonzalez Paz, Odalys
- Fiore, Fabrizio
- Steinkühler, Christian
- Jones, Philip
Producer: 20090701
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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3.
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SAR and pharmacokinetic studies on phenethylamide inhibitors of the hepatitis C virus NS3/NS4A serine protease. [electronic resource] by
- Malancona, Savina
- Colarusso, Stefania
- Ontoria, Jesus M
- Marchetti, Antonella
- Poma, Marco
- Stansfield, Ian
- Laufer, Ralph
- Di Marco, Annalise
- Taliani, Marina
- Verdirame, Maria
- Gonzalez-Paz, Odalys
- Matassa, Victor G
- Narjes, Frank
Producer: 20050209
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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4.
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A structure-guided approach to an orthogonal estrogen-receptor-based gene switch activated by ligands suitable for in vivo studies. [electronic resource] by
- Kinzel, Olaf
- Fattori, Daniela
- Muraglia, Ester
- Gallinari, Paola
- Nardi, Maria Chiara
- Paolini, Chantal
- Roscilli, Giuseppe
- Toniatti, Carlo
- Gonzalez Paz, Odalys
- Laufer, Ralph
- Lahm, Armin
- Tramontano, Anna
- Cortese, Riccardo
- De Francesco, Raffaele
- Ciliberto, Gennaro
- Koch, Uwe
Producer: 20061016
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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5.
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Cyclic phosphoramidates as prodrugs of 2'-C-methylcytidine. [electronic resource] by
- Meppen, Malte
- Pacini, Barbara
- Bazzo, Renzo
- Koch, Uwe
- Leone, Joseph F
- Koeplinger, Kenneth A
- Rowley, Michael
- Altamura, Sergio
- Di Marco, Annalise
- Fiore, Fabrizio
- Giuliano, Claudio
- Gonzalez-Paz, Odalys
- Laufer, Ralph
- Pucci, Vincenzo
- Narjes, Frank
- Gardelli, Cristina
Producer: 20091014
In:
European journal of medicinal chemistry vol. 44
Availability: No items available.
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6.
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Establishment of an in Vitro Human Blood-Brain Barrier Model Derived from Induced Pluripotent Stem Cells and Comparison to a Porcine Cell-Based System. [electronic resource] by
- Di Marco, Annalise
- Vignone, Domenico
- Gonzalez Paz, Odalys
- Fini, Ivan
- Battista, Maria Rosaria
- Cellucci, Antonella
- Bracacel, Elena
- Auciello, Giulio
- Veneziano, Maria
- Khetarpal, Vinod
- Rose, Mark
- Rosa, Alessandro
- Gloaguen, Isabelle
- Monteagudo, Edith
- Herbst, Todd
- Dominguez, Celia
- Muñoz-Sanjuán, Ignacio
Producer: 20210305
In:
Cells vol. 9
Availability: No items available.
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7.
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Construction of an rtTA2(s)-m2/tts(kid)-based transcription regulatory switch that displays no basal activity, good inducibility, and high responsiveness to doxycycline in mice and non-human primates. [electronic resource] by
- Lamartina, Stefania
- Silvi, Luisa
- Roscilli, Giuseppe
- Casimiro, Danilo
- Simon, Adam J
- Davies, Mary-Ellen
- Shiver, John W
- Rinaudo, Cira Daniela
- Zampaglione, Immacolata
- Fattori, Elena
- Colloca, Stefano
- Gonzalez Paz, Odalys
- Laufer, Ralph
- Bujard, Hermann
- Cortese, Riccardo
- Ciliberto, Gennaro
- Toniatti, Carlo
Producer: 20030911
In:
Molecular therapy : the journal of the American Society of Gene Therapy vol. 7
Availability: No items available.
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8.
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Design and synthesis of bicyclic pyrimidinones as potent and orally bioavailable HIV-1 integrase inhibitors. [electronic resource] by
- Muraglia, Ester
- Kinzel, Olaf
- Gardelli, Cristina
- Crescenzi, Benedetta
- Donghi, Monica
- Ferrara, Marco
- Nizi, Emanuela
- Orvieto, Federica
- Pescatore, Giovanna
- Laufer, Ralph
- Gonzalez-Paz, Odalys
- Di Marco, Annalise
- Fiore, Fabrizio
- Monteagudo, Edith
- Fonsi, Massimiliano
- Felock, Peter J
- Rowley, Michael
- Summa, Vincenzo
Producer: 20080519
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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9.
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Application of an in Vitro Blood-Brain Barrier Model in the Selection of Experimental Drug Candidates for the Treatment of Huntington's Disease. [electronic resource] by
- Di Marco, Annalise
- Gonzalez Paz, Odalys
- Fini, Ivan
- Vignone, Domenico
- Cellucci, Antonella
- Battista, Maria Rosaria
- Auciello, Giulio
- Orsatti, Laura
- Zini, Matteo
- Monteagudo, Edith
- Khetarpal, Vinod
- Rose, Mark
- Dominguez, Celia
- Herbst, Todd
- Toledo-Sherman, Leticia
- Summa, Vincenzo
- Muñoz-Sanjuán, Ignacio
Producer: 20200310
In:
Molecular pharmaceutics vol. 16
Availability: No items available.
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10.
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Dihydroxypyrimidine-4-carboxamides as novel potent and selective HIV integrase inhibitors. [electronic resource] by
- Pace, Paola
- Di Francesco, M Emilia
- Gardelli, Cristina
- Harper, Steven
- Muraglia, Ester
- Nizi, Emanuela
- Orvieto, Federica
- Petrocchi, Alessia
- Poma, Marco
- Rowley, Michael
- Scarpelli, Rita
- Laufer, Ralph
- Gonzalez Paz, Odalys
- Monteagudo, Edith
- Bonelli, Fabio
- Hazuda, Daria
- Stillmock, Kara A
- Summa, Vincenzo
Producer: 20070626
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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11.
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Discovery of raltegravir, a potent, selective orally bioavailable HIV-integrase inhibitor for the treatment of HIV-AIDS infection. [electronic resource] by
- Summa, Vincenzo
- Petrocchi, Alessia
- Bonelli, Fabio
- Crescenzi, Benedetta
- Donghi, Monica
- Ferrara, Marco
- Fiore, Fabrizio
- Gardelli, Cristina
- Gonzalez Paz, Odalys
- Hazuda, Daria J
- Jones, Philip
- Kinzel, Olaf
- Laufer, Ralph
- Monteagudo, Edith
- Muraglia, Ester
- Nizi, Emanuela
- Orvieto, Federica
- Pace, Paola
- Pescatore, Giovanna
- Scarpelli, Rita
- Stillmock, Kara
- Witmer, Marc V
- Rowley, Michael
Producer: 20081009
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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