Results
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1.
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Discovery of AC710, a Globally Selective Inhibitor of Platelet-Derived Growth Factor Receptor-Family Kinases. [electronic resource] by
- Liu, Gang
- Campbell, Brian T
- Holladay, Mark W
- Ford Pulido, Julia M
- Hua, Helen
- Gitnick, Dana
- Gardner, Michael F
- James, Joyce
- Breider, Mike A
- Brigham, Daniel
- Belli, Barbara
- Armstrong, Robert C
- Treiber, Daniel K
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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2.
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Discovery and optimization of a highly efficacious class of 5-aryl-2-aminopyridines as FMS-like tyrosine kinase 3 (FLT3) inhibitors. [electronic resource] by
- Liu, Gang
- Abraham, Sunny
- Liu, Xing
- Xu, Shimin
- Rooks, Allison M
- Nepomuceno, Ron
- Dao, Alan
- Brigham, Daniel
- Gitnick, Dana
- Insko, Darren E
- Gardner, Michael F
- Zarrinkar, Patrick P
- Christopher, Ron
- Belli, Barbara
- Armstrong, Robert C
- Holladay, Mark W
Producer: 20160518
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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3.
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Novel series of pyrrolotriazine analogs as highly potent pan-Aurora kinase inhibitors. [electronic resource] by
- Abraham, Sunny
- Hadd, Michael J
- Tran, Lan
- Vickers, Troy
- Sindac, Janice
- Milanov, Zdravko V
- Holladay, Mark W
- Bhagwat, Shripad S
- Hua, Helen
- Ford Pulido, Julia M
- Cramer, Merryl D
- Gitnick, Dana
- James, Joyce
- Dao, Alan
- Belli, Barbara
- Armstrong, Robert C
- Treiber, Daniel K
- Liu, Gang
Producer: 20111219
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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4.
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4-Quinazolinyloxy-diaryl ureas as novel BRAFV600E inhibitors. [electronic resource] by
- Holladay, Mark W
- Campbell, Brian T
- Rowbottom, Martin W
- Chao, Qi
- Sprankle, Kelly G
- Lai, Andiliy G
- Abraham, Sunny
- Setti, Eduardo
- Faraoni, Raffaella
- Tran, Lan
- Armstrong, Robert C
- Gunawardane, Ruwanthi N
- Gardner, Michael F
- Cramer, Merryl D
- Gitnick, Dana
- Ator, Mark A
- Dorsey, Bruce D
- Ruggeri, Bruce R
- Williams, Michael
- Bhagwat, Shripad S
- James, Joyce
Producer: 20111219
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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5.
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Discovery of highly potent and selective pan-Aurora kinase inhibitors with enhanced in vivo antitumor therapeutic index. [electronic resource] by
- Liu, Gang
- Abraham, Sunny
- Tran, Lan
- Vickers, Troy D
- Xu, Shimin
- Hadd, Michael J
- Quiambao, Sheena
- Holladay, Mark W
- Hua, Helen
- Ford Pulido, Julia M
- Gunawardane, Ruwanthi N
- Davis, Mindy I
- Eichelberger, Shawn R
- Apuy, Julius L
- Gitnick, Dana
- Gardner, Michael F
- James, Joyce
- Breider, Mike A
- Belli, Barbara
- Armstrong, Robert C
- Treiber, Daniel K
Producer: 20120831
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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6.
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CEP-32496: a novel orally active BRAF(V600E) inhibitor with selective cellular and in vivo antitumor activity. [electronic resource] by
- James, Joyce
- Ruggeri, Bruce
- Armstrong, Robert C
- Rowbottom, Martin W
- Jones-Bolin, Susan
- Gunawardane, Ruwanthi N
- Dobrzanski, Pawel
- Gardner, Michael F
- Zhao, Hugh
- Cramer, Merryl D
- Hunter, Kathryn
- Nepomuceno, Ronald R
- Cheng, Mangeng
- Gitnick, Dana
- Yazdanian, Mehran
- Insko, Darren E
- Ator, Mark A
- Apuy, Julius L
- Faraoni, Raffaella
- Dorsey, Bruce D
- Williams, Michael
- Bhagwat, Shripad S
- Holladay, Mark W
Producer: 20121016
In:
Molecular cancer therapeutics vol. 11
Availability: No items available.
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7.
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Identification of 1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(5-(1,1,1-trifluoro-2-methylpropan-2-yl)isoxazol-3-yl)urea hydrochloride (CEP-32496), a highly potent and orally efficacious inhibitor of V-RAF murine sarcoma viral oncogene homologue B1 (BRAF) V600E. [electronic resource] by
- Rowbottom, Martin W
- Faraoni, Raffaella
- Chao, Qi
- Campbell, Brian T
- Lai, Andiliy G
- Setti, Eduardo
- Ezawa, Maiko
- Sprankle, Kelly G
- Abraham, Sunny
- Tran, Lan
- Struss, Brian
- Gibney, Michael
- Armstrong, Robert C
- Gunawardane, Ruwanthi N
- Nepomuceno, Ronald R
- Valenta, Ianina
- Hua, Helen
- Gardner, Michael F
- Cramer, Merryl D
- Gitnick, Dana
- Insko, Darren E
- Apuy, Julius L
- Jones-Bolin, Susan
- Ghose, Arup K
- Herbertz, Torsten
- Ator, Mark A
- Dorsey, Bruce D
- Ruggeri, Bruce
- Williams, Michael
- Bhagwat, Shripad
- James, Joyce
- Holladay, Mark W
Producer: 20120423
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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