An orally effective dihydropyrimidone (DHPM) analogue induces apoptosis-like cell death in clinical isolates of Leishmania donovani overexpressing pteridine reductase 1. [electronic resource]
Producer: 20091117Description: 1317-25 p. digitalISSN:- 1432-1955
- Animals
- Annexin A5 -- pharmacology
- Antiprotozoal Agents -- chemistry
- Apoptosis
- Cell Death
- Cell Survival
- Cricetinae
- DNA Fragmentation -- drug effects
- Drug Evaluation, Preclinical -- methods
- Indicators and Reagents -- pharmacology
- Leishmania donovani -- drug effects
- Leishmaniasis, Visceral -- parasitology
- Membrane Potential, Mitochondrial -- drug effects
- Oxidoreductases -- biosynthesis
- Propidium -- pharmacology
- Pyrimidinones -- chemistry
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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