Results
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1.
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Discovery of 4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]pyridin-2-yl}-N-(tetrahydro-2H- pyran-4-yl)benzamide (GW788388): a potent, selective, and orally active transforming growth factor-beta type I receptor inhibitor. [electronic resource] by
- Gellibert, Françoise
- de Gouville, Anne-Charlotte
- Woolven, James
- Mathews, Neil
- Nguyen, Van-Loc
- Bertho-Ruault, Cécile
- Patikis, Angela
- Grygielko, Eugene T
- Laping, Nicholas J
- Huet, Stéphane
Producer: 20060502
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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2.
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Inhibition of ALK5 signaling induces physeal dysplasia in rats. [electronic resource] by
- Frazier, Kendall
- Thomas, Roberta
- Scicchitano, Marshall
- Mirabile, Rosanna
- Boyce, Rogely
- Zimmerman, Dawn
- Grygielko, Eugene
- Nold, James
- DeGouville, Anne-Charlotte
- Huet, Stephane
- Laping, Nicholas
- Gellibert, Francoise
Producer: 20070501
In:
Toxicologic pathology vol. 35
Availability: No items available.
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3.
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Inhibition of TGF-beta signaling by an ALK5 inhibitor protects rats from dimethylnitrosamine-induced liver fibrosis. [electronic resource] by
- de Gouville, Anne-Charlotte
- Boullay, Valerie
- Krysa, Gael
- Pilot, Julia
- Brusq, Jean-Marie
- Loriolle, Florence
- Gauthier, Jean-Michel
- Papworth, Stephen A
- Laroze, Alain
- Gellibert, Françoise
- Huet, Stephane
Producer: 20050823
In:
British journal of pharmacology vol. 145
Availability: No items available.
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4.
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Naphthyridines as novel BET family bromodomain inhibitors. [electronic resource] by
- Mirguet, Olivier
- Lamotte, Yann
- Chung, Chun-Wa
- Bamborough, Paul
- Delannée, Delphine
- Bouillot, Anne
- Gellibert, Françoise
- Krysa, Gael
- Lewis, Antonia
- Witherington, Jason
- Huet, Pascal
- Dudit, Yann
- Trottet, Lionel
- Nicodeme, Edwige
Producer: 20141111
In:
ChemMedChem vol. 9
Availability: No items available.
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5.
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Identification of 1,5-naphthyridine derivatives as a novel series of potent and selective TGF-beta type I receptor inhibitors. [electronic resource] by
- Gellibert, Françoise
- Woolven, James
- Fouchet, Marie-Hélène
- Mathews, Neil
- Goodland, Helen
- Lovegrove, Victoria
- Laroze, Alain
- Nguyen, Van-Loc
- Sautet, Stéphane
- Wang, Ruolan
- Janson, Cheryl
- Smith, Ward
- Krysa, Gaël
- Boullay, Valérie
- De Gouville, Anne-Charlotte
- Huet, Stéphane
- Hartley, David
Producer: 20040924
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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6.
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From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151. [electronic resource] by
- Mirguet, Olivier
- Lamotte, Yann
- Donche, Frédéric
- Toum, Jérôme
- Gellibert, Françoise
- Bouillot, Anne
- Gosmini, Romain
- Nguyen, Van-Loc
- Delannée, Delphine
- Seal, Jonathan
- Blandel, Florence
- Boullay, Anne-Bénédicte
- Boursier, Eric
- Martin, Sandrine
- Brusq, Jean-Marie
- Krysa, Gael
- Riou, Alizon
- Tellier, Rémi
- Costaz, Agnès
- Huet, Pascal
- Dudit, Yann
- Trottet, Lionel
- Kirilovsky, Jorge
- Nicodeme, Edwige
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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7.
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Identification of a novel series of BET family bromodomain inhibitors: binding mode and profile of I-BET151 (GSK1210151A). [electronic resource] by
- Seal, Jonathan
- Lamotte, Yann
- Donche, Frédéric
- Bouillot, Anne
- Mirguet, Olivier
- Gellibert, Françoise
- Nicodeme, Edwige
- Krysa, Gael
- Kirilovsky, Jorge
- Beinke, Soren
- McCleary, Scott
- Rioja, Inma
- Bamborough, Paul
- Chung, Chun-Wa
- Gordon, Laurie
- Lewis, Toni
- Walker, Ann L
- Cutler, Leanne
- Lugo, David
- Wilson, David M
- Witherington, Jason
- Lee, Kevin
- Prinjha, Rab K
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
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8.
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Comparison of soluble guanylate cyclase stimulators and activators in models of cardiovascular disease associated with oxidative stress. [electronic resource] by
- Costell, Melissa H
- Ancellin, Nicolas
- Bernard, Roberta E
- Zhao, Shufang
- Upson, John J
- Morgan, Lisa A
- Maniscalco, Kristeen
- Olzinski, Alan R
- Ballard, Victoria L T
- Herry, Kenny
- Grondin, Pascal
- Dodic, Nerina
- Mirguet, Olivier
- Bouillot, Anne
- Gellibert, Francoise
- Coatney, Robert W
- Lepore, John J
- Jucker, Beat M
- Jolivette, Larry J
- Willette, Robert N
- Schnackenberg, Christine G
- Behm, David J
Producer: 20121002
In:
Frontiers in pharmacology vol. 3
Availability: No items available.
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9.
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Substituted 2-[(4-aminomethyl)phenoxy]-2-methylpropionic acid PPARalpha agonists. 1. Discovery of a novel series of potent HDLc raising agents. [electronic resource] by
- Sierra, Michael L
- Beneton, Véronique
- Boullay, Anne-Bénédict
- Boyer, Thierry
- Brewster, Andrew G
- Donche, Frédéric
- Forest, Marie-Claire
- Fouchet, Marie-Hélène
- Gellibert, Françoise J
- Grillot, Didier A
- Lambert, Millard H
- Laroze, Alain
- Le Grumelec, Christelle
- Linget, Jean Michel
- Montana, Valerie G
- Nguyen, Van-Loc
- Nicodème, Edwige
- Patel, Vipul
- Penfornis, Annie
- Pineau, Olivier
- Pohin, Danig
- Potvain, Florent
- Poulain, Géraldine
- Ruault, Cécile Bertho
- Saunders, Michael
- Toum, Jérôme
- Xu, H Eric
- Xu, Robert X
- Pianetti, Pascal M
Producer: 20070327
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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10.
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Discovery and characterization of small molecule inhibitors of the BET family bromodomains. [electronic resource] by
- Chung, Chun-Wa
- Coste, Herve
- White, Julia H
- Mirguet, Olivier
- Wilde, Jonathan
- Gosmini, Romain L
- Delves, Chris
- Magny, Sylvie M
- Woodward, Robert
- Hughes, Stephen A
- Boursier, Eric V
- Flynn, Helen
- Bouillot, Anne M
- Bamborough, Paul
- Brusq, Jean-Marie G
- Gellibert, Francoise J
- Jones, Emma J
- Riou, Alizon M
- Homes, Paul
- Martin, Sandrine L
- Uings, Iain J
- Toum, Jerome
- Clement, Catherine A
- Boullay, Anne-Benedicte
- Grimley, Rachel L
- Blandel, Florence M
- Prinjha, Rab K
- Lee, Kevin
- Kirilovsky, Jorge
- Nicodeme, Edwige
Producer: 20110817
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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